Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50015098
TargetBromodomain-containing protein 4(Human)
Maruho Co.

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50254357BDBM50254357(CHEMBL6103057)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of EphB4 autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Maruho Co.

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50254398BDBM50254398(CHEMBL6109028)
Affinity DataIC50: 3.70nMAssay Description:Inhibition of VEGFR2 autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Maruho Co.

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50254356BDBM50254356(CHEMBL6074578)
Affinity DataIC50: 6.30nMAssay Description:Inhibition of ROCK2 assessed as myosin light chain phosphorylation by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Maruho Co.

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50254399BDBM50254399(CHEMBL6092038)
Affinity DataIC50: 8.90nMAssay Description:Inhibition of ROCK2 assessed as myosin light chain phosphorylation by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Maruho Co.

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50254399BDBM50254399(CHEMBL6092038)
Affinity DataIC50: 9.40nMAssay Description:Inhibition of Tie2 autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Maruho Co.

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50254354BDBM50254354(CHEMBL6074546)
Affinity DataIC50: 13nMAssay Description:Inhibition of ROCK2 assessed as myosin light chain phosphorylation by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Maruho Co.

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50254400BDBM50254400(CHEMBL6074576)
Affinity DataIC50: 14nMAssay Description:Antagonist activity at human prostaglandin D2 receptor assessed as inhibition of PGD2-induced receptor activation by cell based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Maruho Co.

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50254355BDBM50254355(CHEMBL6083172)
Affinity DataIC50: 16nMAssay Description:Inhibition of ROCK2 assessed as myosin light chain phosphorylation by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Maruho Co.

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50629953BDBM50629953(CHEMBL5438588)
Affinity DataIC50: 16nMAssay Description:Inhibition of ROCK2 assessed as myosin light chain phosphorylation by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Maruho Co.

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50254352BDBM50254352(CHEMBL6078393)
Affinity DataIC50: 16nMAssay Description:Inhibition of ROCK2 assessed as myosin light chain phosphorylation by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details Article
PubMed
TargetBromodomain-containing protein 3(Human)
Maruho Co.

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50254399BDBM50254399(CHEMBL6092038)
Affinity DataIC50: 19nMAssay Description:Inhibition of ROCK2 assessed as myosin light chain phosphorylation by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details Article
PubMed
TargetBromodomain-containing protein 2(Human)
Maruho Co.

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50254399BDBM50254399(CHEMBL6092038)
Affinity DataIC50: 20nMAssay Description:Inhibition of ROCK2 assessed as myosin light chain phosphorylation by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Maruho Co.

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50254351BDBM50254351(CHEMBL6078336)
Affinity DataIC50: 21nMAssay Description:Inhibition of ROCK2 assessed as myosin light chain phosphorylation by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Maruho Co.

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50254350BDBM50254350(CHEMBL6103008)
Affinity DataIC50: 21nMAssay Description:Inhibition of ROCK2 assessed as myosin light chain phosphorylation by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details Article
PubMed
TargetBromodomain testis-specific protein(Human)
Maruho Co.

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50254399BDBM50254399(CHEMBL6092038)
Affinity DataIC50: 22nMAssay Description:Inhibition of ROCK2 assessed as myosin light chain phosphorylation by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Maruho Co.

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50380682BDBM50380682(CHEMBL2017291 | I-BET151 (16))
Affinity DataIC50: 25nMAssay Description:Inhibition of VEGFR2 autophosphorylation by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Maruho Co.

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50254353BDBM50254353(CHEMBL6078396)
Affinity DataIC50: 38nMAssay Description:Inhibition of ROCK2 assessed as myosin light chain phosphorylation by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Maruho Co.

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50254399BDBM50254399(CHEMBL6092038)
Affinity DataIC50: 114nMAssay Description:Inhibition of ROCK2 assessed as myosin light chain phosphorylation by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details Article
PubMed