Compile Data Set for Download or QSAR
Report error Found 48 Enz. Inhib. hit(s) with all data for entry = 50022154
LigandPNGBDBM50648689(CHEMBL5612531)
Affinity DataIC50: 3nMAssay Description:Inhibition of PRMT1 (unknown origin) by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50636218(CHEMBL5559689)
Affinity DataIC50: 3nMAssay Description:Inhibition of PRMT1 (unknown origin) by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50648690(CHEMBL5613916)
Affinity DataIC50: 17nMAssay Description:Inhibition of PRMT1 (unknown origin) by fluorescence based analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50009672(AdoHcy | S-[1-(adenin-9-yl)-1,5-dideoxy-beta-D-rib...)
Affinity DataIC50: 550nMAssay Description:Inhibition of PRMT1 (unknown origin) incubated for 30 mins by AlphaLISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50648686(CHEMBL5612079)
Affinity DataIC50: 1.21E+3nMAssay Description:Inhibition of PRMT1 (unknown origin) incubated for 30 mins by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50648705(CHEMBL5613322)
Affinity DataIC50: 1.33E+3nMAssay Description:Inhibition of human PRMT1 using [3H]methylated biotin-labeled peptide as substrate by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50648684(CHEMBL5613456)
Affinity DataIC50: 1.49E+3nMAssay Description:Inhibition of PRMT1 (unknown origin) incubated for 30 mins by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50378739(SINEFUNGIN | jm2c00120, Sinefungin)
Affinity DataIC50: 1.63E+3nMAssay Description:Inhibition of recombinant C-terminal GST-tagged PRMT1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50206427(AMI-1 | 7,7'-carbonylbis(azanediyl)bis(4-hydroxyna...)
Affinity DataIC50: 1.63E+3nMAssay Description:Inhibition of recombinant C-terminal GST-tagged PRMT1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50648698(CHEMBL5614156)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of N-terminal His-tagged human PRMT1 (22 to 361 residues)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50648698(CHEMBL5614156)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of PRMT1 (unknown origin) using Histone H4 as substrate incubated for 1 hr by fluorescence based analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50648713(CHEMBL5613467)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of N-terminal hexa-histidine tagged human recombinant PRMT1 extracted from Escherichia coli BL21 (DE3) incubated for 1 hrs by scintillatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50648688(CHEMBL5612606)
Affinity DataIC50: 2.06E+3nMAssay Description:Inhibition of PRMT1 (unknown origin) incubated for 30 mins by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50648702(CHEMBL5613827)
Affinity DataIC50: 2.51E+3nMAssay Description:Inhibition of human PRMT1 using [3H]methylated biotin-labeled peptide as substrate by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50550091(CHEMBL4648477)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of human recombinant His-tagged PRMT1 extracted from Escherichia coli incubated for 1 hr by Bradford assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50648687(CHEMBL5612674)
Affinity DataIC50: 2.66E+3nMAssay Description:Inhibition of PRMT1 (unknown origin) incubated for 30 mins by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50648699(CHEMBL5612557)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of PRMT1 (unknown origin) using Histone H4 as substrate incubated for 1 hr by fluorescence based analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50648699(CHEMBL5612557)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of N-terminal His-tagged human PRMT1 (22 to 361 residues)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50378739(SINEFUNGIN | jm2c00120, Sinefungin)
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of 6His-tagged human recombinant PRMT1 using Histone H4 as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50648685(CHEMBL5612584)
Affinity DataIC50: 4.14E+3nMAssay Description:Inhibition of PRMT1 (unknown origin) incubated for 30 mins by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50648704(CHEMBL5612710)
Affinity DataIC50: 4.66E+3nMAssay Description:Inhibition of human PRMT1 using [3H]methylated biotin-labeled peptide as substrate by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50648703(CHEMBL5612838)
Affinity DataIC50: 5.36E+3nMAssay Description:Inhibition of human PRMT1 using [3H]methylated biotin-labeled peptide as substrate by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50648691(CHEMBL5613163)
Affinity DataIC50: 7.20E+3nMAssay Description:Inhibition of N-terminal His-tagged human PRMT1 (22 to 361 residues)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50009672(AdoHcy | S-[1-(adenin-9-yl)-1,5-dideoxy-beta-D-rib...)
Affinity DataIC50: 8.30E+3nMAssay Description:Inhibition of PRMT1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50009672(AdoHcy | S-[1-(adenin-9-yl)-1,5-dideoxy-beta-D-rib...)
Affinity DataIC50: 8.39E+3nMAssay Description:Inhibition of 6His-tagged human recombinant PRMT1 using Histone H4 as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50637546(CHEMBL5563346)
Affinity DataIC50: 8.73E+3nMAssay Description:Inhibition of PRMT1 (unknown origin) using Histone H4 as substrate preincubated for 30 mins followed by substrate addition and measured after 60 mins...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50648696(CHEMBL5613658)
Affinity DataIC50: 1.11E+4nMAssay Description:Inhibition of N-terminal His-tagged human PRMT1 (22 to 361 residues)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50648693(CHEMBL5613822)
Affinity DataIC50: 1.16E+4nMAssay Description:Inhibition of N-terminal His-tagged human PRMT1 (22 to 361 residues)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50648692(CHEMBL5613835)
Affinity DataIC50: 1.18E+4nMAssay Description:Inhibition of N-terminal His-tagged human PRMT1 (22 to 361 residues)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50648701(CHEMBL5613919)
Affinity DataIC50: 1.39E+4nMAssay Description:Inhibition of 6His-tagged human recombinant PRMT1 using Histone H4 as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50648712(CHEMBL5613820)
Affinity DataIC50: 1.39E+4nMAssay Description:Inhibition of Histidine-tagged human recombinant PRMT1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50648715(CHEMBL5612198)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of PRMT1 (unknown origin) using Histone H4 as substrate preincubated for 30 mins followed by substrate addition and measured after 60 mins...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50648711(CHEMBL5611982)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of Histidine-tagged human recombinant PRMT1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50648706(CHEMBL5614296)
Affinity DataIC50: 1.85E+4nMAssay Description:Inhibition of PRMT1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50648710(CHEMBL5612942)
Affinity DataIC50: 1.92E+4nMAssay Description:Inhibition of Histidine-tagged human recombinant PRMT1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50648694(CHEMBL1199038)
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibition of N-terminal His-tagged human PRMT1 (22 to 361 residues)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50648695(CHEMBL5612328)
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibition of N-terminal His-tagged human PRMT1 (22 to 361 residues)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50648697(CHEMBL5613423)
Affinity DataIC50: 2.53E+4nMAssay Description:Inhibition of N-terminal His-tagged human PRMT1 (22 to 361 residues)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50648707(CHEMBL5612611)
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of PRMT1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50648709(CHEMBL5612412)
Affinity DataIC50: 2.90E+4nMAssay Description:Inhibition of Histidine-tagged human recombinant PRMT1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM178103(MS023 (Compound 3) | N1-((4-(4-isopropoxyphenyl)-1...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of PRMT1 (unknown origin) by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50648708(CHEMBL5611944)
Affinity DataIC50: 3.04E+4nMAssay Description:Inhibition of PRMT1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50648716(CHEMBL5612247)
Affinity DataIC50: 5.91E+4nMAssay Description:Inhibition of PRMT1 (unknown origin) using Histone H4 as substrate preincubated for 30 mins followed by substrate addition and measured after 60 mins...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50648714(CHEMBL5613541)
Affinity DataIC50: 9.40E+4nMAssay Description:Inhibition of N-terminal hexa-histidine tagged human recombinant PRMT1 extracted from Escherichia coli BL21 (DE3) incubated for 1 hrs by scintillatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50598014(CHEMBL2179350)
Affinity DataIC50: 1.12E+5nMAssay Description:Inhibition of recombinant C-terminal GST-tagged PRMT1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50637542(CHEMBL5531978)
Affinity DataIC50: 2.98E+5nMAssay Description:Inhibition of GST-tagged PRMT1 (unknown origin) extracted from Escherichia coli BL21 incubated for 30 mins by liquid scintillation methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50206427(AMI-1 | 7,7'-carbonylbis(azanediyl)bis(4-hydroxyna...)
Affinity DataIC50: 3.50E+5nMAssay Description:Inhibition of PRMT1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50648700(CHEMBL5613648)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibition of 6His-tagged human recombinant PRMT1 using Histone H4 as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed