Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50022143
LigandPNGBDBM50511374(CHEMBL4522276)
Affinity DataIC50: 43nMAssay Description:Inhibition of FLAG-tagged full-length recombinant wild-type human CDKL2 expressed in HeLa cells using MBP as substrate incubated for 30 mins in prese...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50511374(CHEMBL4522276)
Affinity DataIC50: 160nMAssay Description:Inhibition of AAK1 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50511374(CHEMBL4522276)
Affinity DataIC50: 230nMAssay Description:Inhibition of CDKL2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50511374(CHEMBL4522276)
Affinity DataIC50: 320nMAssay Description:Inhibition of BMP2K (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50511399(CHEMBL4542463)
Affinity DataIC50: 450nMAssay Description:Inhibition of CDKL2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50511374(CHEMBL4522276)
Affinity DataIC50: 460nMAssay Description:Displacement of tracer K10 from N-terminal NLuc-fused full-length CDKL2 (unknown origin) expressed in HEK293 cells by NanoBRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50511399(CHEMBL4542463)
Affinity DataIC50: 700nMAssay Description:Displacement of tracer K10 from N-terminal NLuc-fused full-length CDKL2 (unknown origin) expressed in HEK293 cells by NanoBRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50648617(CHEMBL5614135)
Affinity DataIC50: 1.20E+3nMAssay Description:Displacement of tracer K10 from N-terminal NLuc-fused full-length CDKL2 (unknown origin) expressed in HEK293 cells by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50511374(CHEMBL4522276)
Affinity DataIC50: 2.30E+3nMAssay Description:Displacement of tracer K10 from N-terminal NLuc-fused AAK1 (1 to 353 residues)(unknown origin) expressed in HEK293 cells by NanoBRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50511374(CHEMBL4522276)
Affinity DataIC50: 5.70E+3nMAssay Description:Displacement of tracer K10 from N-terminal NLuc-fused BMP2K (1 to 367 residues)(unknown origin) expressed in HEK293 cells by NanoBRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50511397(CHEMBL4452939)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of tracer K10 from N-terminal NLuc-fused full-length CDKL2 (unknown origin) expressed in HEK293 cells by NanoBRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50648620(CHEMBL5612618)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of tracer K10 from N-terminal NLuc-fused full-length CDKL2 (unknown origin) expressed in HEK293 cells by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50648619(CHEMBL5614070)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of tracer K10 from N-terminal NLuc-fused full-length CDKL2 (unknown origin) expressed in HEK293 cells by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50648618(CHEMBL5613154)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of tracer K10 from N-terminal NLuc-fused full-length CDKL2 (unknown origin) expressed in HEK293 cells by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50511374(CHEMBL4522276)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PRP4 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50511374(CHEMBL4522276)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of GRK4 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50511374(CHEMBL4522276)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PIP5K1A (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50511374(CHEMBL4522276)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of MEK5 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetSRSF protein kinase 1(Human)TBA
LigandPNGBDBM50511374(CHEMBL4522276)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of SRPK1 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetSRSF protein kinase 3(Human)TBA
LigandPNGBDBM50511374(CHEMBL4522276)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of SRPK3 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50511374(CHEMBL4522276)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of FLAG-tagged full-length recombinant wild-type human CDKL1 expressed in HeLa cells using MBP as substrate incubated for 30 mins in prese...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCyclin-dependent kinase-like 5(Homo sapiens)TBA
LigandPNGBDBM50511374(CHEMBL4522276)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of FLAG-tagged full-length recombinant wild-type human CDKL5 expressed in HeLa cells using MBP as substrate incubated for 30 mins in prese...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50511374(CHEMBL4522276)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of FLAG-tagged full-length recombinant wild-type human CDKL4 expressed in HeLa cells using MBP as substrate incubated for 30 mins in prese...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50511374(CHEMBL4522276)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of FLAG-tagged full-length recombinant wild-type human CDKL3 expressed in HeLa cells using MBP as substrate incubated for 30 mins in prese...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed