Report error Found 75 Enz. Inhib. hit(s) with all data for entry = 50021995
Affinity DataKd: <0.100nMAssay Description:Binding affinity to MDM2 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKd: 2nMAssay Description:Binding affinity to GST-tagged human MDM2 extracted from Escherichia coli BL21 (DE3) assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of MDMX (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of MDMX (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibition of MDM2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of MDM2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 10nMAssay Description:Binding affinity to N-terminal human MDMX (22 to 110 residues) extracted from Escherichia coli BL21 (DE3) assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Inhibition of MDMX (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 20nMAssay Description:Binding affinity to GST-tagged human MDM2 extracted from Escherichia coli BL21 (DE3) assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKd: 20nMAssay Description:Binding affinity to MDMX (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of MDMX (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of MDM2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of MDMX (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 20nMAssay Description:Binding affinity to MDM2 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKd: 20nMAssay Description:Binding affinity to His-tagged MDM2 (1 to 110 residues) (unknown origin) assessed as dissociation constant by MST assayMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of MDM2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of MDMX (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of MDM2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of MDM2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of MDM2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of MDMX (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 41nMAssay Description:Inhibition of MDMX (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:Inhibition of MDMX (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Inhibition of MDMX (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Inhibition of MDM2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 80nMAssay Description:Inhibition of MDMX (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 90nMAssay Description:Inhibition of MDM2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:Inhibition of MDM2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 200nMAssay Description:Binding affinity to MDMX (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibition of MDMX (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 200nMAssay Description:Binding affinity to MDM2 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKd: 300nMAssay Description:Binding affinity to MDM2 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition of MDM2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 600nMAssay Description:Binding affinity to N-terminal human MDMX (22 to 110 residues) extracted from Escherichia coli BL21 (DE3) assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKd: 600nMAssay Description:Binding affinity to N-terminal human MDMX (22 to 110 residues) extracted from Escherichia coli BL21 (DE3) assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKd: 900nMAssay Description:Binding affinity to N-terminal MDM2 (24 to 109 residues) (unknown origin) extracted from Escherichia coli BL21-Gold (DE3) assessed as dissociation co...More data for this Ligand-Target Pair
Affinity DataKd: 1.40E+3nMAssay Description:Binding affinity to N-terminal MDM2 (24 to 109 residues) (unknown origin) extracted from Escherichia coli BL21-Gold (DE3) assessed as dissociation co...More data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of MDMX (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 1.80E+3nMAssay Description:Binding affinity to MDM2 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKd: 2.50E+3nMAssay Description:Binding affinity to MDMX (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKd: 2.70E+3nMAssay Description:Binding affinity to N-terminal MDM2 (24 to 109 residues) (unknown origin) extracted from Escherichia coli BL21-Gold (DE3) assessed as dissociation co...More data for this Ligand-Target Pair
Affinity DataKd: 3.50E+3nMAssay Description:Binding affinity to GST-tagged human MDM2 extracted from Escherichia coli BL21 (DE3) assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKd: 3.50E+3nMAssay Description:Binding affinity to MDMX (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of MDMX (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 4.10E+3nMAssay Description:Binding affinity to N-terminal human MDMX (22 to 110 residues) extracted from Escherichia coli BL21 (DE3) assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKd: 5.00E+3nMAssay Description:Binding affinity to MDMX (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibition of MDMX (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 6.50E+3nMAssay Description:Binding affinity to MDMX (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKd: 6.50E+3nMAssay Description:Binding affinity to N-terminal human MDMX (22 to 110 residues) extracted from Escherichia coli BL21 (DE3) assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKd: 6.70E+3nMAssay Description:Binding affinity to MDM2 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair







3D Structure (crystal)





















