Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50021922
TargetPyruvate kinase PKM(Human)
National Institute of Pharmaceutical Education and Research-Ahmedabad (NIPER-A)

Curated by ChEMBL
LigandPNGBDBM50646189(CHEMBL5590652)
Affinity DataEC50:  0.600nMAssay Description:Activation of PKM2 (unknown origin) by LDH enzyme coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetMitogen-activated protein kinase 14(Human)
National Institute of Pharmaceutical Education and Research-Ahmedabad (NIPER-A)

Curated by ChEMBL
LigandPNGBDBM50646192(CHEMBL5589815)
Affinity DataIC50: 1nMAssay Description:Inhibition of p38alpha (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
National Institute of Pharmaceutical Education and Research-Ahmedabad (NIPER-A)

Curated by ChEMBL
LigandPNGBDBM50646191(CHEMBL5591579)
Affinity DataIC50: 2.70nMAssay Description:Inhibition of human VEGFR2 by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetCyclin-dependent kinase 2(Human)
National Institute of Pharmaceutical Education and Research-Ahmedabad (NIPER-A)

Curated by ChEMBL
LigandPNGBDBM7660(4-[(4-{imidazo[1,2-a]pyridin-3-yl}pyrimidin-2-yl)a...)
Affinity DataIC50: 4nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
National Institute of Pharmaceutical Education and Research-Ahmedabad (NIPER-A)

Curated by ChEMBL
LigandPNGBDBM50119621(CHEMBL3618245)
Affinity DataIC50: 11nMAssay Description:Inhibition of PI3Kalpha (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
National Institute of Pharmaceutical Education and Research-Ahmedabad (NIPER-A)

Curated by ChEMBL
LigandPNGBDBM50119621(CHEMBL3618245)
Affinity DataIC50: 206nMAssay Description:Inhibition of mTOR (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPyruvate kinase PKM(Human)
National Institute of Pharmaceutical Education and Research-Ahmedabad (NIPER-A)

Curated by ChEMBL
LigandPNGBDBM50646190(CHEMBL1090777)
Affinity DataEC50:  241nMAssay Description:Activation of PKM2 (unknown origin) by LDH enzyme coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed