Compile Data Set for Download or QSAR
Report error Found 34 Enz. Inhib. hit(s) with all data for entry = 50022168
TargetBcl-2-related protein A1(Human)TBA
LigandPNGBDBM50648874(CHEMBL5613766)
Affinity DataIC50: 22nMAssay Description:Inhibition of N-terminal His6-tagged recombinant Bfl-1 (1 to 151 residues)(unknown origin) extracted from Escherichia coli BL21-Gold (DE3) using HyLi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)TBA
LigandPNGBDBM50648872(CHEMBL5613621)
Affinity DataIC50: 63nMAssay Description:Inhibition of N-terminal His6-tagged recombinant Bfl-1 (1 to 151 residues)(unknown origin) extracted from Escherichia coli BL21-Gold (DE3) using HyLi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)TBA
LigandPNGBDBM50648869(CHEMBL5613029)
Affinity DataIC50: 300nMAssay Description:Inhibition of N-terminal His6-tagged recombinant Bfl-1 (1 to 151 residues)(unknown origin) extracted from Escherichia coli BL21-Gold (DE3) using HyLi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)TBA
LigandPNGBDBM50648859(CHEMBL5612066)
Affinity DataIC50: 340nMAssay Description:Inhibition of N-terminal His6-tagged recombinant Bfl-1 (1 to 151 residues)(unknown origin) extracted from Escherichia coli BL21-Gold (DE3) using HyLi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
TBA
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetBcl-2-related protein A1(Human)TBA
LigandPNGBDBM50648868(CHEMBL5612634)
Affinity DataIC50: 350nMAssay Description:Inhibition of N-terminal His6-tagged recombinant Bfl-1 (1 to 151 residues)(unknown origin) extracted from Escherichia coli BL21-Gold (DE3) using HyLi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)TBA
LigandPNGBDBM50648866(CHEMBL5612663)
Affinity DataIC50: 360nMAssay Description:Inhibition of N-terminal His6-tagged recombinant Bfl-1 (1 to 151 residues)(unknown origin) extracted from Escherichia coli BL21-Gold (DE3) using HyLi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)TBA
LigandPNGBDBM50648874(CHEMBL5613766)
Affinity DataEC50:  370nMAssay Description:Inhibition of Bfl-1 in human SU-DHL-1 cells assessed as caspase-3/7 activation measured after 6 hrs by UPLC-MRM MS analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)TBA
LigandPNGBDBM50648862(CHEMBL5613581)
Affinity DataIC50: 380nMAssay Description:Inhibition of N-terminal His6-tagged recombinant Bfl-1 (1 to 151 residues)(unknown origin) extracted from Escherichia coli BL21-Gold (DE3) using HyLi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)TBA
LigandPNGBDBM50648863(CHEMBL5614022)
Affinity DataIC50: 440nMAssay Description:Inhibition of N-terminal His6-tagged recombinant Bfl-1 (1 to 151 residues)(unknown origin) extracted from Escherichia coli BL21-Gold (DE3) using HyLi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)TBA
LigandPNGBDBM50648859(CHEMBL5612066)
Affinity DataIC50: 450nMAssay Description:Inhibition of N-terminal His6-tagged recombinant Bfl-1 (1 to 151 residues)(unknown origin) extracted from Escherichia coli BL21-Gold (DE3) using HyLi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
TBA
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetBcl-2-related protein A1(Human)TBA
LigandPNGBDBM50648864(CHEMBL5612546)
Affinity DataIC50: 460nMAssay Description:Inhibition of N-terminal His6-tagged recombinant Bfl-1 (1 to 151 residues)(unknown origin) extracted from Escherichia coli BL21-Gold (DE3) using HyLi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)TBA
LigandPNGBDBM50648870(CHEMBL5612215)
Affinity DataIC50: 550nMAssay Description:Inhibition of N-terminal His6-tagged recombinant Bfl-1 (1 to 151 residues)(unknown origin) extracted from Escherichia coli BL21-Gold (DE3) using HyLi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)TBA
LigandPNGBDBM50648867(CHEMBL5614064)
Affinity DataIC50: 720nMAssay Description:Inhibition of N-terminal His6-tagged recombinant Bfl-1 (1 to 151 residues)(unknown origin) extracted from Escherichia coli BL21-Gold (DE3) using HyLi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)TBA
LigandPNGBDBM50648873(CHEMBL5613885)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of N-terminal His6-tagged recombinant Bfl-1 (1 to 151 residues)(unknown origin) extracted from Escherichia coli BL21-Gold (DE3) using HyLi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)TBA
LigandPNGBDBM50648872(CHEMBL5613621)
Affinity DataEC50:  1.60E+3nMAssay Description:Inhibition of Bfl-1 in human SU-DHL-1 cells assessed as caspase-3/7 activation measured after 6 hrs by UPLC-MRM MS analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)TBA
LigandPNGBDBM50648869(CHEMBL5613029)
Affinity DataEC50:  1.80E+3nMAssay Description:Inhibition of Bfl-1 in human SU-DHL-1 cells assessed as caspase-3/7 activation measured after 6 hrs by UPLC-MRM MS analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)TBA
LigandPNGBDBM50648867(CHEMBL5614064)
Affinity DataEC50:  2.60E+3nMAssay Description:Inhibition of Bfl-1 in human SU-DHL-1 cells assessed as caspase-3/7 activation measured after 6 hrs by UPLC-MRM MS analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)TBA
LigandPNGBDBM50648871(CHEMBL5613717)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of N-terminal His6-tagged recombinant Bfl-1 (1 to 151 residues)(unknown origin) extracted from Escherichia coli BL21-Gold (DE3) using HyLi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)TBA
LigandPNGBDBM50648868(CHEMBL5612634)
Affinity DataEC50:  3.70E+3nMAssay Description:Inhibition of Bfl-1 in human SU-DHL-1 cells assessed as caspase-3/7 activation measured after 6 hrs by UPLC-MRM MS analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)TBA
LigandPNGBDBM50648858(CHEMBL5612442)
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibition of N-terminal His6-tagged recombinant Bfl-1 (1 to 151 residues)(unknown origin) extracted from Escherichia coli BL21-Gold (DE3) using HyLi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
TBA
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetBcl-2-related protein A1(Human)TBA
LigandPNGBDBM50648860(CHEMBL5613858)
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibition of N-terminal His6-tagged recombinant Bfl-1 (1 to 151 residues)(unknown origin) extracted from Escherichia coli BL21-Gold (DE3) using HyLi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)TBA
LigandPNGBDBM50648873(CHEMBL5613885)
Affinity DataEC50:  6.90E+3nMAssay Description:Inhibition of Bfl-1 in human SU-DHL-1 cells assessed as caspase-3/7 activation measured after 6 hrs by UPLC-MRM MS analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)TBA
LigandPNGBDBM50648859(CHEMBL5612066)
Affinity DataEC50:  7.40E+3nMAssay Description:Inhibition of Bfl-1 in human SU-DHL-1 cells assessed as caspase-3/7 activation measured after 6 hrs by UPLC-MRM MS analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
TBA
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetBcl-2-related protein A1(Human)TBA
LigandPNGBDBM50648857(CHEMBL5613623)
Affinity DataIC50: 9.80E+3nMAssay Description:Inhibition of N-terminal His6-tagged recombinant Bfl-1 (1 to 151 residues)(unknown origin) extracted from Escherichia coli BL21-Gold (DE3) using HyLi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)TBA
LigandPNGBDBM50648871(CHEMBL5613717)
Affinity DataEC50:  1.10E+4nMAssay Description:Inhibition of Bfl-1 in human SU-DHL-1 cells assessed as caspase-3/7 activation measured after 6 hrs by UPLC-MRM MS analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)TBA
LigandPNGBDBM50648855(CHEMBL5613897)
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of N-terminal His6-tagged recombinant Bfl-1 (1 to 151 residues)(unknown origin) extracted from Escherichia coli BL21-Gold (DE3) using HyLi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)TBA
LigandPNGBDBM50648865(CHEMBL5614038)
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibition of N-terminal His6-tagged recombinant Bfl-1 (1 to 151 residues)(unknown origin) extracted from Escherichia coli BL21-Gold (DE3) using HyLi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)TBA
LigandPNGBDBM50635693(CHEMBL5517789)
Affinity DataIC50: 2.30E+4nMAssay Description:Inhibition of N-terminal His6-tagged recombinant Bfl-1 (1 to 151 residues)(unknown origin) extracted from Escherichia coli BL21-Gold (DE3) using HyLi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)TBA
LigandPNGBDBM50648854(CHEMBL5613419)
Affinity DataIC50: 2.90E+4nMAssay Description:Inhibition of N-terminal His6-tagged recombinant Bfl-1 (1 to 151 residues)(unknown origin) extracted from Escherichia coli BL21-Gold (DE3) using HyLi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetBcl-2-like protein 1(Human)TBA
LigandPNGBDBM50648874(CHEMBL5613766)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of Bcl-xl (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50648874(CHEMBL5613766)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of Bcl-2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)TBA
LigandPNGBDBM50648861(CHEMBL5614214)
Affinity DataIC50: 4.20E+4nMAssay Description:Inhibition of N-terminal His6-tagged recombinant Bfl-1 (1 to 151 residues)(unknown origin) extracted from Escherichia coli BL21-Gold (DE3) using HyLi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetBcl-2-related protein A1(Human)TBA
LigandPNGBDBM50648856(CHEMBL5612726)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of N-terminal His6-tagged recombinant Bfl-1 (1 to 151 residues)(unknown origin) extracted from Escherichia coli BL21-Gold (DE3) using HyLi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50648874(CHEMBL5613766)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Mcl-1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed