Compile Data Set for Download or QSAR
Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 50022162
TargetIntegrase(Human immunodeficiency virus type 1)
"Sapienza" Universita di Roma

Curated by ChEMBL
LigandPNGBDBM50479082(CHEMBL497501)
Affinity DataIC50: 70nMAssay Description:Inhibition of HIV-1 integrase catalytic activity incubated for 1 hrs in absence of LEDGF/p75 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
"Sapienza" Universita di Roma

Curated by ChEMBL
LigandPNGBDBM50648820(CHEMBL5613927)
Affinity DataIC50: 77nMAssay Description:Inhibition of HIV-1 integrase catalytic activity incubated for 1 hrs in absence of LEDGF/p75 by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
"Sapienza" Universita di Roma

Curated by ChEMBL
LigandPNGBDBM50648816(CHEMBL5613849)
Affinity DataIC50: 181nMAssay Description:Inhibition of HIV-1 integrase catalytic activity incubated for 1 hrs in absence of LEDGF/p75 by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
"Sapienza" Universita di Roma

Curated by ChEMBL
LigandPNGBDBM50648818(CHEMBL5612575)
Affinity DataIC50: 480nMAssay Description:Inhibition of HIV-1 integrase catalytic activity incubated for 1 hrs in absence of LEDGF/p75 by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
"Sapienza" Universita di Roma

Curated by ChEMBL
LigandPNGBDBM50648821(CHEMBL5613097)
Affinity DataIC50: 741nMAssay Description:Inhibition of HIV-1 integrase catalytic activity incubated for 1 hrs in absence of LEDGF/p75 by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
"Sapienza" Universita di Roma

Curated by ChEMBL
LigandPNGBDBM50648819(CHEMBL5613277)
Affinity DataIC50: 782nMAssay Description:Inhibition of HIV-1 integrase catalytic activity incubated for 1 hrs in absence of LEDGF/p75 by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
"Sapienza" Universita di Roma

Curated by ChEMBL
LigandPNGBDBM50648817(CHEMBL5612913)
Affinity DataIC50: 800nMAssay Description:Inhibition of HIV-1 integrase catalytic activity incubated for 1 hrs in absence of LEDGF/p75 by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
"Sapienza" Universita di Roma

Curated by ChEMBL
LigandPNGBDBM50648823(CHEMBL5613833)
Affinity DataEC50: >2.00E+3nMAssay Description:Inhibition of HIV1 integrase activity by measuring multimerization of His-tagged integrase/FLAG-tagged integrase incubated for 3 hrs by fluorescence ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
"Sapienza" Universita di Roma

Curated by ChEMBL
LigandPNGBDBM50486611(CHEMBL2236593)
Affinity DataIC50: 2.34E+3nMAssay Description:Inhibition of HIV-1 integrase catalytic activity incubated for 1 hrs in absence of LEDGF/p75 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
"Sapienza" Universita di Roma

Curated by ChEMBL
LigandPNGBDBM50486621(CHEMBL2236594)
Affinity DataIC50: 3.14E+3nMAssay Description:Inhibition of HIV-1 integrase catalytic activity incubated for 1 hrs in absence of LEDGF/p75 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
"Sapienza" Universita di Roma

Curated by ChEMBL
LigandPNGBDBM50648823(CHEMBL5613833)
Affinity DataIC50: 6.28E+3nMAssay Description:Inhibition of HIV-1 integrase catalytic activity incubated for 1 hrs in absence of LEDGF/p75 by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
"Sapienza" Universita di Roma

Curated by ChEMBL
LigandPNGBDBM50587969(CHEMBL5173288)
Affinity DataIC50: 3.65E+4nMAssay Description:Inhibition of HIV-1 integrase catalytic activity incubated for 1 hrs in absence of LEDGF/p75 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
"Sapienza" Universita di Roma

Curated by ChEMBL
LigandPNGBDBM50587988(CHEMBL5172754)
Affinity DataIC50: 4.19E+4nMAssay Description:Inhibition of HIV-1 integrase catalytic activity incubated for 1 hrs in absence of LEDGF/p75 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
"Sapienza" Universita di Roma

Curated by ChEMBL
LigandPNGBDBM50648822(CHEMBL5613898)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of HIV-1 integrase catalytic activity incubated for 1 hrs in absence of LEDGF/p75 by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
"Sapienza" Universita di Roma

Curated by ChEMBL
LigandPNGBDBM50587963(CHEMBL5171239)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of HIV-1 integrase catalytic activity incubated for 1 hrs in absence of LEDGF/p75 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
"Sapienza" Universita di Roma

Curated by ChEMBL
LigandPNGBDBM50648824(CHEMBL5612322)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of HIV-1 integrase catalytic activity incubated for 1 hrs in absence of LEDGF/p75 by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
"Sapienza" Universita di Roma

Curated by ChEMBL
LigandPNGBDBM50587988(CHEMBL5172754)
Affinity DataEC50: >2.00E+5nMAssay Description:Inhibition of HIV1 integrase activity by measuring multimerization of His-tagged integrase/FLAG-tagged integrase incubated for 3 hrs by fluorescence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
"Sapienza" Universita di Roma

Curated by ChEMBL
LigandPNGBDBM50587969(CHEMBL5173288)
Affinity DataEC50: >2.00E+5nMAssay Description:Inhibition of HIV1 integrase activity by measuring multimerization of His-tagged integrase/FLAG-tagged integrase incubated for 3 hrs by fluorescence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
"Sapienza" Universita di Roma

Curated by ChEMBL
LigandPNGBDBM50648818(CHEMBL5612575)
Affinity DataEC50: >2.00E+5nMAssay Description:Inhibition of HIV1 integrase activity by measuring multimerization of His-tagged integrase/FLAG-tagged integrase incubated for 3 hrs by fluorescence ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed