Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50023730
TargetCannabinoid receptor 2(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50667404BDBM50667404(CHEMBL6193707)
Affinity DataKi:  0.900nMAssay Description:Binding affinity to human CB2 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetEpithelial discoidin domain-containing receptor 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50667405BDBM50667405(CHEMBL6193264)
Affinity DataIC50: 10nMAssay Description:Inhibition of human DDR1More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetAmyloid-beta precursor protein(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50667406BDBM50667406(CHEMBL6192437)
Affinity DataKd:  20nMAssay Description:Binding affinity to amyloid beta fibril ( 1 to 42 residues) (unknown origin) assessed as dissociation constant by fluorescence based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetAmyloid-beta precursor protein(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50667407BDBM50667407(CHEMBL6189106)
Affinity DataKd:  20nMAssay Description:Binding affinity to amyloid beta fibril ( 1 to 42 residues) (unknown origin) assessed as dissociation constant by fluorescence based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetRho-associated protein kinase 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50667405BDBM50667405(CHEMBL6193264)
Affinity DataKi:  38nMAssay Description:Binding affinity to N-terminal GST-tagged human ROCK1 catalytic domain (1 to 477 residues) expressed in Sf21 insect cells assessed as inhibition cons...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetTyrosine-protein kinase JAK2(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50667405BDBM50667405(CHEMBL6193264)
Affinity DataIC50: 70nMAssay Description:Inhibition of JAK2 (unknown origin) by Z'-LYTE kinase assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetForkhead box protein M1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50667402BDBM50667402(CHEMBL2205761)
Affinity DataKd:  910nMAssay Description:Binding affinity to FOXM1 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetAndrogen receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50667400BDBM50667400(CHEMBL6191318)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of full length human Androgen receptor DNA binding domain dimerizationMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetSpeckle-type POZ protein(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50667408BDBM50667408(CHEMBL6190856)
Affinity DataIC50: 4.51E+3nMAssay Description:Inhibition of recombinant GST-tagged SPOP (unknown origin) extracted from Escherichia coli BL21-CodonPlus (DE3)-RIPL cells using FITC-LACDEVTSTTSSSTA...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetAndrogen receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50667399BDBM50667399(CHEMBL6189480)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of full length human Androgen receptor DNA binding domain dimerizationMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetMyeloid differentiation primary response protein MyD88(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50667401BDBM50667401(CHEMBL6192241)
Affinity DataKd:  1.65E+5nMAssay Description:Binding affinity to MYD88 Toll/interleukin-1 receptor domain (unknown origin) assessed as dissociation constant by SPR assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetSerine/threonine-protein kinase Sgk3(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50667403BDBM50667403(CHEMBL6190297)
Affinity DataIC50: 1.79E+5nMAssay Description:Inhibition of SGK3 (unknown origin)More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed