Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50022692
TargetIntegrin alpha-V/beta-3(Human)
University of Bradford

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50653145BDBM50653145(CHEMBL6087354)
Affinity DataIC50: 340nMAssay Description:Inhibition of human 11betaHSD1 expressed in CHO cells by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetIntegrin alpha-V/beta-3(Human)
University of Bradford

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50653144BDBM50653144(CHEMBL6108996)
Affinity DataIC50: 600nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetIntegrin alpha-V/beta-3(Human)
University of Bradford

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50653139BDBM50653139(CHEMBL6114896)
Affinity DataIC50: 1.20E+3nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetIntegrin alpha-V/beta-3(Human)
University of Bradford

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50653141BDBM50653141(CHEMBL6102659)
Affinity DataIC50: 1.80E+3nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetIntegrin alpha-V/beta-3(Human)
University of Bradford

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50653143BDBM50653143(CHEMBL6143915)
Affinity DataIC50: 1.80E+3nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetIntegrin alpha-V/beta-3(Human)
University of Bradford

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50653146BDBM50653146(CHEMBL3357753)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of human 11betaHSD1 expressed in CHO cells by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetIntegrin alpha-V/beta-3(Human)
University of Bradford

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50653140BDBM50653140(CHEMBL6134200)
Affinity DataIC50: 3.28E+3nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetIntegrin alpha-V/beta-3(Human)
University of Bradford

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50653136BDBM50653136(CHEMBL6133254)
Affinity DataIC50: 1.15E+4nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetIntegrin alpha-V/beta-3(Human)
University of Bradford

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50653142BDBM50653142(CHEMBL6143260)
Affinity DataIC50: 1.36E+4nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetIntegrin alpha-V/beta-3(Human)
University of Bradford

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50653137BDBM50653137(CHEMBL6078298)
Affinity DataIC50: 2.94E+4nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
TargetIntegrin alpha-V/beta-3(Human)
University of Bradford

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50653138BDBM50653138(CHEMBL6142934)
Affinity DataIC50: 4.95E+4nMAssay Description:Modulation of rat mGlu5 receptor assessed as calcium mobilization by cell based fluorescence assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed