Report error Found 126 Enz. Inhib. hit(s) with all data for entry = 50022837
Affinity DataKi: 0.800nMAssay Description:Antagonist activity at Prolink-tagged human CXCR6 receptor assessed as inhibition of forskolin-induced cAMP accumulation by DiscoveRx cell based assa...More data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Antagonist activity at Prolink-tagged human CXCR6 receptor assessed as inhibition of CXCL16-induced beta-arrestin recruitment by DiscoveRx cell based...More data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:Inhibition of PI3Kbeta (unknown origin) by cell based assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 2.80nMAssay Description:Antagonist activity against HIV-1 Vif in human H9 cells expressing A3G assessed as inhibition of viral infection measured after 16 hrs by cell-based ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 3nMAssay Description:Antagonist activity against HIV-1 Vif in human H9 cells expressing A3G assessed as inhibition of viral infection measured after 16 hrs by cell-based ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 3.30nMAssay Description:Antagonist activity against HIV-1 Vif in human H9 cells expressing A3G assessed as inhibition of viral infection measured after 16 hrs by cell-based ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 3.80nMAssay Description:Antagonist activity at Prolink-tagged human CXCR6 receptor assessed as inhibition of CXCL16-induced beta-arrestin recruitment by DiscoveRx cell based...More data for this Ligand-Target Pair
Affinity DataKi: 4.20nMAssay Description:Inhibition of JAK1/JAK2 (unknown origin) in GM-CSF stimulated cells by cell based assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 4.20nMAssay Description:Antagonist activity against HIV-1 Vif in human H9 cells expressing A3G assessed as inhibition of viral infection measured after 16 hrs by cell-based ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 4.80nMAssay Description:Antagonist activity against HIV-1 Vif in human MT4 cells assessed as inhibition of viral infection measured after 16 hrs by cell-based assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 4.90nMAssay Description:Antagonist activity against HIV-1 Vif in human H9 cells expressing A3G assessed as inhibition of viral infection measured after 16 hrs by cell-based ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 5.40nMAssay Description:Antagonist activity against HIV-1 Vif in human H9 cells expressing A3G assessed as inhibition of viral infection measured after 16 hrs by cell-based ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 5.80nMAssay Description:Antagonist activity against HIV-1 Vif in human H9 cells expressing A3G assessed as inhibition of viral infection measured after 16 hrs by cell-based ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 6.60nMAssay Description:Antagonist activity against HIV-1 Vif in human H9 cells expressing A3G assessed as inhibition of viral infection measured after 16 hrs by cell-based ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 7.10nMAssay Description:Antagonist activity at Prolink-tagged human CXCR6 receptor assessed as inhibition of CXCL16-induced beta-arrestin recruitment by DiscoveRx cell based...More data for this Ligand-Target Pair
Affinity DataKi: 7.5nMAssay Description:Antagonist activity against HIV-1 Vif in human H9 cells expressing A3G assessed as inhibition of viral infection measured after 16 hrs by cell-based ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 9.20nMAssay Description:Antagonist activity against HIV-1 Vif in human H9 cells expressing A3G assessed as inhibition of viral infection measured after 16 hrs by cell-based ...More data for this Ligand-Target Pair
Affinity DataIC50: 9.5nMAssay Description:Antagonist activity at Prolink-tagged human CXCR6 receptor assessed as inhibition of CXCL16-induced beta-arrestin recruitment by DiscoveRx cell based...More data for this Ligand-Target Pair
Affinity DataKi: 9.5nMAssay Description:Inhibition of IDO1 (unknown origin) by cell based assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 10nMAssay Description:Antagonist activity against HIV-1 Vif in human MT4 cells assessed as inhibition of viral infection measured after 16 hrs by cell-based assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 11nMAssay Description:Antagonist activity against HIV-1 Vif in human H9 cells expressing A3G assessed as inhibition of viral infection measured after 16 hrs by cell-based ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 13nMAssay Description:Inhibition of FLT3 (unknown origin) autophosphorylation by cell based enzyme-linked immunosorbent assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 14nMAssay Description:Antagonist activity against HIV-1 Vif in human H9 cells expressing A3G assessed as inhibition of viral infection measured after 16 hrs by cell-based ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 15nMAssay Description:Inhibition of JAK1/JAK3 (unknown origin) in IL-2 stimulated cells by cell based assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 15nMAssay Description:Antagonist activity against HIV-1 Vif in human H9 cells expressing A3G assessed as inhibition of viral infection measured after 16 hrs by cell-based ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 15nMAssay Description:Antagonist activity against HIV-1 Vif in human H9 cells expressing A3G assessed as inhibition of viral infection measured after 16 hrs by cell-based ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 16nMAssay Description:Antagonist activity at OX1R (unknown origin) assessed as inhibition of orexin A-induced intracellular Ca2+ release by cell-based assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 17nMAssay Description:Antagonist activity against HIV-1 Vif in human H9 cells expressing A3G assessed as inhibition of viral infection measured after 16 hrs by cell-based ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 17nMAssay Description:Inhibition of TRPC5 (unknown origin) transfected in HEK293/TREx cells assessed as reduction of rise in intracellular Ca2+ concentration after 60 to 8...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 20nMAssay Description:Antagonist activity against HIV-1 Vif in human H9 cells expressing A3G assessed as inhibition of viral infection measured after 16 hrs by cell-based ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 20nMAssay Description:Inhibition of JAK1/JAK3 (unknown origin) in IL-2 stimulated cells by cell based assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 20nMAssay Description:Antagonist activity against HIV-1 Vif in human H9 cells expressing A3G assessed as inhibition of viral infection measured after 16 hrs by cell-based ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 20nMAssay Description:Inhibition of IDO1 (unknown origin) by cell based assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 20nMAssay Description:Antagonist activity against HIV-1 Vif in human H9 cells expressing A3G assessed as inhibition of viral infection measured after 16 hrs by cell-based ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 20nMAssay Description:Antagonist activity at Prolink-tagged human CXCR6 receptor assessed as inhibition of CXCL16-induced beta-arrestin recruitment by DiscoveRx cell based...More data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Antagonist activity against HIV-1 Vif in human H9 cells expressing A3G assessed as inhibition of viral infection measured after 16 hrs by cell-based ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 23nMAssay Description:Antagonist activity at Prolink-tagged human CXCR6 receptor assessed as inhibition of CXCL16-induced beta-arrestin recruitment by DiscoveRx cell based...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 26nMAssay Description:Antagonist activity against HIV-1 Vif in human H9 cells expressing A3G assessed as inhibition of viral infection measured after 16 hrs by cell-based ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 26nMAssay Description:Antagonist activity at OX1R (unknown origin) assessed as inhibition of orexin A-induced intracellular Ca2+ release by cell-based assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 27nMAssay Description:Antagonist activity against HIV-1 Vif in human H9 cells expressing A3G assessed as inhibition of viral infection measured after 16 hrs by cell-based ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 28nMAssay Description:Inhibition of JAK1/JAK3 (unknown origin) in IL-2 stimulated cells by cell based assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 28nMAssay Description:Antagonist activity against HIV-1 Vif in human H9 cells expressing A3G assessed as inhibition of viral infection measured after 16 hrs by cell-based ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 29nMAssay Description:Antagonist activity against HIV-1 Vif in human H9 cells expressing A3G assessed as inhibition of viral infection measured after 16 hrs by cell-based ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 30nMAssay Description:Antagonist activity against HIV-1 Vif in human H9 cells expressing A3G assessed as inhibition of viral infection measured after 16 hrs by cell-based ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 30nMAssay Description:Antagonist activity at OX1R (unknown origin) assessed as inhibition of orexin A-induced intracellular Ca2+ release by cell-based assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 30nMAssay Description:Inhibition of JAK1/JAK2 (unknown origin) in GM-CSF stimulated cells by cell based assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 31nMAssay Description:Antagonist activity against HIV-1 Vif in human H9 cells expressing A3G assessed as inhibition of viral infection measured after 16 hrs by cell-based ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 32nMAssay Description:Inhibition of PI3Kbeta (unknown origin) by cell based assayMore data for this Ligand-Target Pair
Affinity DataKi: 33nMAssay Description:Antagonist activity against HIV-1 Vif in human H9 cells expressing A3G assessed as inhibition of viral infection measured after 16 hrs by cell-based ...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKi: 35nMAssay Description:Antagonist activity at OX1R (unknown origin) assessed as inhibition of orexin A-induced intracellular Ca2+ release by cell-based assayMore data for this Ligand-Target Pair
Ligand Info


3D Structure (crystal)






























