Compile Data Set for Download or QSAR
maximum 50k data
Found 8 Enz. Inhib. hit(s) with all data for entry = 50003215
TargetHigh affinity choline transporter 1(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50026216(1-Ethyl-1-(2-hydroxy-ethyl)-aziridinium; chloride ...)
Affinity DataIC50:  1.50E+3nMAssay Description:Compound was evaluated in vitro for its ability to inhibit the transport of [3H]-choline in to high affinity choline transport system HAChTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50026220(2-hydroxy-N,N,N-trimethylethanaminium | CHEMBL2824...)
Affinity DataIC50:  1.60E+3nMAssay Description:Compound was evaluated in vitro for its ability to inhibit the transport of [3H]-choline in to high affinity choline transport system HAChTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50026218(1-(2-Hydroxy-ethyl)-1-isopropyl-aziridinium; chlor...)
Affinity DataIC50:  2.60E+3nMAssay Description:Compound was evaluated in vitro for its ability to inhibit the transport of [3H]-choline in to high affinity choline transport system HAChTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50026215(1-Cyclopropyl-1-(2-hydroxy-ethyl)-aziridinium; chl...)
Affinity DataIC50:  3.90E+3nMAssay Description:Compound was evaluated in vitro for its ability to inhibit the transport of [3H]-choline in to high affinity choline transport system HAChTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50026215(1-Cyclopropyl-1-(2-hydroxy-ethyl)-aziridinium; chl...)
Affinity DataIC50:  6.25E+3nMAssay Description:Compound was tested in vitro for its ability to displace [3H]-QNB from brain Muscarinic acetylcholine receptor by 50 %More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50026219(1-(2-Hydroxy-ethyl)-1-propyl-aziridinium; chloride...)
Affinity DataIC50:  7.50E+3nMAssay Description:Compound was evaluated in vitro for its ability to inhibit the transport of [3H]-choline in to high affinity choline transport system HAChTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50026217(1-(2-Hydroxy-ethyl)-1-isobutyl-aziridinium; chlori...)
Affinity DataIC50:  3.10E+4nMAssay Description:Compound was evaluated in vitro for its ability to inhibit the transport of [3H]-choline in to high affinity choline transport system HAChTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50026221(1-Butyl-1-(2-hydroxy-ethyl)-aziridinium; chloride ...)
Affinity DataIC50: >1.00E+6nMAssay Description:Compound was evaluated in vitro for its ability to inhibit the transport of [3H]-choline in to high affinity choline transport system HAChTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed