Compile Data Set for Download or QSAR
Report error Found 29 Enz. Inhib. hit(s) with all data for entry = 50022967
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Univ. Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50656843BDBM50656843(CHEMBL6102768)
Affinity DataIC50: 1.72E+3nMAssay Description:Inhibition of recombinant human ERAP1 using L-AMC as substrate preincubated for 30 mins followed by substrate addition and measured after 1 hr by flu...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Univ. Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50656839BDBM50656839(CHEMBL1720102)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of recombinant human ERAP1 using L-AMC as substrate preincubated for 30 mins followed by substrate addition and measured after 1 hr by flu...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Univ. Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50656832BDBM50656832(CHEMBL6161623)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of human ERAP1 using L-SIINFEKL as substrate by LC-MS/MS methodMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Univ. Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50656832BDBM50656832(CHEMBL6161623)
Affinity DataIC50: 7.30E+3nMAssay Description:Inhibition of recombinant human ERAP1 using L-AMC as substrate preincubated for 30 mins followed by substrate addition and measured after 1 hr by flu...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Univ. Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50656839BDBM50656839(CHEMBL1720102)
Affinity DataIC50: 1.03E+4nMAssay Description:Inhibition of human ERAP1 using L-SIINFEKL as substrate by LC-MS/MS methodMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetInterleukin-1 receptor antagonist protein(Human)
Univ. Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50656850BDBM50656850(CHEMBL6149727)
Affinity DataIC50: 1.33E+4nMAssay Description:Inhibition of recombinant human IRAP using L-AMC as substrate preincubated for 30 mins followed by substrate addition and measured after 1 hr by fluo...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetInterleukin-1 receptor antagonist protein(Human)
Univ. Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50656848BDBM50656848(CHEMBL6133600)
Affinity DataIC50: 1.44E+4nMAssay Description:Inhibition of recombinant human IRAP using L-AMC as substrate preincubated for 30 mins followed by substrate addition and measured after 1 hr by fluo...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetInterleukin-1 receptor antagonist protein(Human)
Univ. Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50656849BDBM50656849(CHEMBL6133751)
Affinity DataIC50: 1.51E+4nMAssay Description:Inhibition of recombinant human IRAP using L-AMC as substrate preincubated for 30 mins followed by substrate addition and measured after 1 hr by fluo...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetInterleukin-1 receptor antagonist protein(Human)
Univ. Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50656846BDBM50656846(CHEMBL6146245)
Affinity DataIC50: 1.63E+4nMAssay Description:Inhibition of recombinant human IRAP using L-AMC as substrate preincubated for 30 mins followed by substrate addition and measured after 1 hr by fluo...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Univ. Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50656844BDBM50656844(CHEMBL6142965)
Affinity DataIC50: 1.84E+4nMAssay Description:Inhibition of recombinant human ERAP1 using L-AMC as substrate preincubated for 30 mins followed by substrate addition and measured after 1 hr by flu...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Univ. Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50359684BDBM50359684(CHEMBL1929273)
Affinity DataIC50: 1.95E+4nMAssay Description:Inhibition of recombinant human ERAP1 using L-AMC as substrate preincubated for 30 mins followed by substrate addition and measured after 1 hr by flu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Univ. Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 80675BDBM80675(2-(5-pyrrolidin-1-ylsulfonylthiophen-2-yl)ethanoic...)
Affinity DataIC50: 2.72E+4nMAssay Description:Inhibition of recombinant human ERAP1 using L-AMC as substrate preincubated for 30 mins followed by substrate addition and measured after 1 hr by flu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Univ. Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50359684BDBM50359684(CHEMBL1929273)
Affinity DataIC50: 2.86E+4nMAssay Description:Inhibition of human ERAP1 using L-SIINFEKL as substrate by LC-MS/MS methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Univ. Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50656837BDBM50656837(CHEMBL6151327)
Affinity DataIC50: 3.18E+4nMAssay Description:Inhibition of human ERAP1 using L-SIINFEKL as substrate by LC-MS/MS methodMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Univ. Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50656840BDBM50656840(CHEMBL6159756)
Affinity DataIC50: 3.38E+4nMAssay Description:Inhibition of recombinant human ERAP1 using L-AMC as substrate preincubated for 30 mins followed by substrate addition and measured after 1 hr by flu...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Univ. Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50656835BDBM50656835(CHEMBL6102785)
Affinity DataIC50: 4.02E+4nMAssay Description:Inhibition of recombinant human ERAP1 using L-AMC as substrate preincubated for 30 mins followed by substrate addition and measured after 1 hr by flu...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetInterleukin-1 receptor antagonist protein(Human)
Univ. Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50359684BDBM50359684(CHEMBL1929273)
Affinity DataIC50: 4.09E+4nMAssay Description:Inhibition of recombinant human IRAP using L-AMC as substrate preincubated for 30 mins followed by substrate addition and measured after 1 hr by fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Univ. Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50656842BDBM50656842(CHEMBL6148773)
Affinity DataIC50: 4.27E+4nMAssay Description:Inhibition of recombinant human ERAP1 using L-AMC as substrate preincubated for 30 mins followed by substrate addition and measured after 1 hr by flu...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Univ. Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50656838BDBM50656838(CHEMBL590160)
Affinity DataIC50: 4.50E+4nMAssay Description:Inhibition of recombinant human ERAP1 using L-AMC as substrate preincubated for 30 mins followed by substrate addition and measured after 1 hr by flu...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Univ. Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50656837BDBM50656837(CHEMBL6151327)
Affinity DataIC50: 4.52E+4nMAssay Description:Inhibition of recombinant human ERAP1 using L-AMC as substrate preincubated for 30 mins followed by substrate addition and measured after 1 hr by flu...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Univ. Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50656836BDBM50656836(CHEMBL6149786)
Affinity DataIC50: 5.23E+4nMAssay Description:Inhibition of human ERAP1 using L-SIINFEKL as substrate by LC-MS/MS methodMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Univ. Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50656836BDBM50656836(CHEMBL6149786)
Affinity DataIC50: 5.64E+4nMAssay Description:Inhibition of recombinant human ERAP1 using L-AMC as substrate preincubated for 30 mins followed by substrate addition and measured after 1 hr by flu...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Univ. Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50656833BDBM50656833(CHEMBL1468092)
Affinity DataIC50: 5.83E+4nMAssay Description:Inhibition of recombinant human ERAP1 using L-AMC as substrate preincubated for 30 mins followed by substrate addition and measured after 1 hr by flu...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetInterleukin-1 receptor antagonist protein(Human)
Univ. Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50656845BDBM50656845(CHEMBL6141829)
Affinity DataIC50: 6.03E+4nMAssay Description:Inhibition of recombinant human IRAP using L-AMC as substrate preincubated for 30 mins followed by substrate addition and measured after 1 hr by fluo...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Univ. Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50656831BDBM50656831(CHEMBL6134124)
Affinity DataIC50: 6.14E+4nMAssay Description:Inhibition of human ERAP1 using L-SIINFEKL as substrate by LC-MS/MS methodMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Univ. Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50656834BDBM50656834(CHEMBL6134689)
Affinity DataIC50: 8.26E+4nMAssay Description:Inhibition of recombinant human ERAP1 using L-AMC as substrate preincubated for 30 mins followed by substrate addition and measured after 1 hr by flu...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetInterleukin-1 receptor antagonist protein(Human)
Univ. Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50656847BDBM50656847(CHEMBL1550354)
Affinity DataIC50: 8.81E+4nMAssay Description:Inhibition of recombinant human IRAP using L-AMC as substrate preincubated for 30 mins followed by substrate addition and measured after 1 hr by fluo...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Univ. Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50656841BDBM50656841(CHEMBL6147062)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human ERAP1 using L-AMC as substrate preincubated for 30 mins followed by substrate addition and measured after 1 hr by flu...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed
TargetEndoplasmic reticulum aminopeptidase 1(Human)
Univ. Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50656831BDBM50656831(CHEMBL6134124)
Affinity DataIC50: 1.03E+5nMAssay Description:Inhibition of recombinant human ERAP1 using L-AMC as substrate preincubated for 30 mins followed by substrate addition and measured after 1 hr by flu...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details
PubMed