Report error Found 92 Enz. Inhib. hit(s) with all data for entry = 50023516
Affinity DataIC50: 1.20nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human EGFR T790M/L858R mutant (696 to end residues) extracted from baculovirus infect Sf21 insect cel...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.40nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human EGFR T790M/L858R mutant (696 to end residues) extracted from baculovirus infect Sf21 insect cel...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.60nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human EGFR 19del/T790M/C797S mutant (668 to end residues) extracted from Sf9 insect cells incubated f...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.60nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human EGFR T790M/L858R mutant (696 to end residues) extracted from baculovirus infect Sf21 insect cel...More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human EGFR T790M/L858R mutant (696 to end residues) extracted from baculovirus infect Sf21 insect cel...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 2.20nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human EGFR T790M/L858R mutant (696 to end residues) extracted from baculovirus infect Sf21 insect cel...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 2.30nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human EGFR 19del/T790M/C797S mutant (668 to end residues) extracted from Sf9 insect cells incubated f...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 2.70nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human EGFR 19del/T790M/C797S mutant (668 to end residues) extracted from Sf9 insect cells incubated f...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 2.70nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human EGFR 19del/T790M/C797S mutant (668 to end residues) extracted from Sf9 insect cells incubated f...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 2.90nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human EGFR T790M/L858R mutant (696 to end residues) extracted from baculovirus infect Sf21 insect cel...More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human EGFR T790M/L858R mutant (696 to end residues) extracted from baculovirus infect Sf21 insect cel...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 3.10nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human EGFR 19del/T790M/C797S mutant (668 to end residues) extracted from Sf9 insect cells incubated f...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 3.60nMAssay Description:Inhibition of recombinant C-terminal His-tagged/N-terminal GST-tagged human EGFR T790M/C797S/L858R mutant (668 to 1210 residues) extracted from bacul...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 3.60nMAssay Description:Inhibition of recombinant C-terminal His-tagged/N-terminal GST-tagged human EGFR T790M/C797S/L858R mutant (668 to 1210 residues) extracted from bacul...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 4.80nMAssay Description:Inhibition of recombinant wildtype N-terminal GST-tagged human EGFR kinase domain (696 to end residues) extracted from baculovirus infect Sf21 insect...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 5.30nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human EGFR 19del/T790M/C797S mutant (668 to end residues) extracted from Sf9 insect cells incubated f...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 6.10nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human EGFR 19del/T790M/C797S mutant (668 to end residues) extracted from Sf9 insect cells incubated f...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 13nMAssay Description:Inhibition of recombinant C-terminal His-tagged/N-terminal GST-tagged human EGFR T790M/C797S/L858R mutant (668 to 1210 residues) extracted from bacul...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 13nMAssay Description:Inhibition of recombinant C-terminal His-tagged/N-terminal GST-tagged human EGFR T790M/C797S/L858R mutant (668 to 1210 residues) extracted from bacul...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 16nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human EGFR T790M/L858R mutant (696 to end residues) extracted from baculovirus infect Sf21 insect cel...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 20nMAssay Description:Inhibition of recombinant wildtype N-terminal GST-tagged human EGFR kinase domain (696 to end residues) extracted from baculovirus infect Sf21 insect...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 29nMAssay Description:Inhibition of recombinant C-terminal His-tagged/N-terminal GST-tagged human EGFR T790M/C797S/L858R mutant (668 to 1210 residues) extracted from bacul...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 30nMAssay Description:Inhibition of recombinant wildtype N-terminal GST-tagged human EGFR kinase domain (696 to end residues) extracted from baculovirus infect Sf21 insect...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 32nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human EGFR T790M/L858R mutant (696 to end residues) extracted from baculovirus infect Sf21 insect cel...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 33nMAssay Description:Inhibition of recombinant C-terminal His-tagged/N-terminal GST-tagged human EGFR T790M/C797S/L858R mutant (668 to 1210 residues) extracted from bacul...More data for this Ligand-Target Pair
Affinity DataIC50: 33nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human EGFR T790M/L858R mutant (696 to end residues) extracted from baculovirus infect Sf21 insect cel...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 36nMAssay Description:Inhibition of recombinant C-terminal His-tagged/N-terminal GST-tagged human EGFR T790M/C797S/L858R mutant (668 to 1210 residues) extracted from bacul...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 42nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human EGFR T790M/L858R mutant (696 to end residues) extracted from baculovirus infect Sf21 insect cel...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 45nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human EGFR 19del/T790M/C797S mutant (668 to end residues) extracted from Sf9 insect cells incubated f...More data for this Ligand-Target Pair
Affinity DataIC50: 64nMAssay Description:Inhibition of recombinant wildtype N-terminal GST-tagged human EGFR kinase domain (696 to end residues) extracted from baculovirus infect Sf21 insect...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 71nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human EGFR 19del/T790M/C797S mutant (668 to end residues) extracted from Sf9 insect cells incubated f...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 73nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human EGFR T790M/L858R mutant (696 to end residues) extracted from baculovirus infect Sf21 insect cel...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 81nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human EGFR T790M/L858R mutant (696 to end residues) extracted from baculovirus infect Sf21 insect cel...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 82nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human EGFR T790M/L858R mutant (696 to end residues) extracted from baculovirus infect Sf21 insect cel...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 84nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human EGFR T790M/L858R mutant (696 to end residues) extracted from baculovirus infect Sf21 insect cel...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 111nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human EGFR T790M/L858R mutant (696 to end residues) extracted from baculovirus infect Sf21 insect cel...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 113nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human EGFR 19del/T790M/C797S mutant (668 to end residues) extracted from Sf9 insect cells incubated f...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 122nMAssay Description:Inhibition of recombinant C-terminal His-tagged/N-terminal GST-tagged human EGFR T790M/C797S/L858R mutant (668 to 1210 residues) extracted from bacul...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 129nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human EGFR T790M/L858R mutant (696 to end residues) extracted from baculovirus infect Sf21 insect cel...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 130nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human EGFR 19del/T790M/C797S mutant (668 to end residues) extracted from Sf9 insect cells incubated f...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 132nMAssay Description:Inhibition of recombinant wildtype N-terminal GST-tagged human EGFR kinase domain (696 to end residues) extracted from baculovirus infect Sf21 insect...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 135nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human EGFR T790M/L858R mutant (696 to end residues) extracted from baculovirus infect Sf21 insect cel...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 141nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human EGFR 19del/T790M/C797S mutant (668 to end residues) extracted from Sf9 insect cells incubated f...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 145nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human EGFR T790M/L858R mutant (696 to end residues) extracted from baculovirus infect Sf21 insect cel...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 145nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human EGFR 19del/T790M/C797S mutant (668 to end residues) extracted from Sf9 insect cells incubated f...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 145nMAssay Description:Inhibition of recombinant wildtype N-terminal GST-tagged human EGFR kinase domain (696 to end residues) extracted from baculovirus infect Sf21 insect...More data for this Ligand-Target Pair
Affinity DataIC50: 146nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human EGFR 19del/T790M/C797S mutant (668 to end residues) extracted from Sf9 insect cells incubated f...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 146nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human EGFR 19del/T790M/C797S mutant (668 to end residues) extracted from Sf9 insect cells incubated f...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 150nMAssay Description:Inhibition of recombinant C-terminal His-tagged/N-terminal GST-tagged human EGFR T790M/C797S/L858R mutant (668 to 1210 residues) extracted from bacul...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 159nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human EGFR 19del/T790M/C797S mutant (668 to end residues) extracted from Sf9 insect cells incubated f...More data for this Ligand-Target Pair
Ligand Info






3D Structure (crystal)













