Compile Data Set for Download or QSAR
Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 50022080
TargetSerine-protein kinase ATM(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50647908(CHEMBL5597568)
Affinity DataKi:  0.400nMAssay Description:Binding affinity to ATM (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50647907(CHEMBL5598036)
Affinity DataKi:  1nMAssay Description:Binding affinity to ATM (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50624174(CHEMBL5419324)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of ATM (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50647906(CHEMBL5597825)
Affinity DataKi:  2nMAssay Description:Binding affinity to ATM (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
LigandPNGBDBM50378201(CHEMBL4159350)
Affinity DataIC50: 3nMAssay Description:Inhibition of PI3K alpha (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
LigandPNGBDBM50647911(CHEMBL5596626)
Affinity DataIC50: 4nMAssay Description:Inhibition of PI3Kalpha (unknown origin) using PIP2 as substrate measured after 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
LigandPNGBDBM50647911(CHEMBL5596626)
Affinity DataIC50: 5nMAssay Description:Inhibition of PI3Kgamma (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
LigandPNGBDBM50550657(CHEMBL4792737)
Affinity DataIC50: 5nMAssay Description:Inhibition of PI3K alpha (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50647911(CHEMBL5596626)
Affinity DataIC50: 5nMAssay Description:Inhibition of DNA-PK (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPhosphatidylinositol 3-kinase catalytic subunit type 3(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50647908(CHEMBL5597568)
Affinity DataKi:  6nMAssay Description:Binding affinity to Vps34 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50647905(CHEMBL5598055)
Affinity DataKi:  6nMAssay Description:Binding affinity to ATM (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50647911(CHEMBL5596626)
Affinity DataIC50: 7nMAssay Description:Inhibition of ATM (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
LigandPNGBDBM50647911(CHEMBL5596626)
Affinity DataIC50: 7nMAssay Description:Inhibition of PI3Kdelta (unknown origin) using PIP2 as substrate preincubated for 15 mins followed by substrate addition and measured after 1 hr by H...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPhosphatidylinositol 3-kinase catalytic subunit type 3(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50647905(CHEMBL5598055)
Affinity DataKi:  9nMAssay Description:Binding affinity to Vps34 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
LigandPNGBDBM50647909(CHEMBL5597379)
Affinity DataIC50: 20nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50647911(CHEMBL5596626)
Affinity DataIC50: 20nMAssay Description:Inhibition of mTOR (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetAlpha-1-antitrypsin-related protein(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50647911(CHEMBL5596626)
Affinity DataIC50: 20nMAssay Description:Inhibition of ATR (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPhosphatidylinositol 3-kinase catalytic subunit type 3(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50647907(CHEMBL5598036)
Affinity DataKi:  50nMAssay Description:Binding affinity to Vps34 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
LigandPNGBDBM50647911(CHEMBL5596626)
Affinity DataIC50: 75nMAssay Description:Inhibition of PI3Kbeta (unknown origin) using PIP2 as substrate measured for 1 hr by ADP-glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPhosphatidylinositol 3-kinase catalytic subunit type 3(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50647906(CHEMBL5597825)
Affinity DataKi:  90nMAssay Description:Binding affinity to Vps34 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine-protein kinase ATM(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50647910(CHEMBL5597386)
Affinity DataIC50: 600nMAssay Description:Inhibition of ATM (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50647910(CHEMBL5597386)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of mTOR (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed