Compile Data Set for Download or QSAR
Report error Found 167 Enz. Inhib. hit(s) with all data for entry = 50023482
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Affiliated Hengyang Hospital of Hunan Normal University & Hengyang Central Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 296429BDBM296429(US10112942, Example 163 | US10112942, Example 183 ...)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of RET V804L mutant (unknown origin) by FRET-based ZLyte kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Affiliated Hengyang Hospital of Hunan Normal University & Hengyang Central Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50664122BDBM50664122(CHEMBL6162402)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of RET V804L mutant (unknown origin) by FRET-based ZLyte kinase assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Affiliated Hengyang Hospital of Hunan Normal University & Hengyang Central Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 296429BDBM296429(US10112942, Example 163 | US10112942, Example 183 ...)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of RET M918T mutant (unknown origin) by FRET-based ZLyte kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Affiliated Hengyang Hospital of Hunan Normal University & Hengyang Central Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50664118BDBM50664118(CHEMBL6161713)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of RET V804L mutant (unknown origin) by FRET-based ZLyte kinase assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Affiliated Hengyang Hospital of Hunan Normal University & Hengyang Central Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50664102BDBM50664102(CHEMBL6162327)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of RET V804L mutant (unknown origin) by FRET-based ZLyte kinase assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Affiliated Hengyang Hospital of Hunan Normal University & Hengyang Central Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50664122BDBM50664122(CHEMBL6162402)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of RET M918T mutant (unknown origin) by FRET-based ZLyte kinase assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Affiliated Hengyang Hospital of Hunan Normal University & Hengyang Central Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50664118BDBM50664118(CHEMBL6161713)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of RET M918T mutant (unknown origin) by FRET-based ZLyte kinase assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Affiliated Hengyang Hospital of Hunan Normal University & Hengyang Central Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50664101BDBM50664101(CHEMBL6161307)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of RET V804L mutant (unknown origin) by FRET-based ZLyte kinase assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Affiliated Hengyang Hospital of Hunan Normal University & Hengyang Central Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50664102BDBM50664102(CHEMBL6162327)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of RET M918T mutant (unknown origin) by FRET-based ZLyte kinase assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Affiliated Hengyang Hospital of Hunan Normal University & Hengyang Central Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50331094BDBM50331094(4-(3-chloro-4-(3-cyclopropylureido)phenoxy)-7-meth...)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of human full-length RETMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Affiliated Hengyang Hospital of Hunan Normal University & Hengyang Central Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50664122BDBM50664122(CHEMBL6162402)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of RET V804M mutant (unknown origin) by FRET-based ZLyte kinase assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Affiliated Hengyang Hospital of Hunan Normal University & Hengyang Central Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 296429BDBM296429(US10112942, Example 163 | US10112942, Example 183 ...)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of RET V804M mutant (unknown origin) by FRET-based ZLyte kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Affiliated Hengyang Hospital of Hunan Normal University & Hengyang Central Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50664115BDBM50664115(CHEMBL6134510)
Affinity DataIC50: 2.30nMAssay Description:Inhibition of RET V804L mutant (unknown origin) by FRET-based ZLyte kinase assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Affiliated Hengyang Hospital of Hunan Normal University & Hengyang Central Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50664108BDBM50664108(CHEMBL6163978)
Affinity DataIC50: 2.30nMAssay Description:Inhibition of RET V804L mutant (unknown origin) by FRET-based ZLyte kinase assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Affiliated Hengyang Hospital of Hunan Normal University & Hengyang Central Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50664107BDBM50664107(CHEMBL6162262)
Affinity DataIC50: 2.60nMAssay Description:Inhibition of RET V804L mutant (unknown origin) by FRET-based ZLyte kinase assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Affiliated Hengyang Hospital of Hunan Normal University & Hengyang Central Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50664108BDBM50664108(CHEMBL6163978)
Affinity DataIC50: 3nMAssay Description:Inhibition of RET M918T mutant (unknown origin) by FRET-based ZLyte kinase assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Affiliated Hengyang Hospital of Hunan Normal University & Hengyang Central Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50664117BDBM50664117(CHEMBL6151761)
Affinity DataIC50: 3.10nMAssay Description:Inhibition of RET V804L mutant (unknown origin) by FRET-based ZLyte kinase assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Affiliated Hengyang Hospital of Hunan Normal University & Hengyang Central Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50664122BDBM50664122(CHEMBL6162402)
Affinity DataIC50: 3.20nMAssay Description:Inhibition of wild type RET (unknown origin) by FRET-based ZLyte kinase assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Affiliated Hengyang Hospital of Hunan Normal University & Hengyang Central Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 296429BDBM296429(US10112942, Example 163 | US10112942, Example 183 ...)
Affinity DataIC50: 3.60nMAssay Description:Inhibition of wild type RET (unknown origin) by FRET-based ZLyte kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Affiliated Hengyang Hospital of Hunan Normal University & Hengyang Central Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50664102BDBM50664102(CHEMBL6162327)
Affinity DataIC50: 3.80nMAssay Description:Inhibition of wild type RET (unknown origin) by FRET-based ZLyte kinase assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Affiliated Hengyang Hospital of Hunan Normal University & Hengyang Central Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50664109BDBM50664109(CHEMBL6166963)
Affinity DataIC50: 4nMAssay Description:Inhibition of RET V804L mutant (unknown origin) by FRET-based ZLyte kinase assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Affiliated Hengyang Hospital of Hunan Normal University & Hengyang Central Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50664110BDBM50664110(CHEMBL6172802)
Affinity DataIC50: 4.70nMAssay Description:Inhibition of RET V804L mutant (unknown origin) by FRET-based ZLyte kinase assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Affiliated Hengyang Hospital of Hunan Normal University & Hengyang Central Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50664117BDBM50664117(CHEMBL6151761)
Affinity DataIC50: 4.70nMAssay Description:Inhibition of RET M918T mutant (unknown origin) by FRET-based ZLyte kinase assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Affiliated Hengyang Hospital of Hunan Normal University & Hengyang Central Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50664108BDBM50664108(CHEMBL6163978)
Affinity DataIC50: 4.80nMAssay Description:Inhibition of wild type RET (unknown origin) by FRET-based ZLyte kinase assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Affiliated Hengyang Hospital of Hunan Normal University & Hengyang Central Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50664107BDBM50664107(CHEMBL6162262)
Affinity DataIC50: 4.90nMAssay Description:Inhibition of RET M918T mutant (unknown origin) by FRET-based ZLyte kinase assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Affiliated Hengyang Hospital of Hunan Normal University & Hengyang Central Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50664115BDBM50664115(CHEMBL6134510)
Affinity DataIC50: 5.10nMAssay Description:Inhibition of RET M918T mutant (unknown origin) by FRET-based ZLyte kinase assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetVascular endothelial growth factor receptor 3(Human)
Affiliated Hengyang Hospital of Hunan Normal University & Hengyang Central Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50664122BDBM50664122(CHEMBL6162402)
Affinity DataIC50: 5.10nMAssay Description:Inhibition of FLT4 (unknown origin) by FRET-based Z-Lyte kinase assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Affiliated Hengyang Hospital of Hunan Normal University & Hengyang Central Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50021574BDBM50021574(CHEBI:72317 | CABOZANTINIB | BMS-907351 | Cometriq...)
Affinity DataIC50: 5.20nMAssay Description:Inhibition of RET (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Affiliated Hengyang Hospital of Hunan Normal University & Hengyang Central Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50664118BDBM50664118(CHEMBL6161713)
Affinity DataIC50: 5.5nMAssay Description:Inhibition of wild type RET (unknown origin) by FRET-based ZLyte kinase assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Affiliated Hengyang Hospital of Hunan Normal University & Hengyang Central Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50664114BDBM50664114(CHEMBL6143395)
Affinity DataIC50: 5.60nMAssay Description:Inhibition of RET V804L mutant (unknown origin) by FRET-based ZLyte kinase assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Affiliated Hengyang Hospital of Hunan Normal University & Hengyang Central Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50664122BDBM50664122(CHEMBL6162402)
Affinity DataIC50: 5.70nMAssay Description:Inhibition of RET G810S mutant (unknown origin) by FRET-based ZLyte kinase assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Affiliated Hengyang Hospital of Hunan Normal University & Hengyang Central Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50664107BDBM50664107(CHEMBL6162262)
Affinity DataIC50: 5.70nMAssay Description:Inhibition of wild type RET (unknown origin) by FRET-based ZLyte kinase assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Affiliated Hengyang Hospital of Hunan Normal University & Hengyang Central Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50664109BDBM50664109(CHEMBL6166963)
Affinity DataIC50: 5.90nMAssay Description:Inhibition of RET M918T mutant (unknown origin) by FRET-based ZLyte kinase assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Affiliated Hengyang Hospital of Hunan Normal University & Hengyang Central Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50664101BDBM50664101(CHEMBL6161307)
Affinity DataIC50: 5.90nMAssay Description:Inhibition of wild type RET (unknown origin) by FRET-based ZLyte kinase assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Affiliated Hengyang Hospital of Hunan Normal University & Hengyang Central Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 16673BDBM16673(BAY439006 | CHEMBL1336 | BAY 43-9006 | 4-[4-({[4-c...)
Affinity DataIC50: 5.90nMAssay Description:Inhibition of recombinant wild type RET (unknown origin) extracted from baculovirusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Affiliated Hengyang Hospital of Hunan Normal University & Hengyang Central Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50664101BDBM50664101(CHEMBL6161307)
Affinity DataIC50: 6.5nMAssay Description:Inhibition of RET M918T mutant (unknown origin) by FRET-based ZLyte kinase assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Affiliated Hengyang Hospital of Hunan Normal University & Hengyang Central Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50664110BDBM50664110(CHEMBL6172802)
Affinity DataIC50: 6.70nMAssay Description:Inhibition of RET M918T mutant (unknown origin) by FRET-based ZLyte kinase assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Affiliated Hengyang Hospital of Hunan Normal University & Hengyang Central Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50664110BDBM50664110(CHEMBL6172802)
Affinity DataIC50: 6.70nMAssay Description:Inhibition of wild type RET (unknown origin) by FRET-based ZLyte kinase assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Affiliated Hengyang Hospital of Hunan Normal University & Hengyang Central Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50664122BDBM50664122(CHEMBL6162402)
Affinity DataIC50: 7.10nMAssay Description:Inhibition of RET G810C mutant (unknown origin) by FRET-based ZLyte kinase assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Affiliated Hengyang Hospital of Hunan Normal University & Hengyang Central Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50664117BDBM50664117(CHEMBL6151761)
Affinity DataIC50: 7.60nMAssay Description:Inhibition of wild type RET (unknown origin) by FRET-based ZLyte kinase assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Affiliated Hengyang Hospital of Hunan Normal University & Hengyang Central Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50664122BDBM50664122(CHEMBL6162402)
Affinity DataIC50: 8.30nMAssay Description:Inhibition of RET G810R mutant (unknown origin) by FRET-based ZLyte kinase assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Affiliated Hengyang Hospital of Hunan Normal University & Hengyang Central Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50664119BDBM50664119(CHEMBL6159712)
Affinity DataIC50: 8.5nMAssay Description:Inhibition of RET V804L mutant (unknown origin) by FRET-based ZLyte kinase assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Affiliated Hengyang Hospital of Hunan Normal University & Hengyang Central Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50664109BDBM50664109(CHEMBL6166963)
Affinity DataIC50: 9.10nMAssay Description:Inhibition of wild type RET (unknown origin) by FRET-based ZLyte kinase assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Affiliated Hengyang Hospital of Hunan Normal University & Hengyang Central Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50664114BDBM50664114(CHEMBL6143395)
Affinity DataIC50: 9.30nMAssay Description:Inhibition of RET M918T mutant (unknown origin) by FRET-based ZLyte kinase assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Affiliated Hengyang Hospital of Hunan Normal University & Hengyang Central Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50664115BDBM50664115(CHEMBL6134510)
Affinity DataIC50: 9.80nMAssay Description:Inhibition of wild type RET (unknown origin) by FRET-based ZLyte kinase assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Affiliated Hengyang Hospital of Hunan Normal University & Hengyang Central Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50664119BDBM50664119(CHEMBL6159712)
Affinity DataIC50: 11nMAssay Description:Inhibition of RET M918T mutant (unknown origin) by FRET-based ZLyte kinase assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Affiliated Hengyang Hospital of Hunan Normal University & Hengyang Central Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50664100BDBM50664100(CHEMBL6169354)
Affinity DataIC50: 13nMAssay Description:Inhibition of RET V804L mutant (unknown origin) by FRET-based ZLyte kinase assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Affiliated Hengyang Hospital of Hunan Normal University & Hengyang Central Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50664116BDBM50664116(CHEMBL6161968)
Affinity DataIC50: 13nMAssay Description:Inhibition of wild type RET (unknown origin) by FRET-based ZLyte kinase assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Affiliated Hengyang Hospital of Hunan Normal University & Hengyang Central Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50664116BDBM50664116(CHEMBL6161968)
Affinity DataIC50: 14nMAssay Description:Inhibition of RET V804L mutant (unknown origin) by FRET-based ZLyte kinase assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Affiliated Hengyang Hospital of Hunan Normal University & Hengyang Central Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50664120BDBM50664120(CHEMBL6170007)
Affinity DataIC50: 14nMAssay Description:Inhibition of RET V804L mutant (unknown origin) by FRET-based ZLyte kinase assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
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