Compile Data Set for Download or QSAR
Report error Found 58 Enz. Inhib. hit(s) with all data for entry = 50022672
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The Second Affiliated Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 144315BDBM144315(US8969336, 577 | US8969336, 547 | Gilteritinib | U...)
Affinity DataIC50: 0.290nMAssay Description:Inhibition of VEGFR2 by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details PubMedPDB3D3D Structure (crystal)
TargetTyrosine-protein kinase receptor UFO(Human)
The Second Affiliated Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 144315BDBM144315(US8969336, 577 | US8969336, 547 | Gilteritinib | U...)
Affinity DataIC50: 0.730nMAssay Description:Inhibition of VEGFR2 by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details PubMed
TargetFibroblast growth factor receptor 1(Human)
The Second Affiliated Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50525939BDBM50525939(Balversa | Erdafitinib | Jnj-42756493)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of VEGFR2 by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details PubMed
TargetFibroblast growth factor receptor 2(Human)
The Second Affiliated Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 161389BDBM161389(US9108973, 2 | US10124003, Ref. Ex. Compound 3 | U...)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of VEGFR2 by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details PubMedPDB3D3D Structure (crystal)
TargetFibroblast growth factor receptor 3(Human)
The Second Affiliated Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 161389BDBM161389(US9108973, 2 | US10124003, Ref. Ex. Compound 3 | U...)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of VEGFR2 by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details PubMed
TargetFibroblast growth factor receptor 1(Human)
The Second Affiliated Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 161389BDBM161389(US9108973, 2 | US10124003, Ref. Ex. Compound 3 | U...)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of VEGFR2 by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details PubMedPDB3D3D Structure (crystal)
TargetFibroblast growth factor receptor 2(Human)
The Second Affiliated Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50525939BDBM50525939(Balversa | Erdafitinib | Jnj-42756493)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of VEGFR2 by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details PubMed
TargetFibroblast growth factor receptor 3(Human)
The Second Affiliated Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50525939BDBM50525939(Balversa | Erdafitinib | Jnj-42756493)
Affinity DataIC50: 3nMAssay Description:Inhibition of VEGFR2 by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details PubMed
TargetFibroblast growth factor receptor 4(Human)
The Second Affiliated Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 161389BDBM161389(US9108973, 2 | US10124003, Ref. Ex. Compound 3 | U...)
Affinity DataIC50: 4.70nMAssay Description:Inhibition of VEGFR2 by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details PubMed
TargetFibroblast growth factor receptor 4(Human)
The Second Affiliated Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50525939BDBM50525939(Balversa | Erdafitinib | Jnj-42756493)
Affinity DataIC50: 5.70nMAssay Description:Inhibition of VEGFR2 by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The Second Affiliated Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50493042BDBM50493042(Akn-028)
Affinity DataIC50: 6nMAssay Description:Inhibition of VEGFR2 by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details PubMed
TargetEndothelin-1 receptor(Human)
The Second Affiliated Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50532593BDBM50532593(ZD-4054 | ZD4054 | Zibotentan)
Affinity DataKi:  13nMAssay Description:Inhibition of VEGFR2 by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details PubMedPDB3D3D Structure (crystal)
TargetFibroblast growth factor receptor 1(Human)
The Second Affiliated Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 6190BDBM6190(CHEMBL189584 | 3-tert-butyl-1-(2-{[4-(diethylamino...)
Affinity DataIC50: 25nMAssay Description:Inhibition of VEGFR2 by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details PubMed
TargetFibroblast growth factor receptor 2(Human)
The Second Affiliated Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50493042BDBM50493042(Akn-028)
Affinity DataIC50: 120nMAssay Description:Inhibition of VEGFR2 by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details PubMed
TargetFibroblast growth factor receptor 2(Human)
The Second Affiliated Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50483568BDBM50483568(CHEMBL6102515)
Affinity DataIC50: 150nMAssay Description:Inhibition of VEGFR2 by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details PubMed
TargetFibroblast growth factor receptor 4(Human)
The Second Affiliated Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50483568BDBM50483568(CHEMBL6102515)
Affinity DataIC50: 270nMAssay Description:Inhibition of VEGFR2 by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details PubMed
TargetFibroblast growth factor receptor 2(Human)
The Second Affiliated Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50483566BDBM50483566(CHEMBL6078359)
Affinity DataIC50: 380nMAssay Description:Inhibition of VEGFR2 by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details PubMed
TargetFibroblast growth factor receptor 2(Human)
The Second Affiliated Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50483571BDBM50483571(CHEMBL6078050)
Affinity DataIC50: 380nMAssay Description:Inhibition of VEGFR2 by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details PubMed
TargetFibroblast growth factor receptor 3(Human)
The Second Affiliated Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50483570BDBM50483570(CHEMBL6074472)
Affinity DataIC50: 450nMAssay Description:Inhibition of VEGFR2 by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details PubMed
TargetFibroblast growth factor receptor 3(Human)
The Second Affiliated Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50483565BDBM50483565(CHEMBL6078164)
Affinity DataIC50: 480nMAssay Description:Inhibition of VEGFR2 by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details PubMed
TargetFibroblast growth factor receptor 3(Human)
The Second Affiliated Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50483571BDBM50483571(CHEMBL6078050)
Affinity DataIC50: 490nMAssay Description:Inhibition of VEGFR2 by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details PubMed
TargetFibroblast growth factor receptor 3(Human)
The Second Affiliated Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50483568BDBM50483568(CHEMBL6102515)
Affinity DataIC50: 520nMAssay Description:Inhibition of VEGFR2 by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details PubMed
TargetFibroblast growth factor receptor 4(Human)
The Second Affiliated Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50483571BDBM50483571(CHEMBL6078050)
Affinity DataIC50: 540nMAssay Description:Inhibition of VEGFR2 by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details PubMed
TargetFibroblast growth factor receptor 2(Human)
The Second Affiliated Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50483570BDBM50483570(CHEMBL6074472)
Affinity DataIC50: 550nMAssay Description:Inhibition of VEGFR2 by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details PubMed
TargetFibroblast growth factor receptor 3(Human)
The Second Affiliated Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50483566BDBM50483566(CHEMBL6078359)
Affinity DataIC50: 550nMAssay Description:Inhibition of VEGFR2 by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details PubMed
TargetFibroblast growth factor receptor 2(Human)
The Second Affiliated Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50483565BDBM50483565(CHEMBL6078164)
Affinity DataIC50: 600nMAssay Description:Inhibition of VEGFR2 by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details PubMed
TargetFibroblast growth factor receptor 1(Human)
The Second Affiliated Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50483569BDBM50483569(CHEMBL6120894)
Affinity DataIC50: 630nMAssay Description:Antagonist activity at human estrogen receptor beta assessed as inhibition of agonist-induced protein interaction with steroid receptor co-activator ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details PubMed
TargetFibroblast growth factor receptor 2(Human)
The Second Affiliated Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50483573BDBM50483573(CHEMBL6077990)
Affinity DataIC50: 630nMAssay Description:Inhibition of VEGFR2 by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details PubMed
TargetFibroblast growth factor receptor 1(Human)
The Second Affiliated Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50483566BDBM50483566(CHEMBL6078359)
Affinity DataIC50: 650nMAssay Description:Antagonist activity at human estrogen receptor beta assessed as inhibition of agonist-induced protein interaction with steroid receptor co-activator ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details PubMed
TargetFibroblast growth factor receptor 2(Human)
The Second Affiliated Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50483569BDBM50483569(CHEMBL6120894)
Affinity DataIC50: 650nMAssay Description:Inhibition of VEGFR2 by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details PubMed
TargetFibroblast growth factor receptor 1(Human)
The Second Affiliated Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50483571BDBM50483571(CHEMBL6078050)
Affinity DataIC50: 720nMAssay Description:Inhibition of human CRTH2 receptor assessed as LTD4-mediated intracellular calcium mobilization by cell-based aequorin luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details PubMed
TargetFibroblast growth factor receptor 4(Human)
The Second Affiliated Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50483565BDBM50483565(CHEMBL6078164)
Affinity DataIC50: 720nMAssay Description:Inhibition of VEGFR2 by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details PubMed
TargetFibroblast growth factor receptor 3(Human)
The Second Affiliated Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50483567BDBM50483567(CHEMBL6096594)
Affinity DataIC50: 740nMAssay Description:Inhibition of VEGFR2 by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details PubMed
TargetFibroblast growth factor receptor 1(Human)
The Second Affiliated Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50483570BDBM50483570(CHEMBL6074472)
Affinity DataIC50: 740nMAssay Description:Inhibition of dopamine transporter (unknown origin) by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details PubMed
TargetFibroblast growth factor receptor 3(Human)
The Second Affiliated Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50483569BDBM50483569(CHEMBL6120894)
Affinity DataIC50: 750nMAssay Description:Inhibition of VEGFR2 by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details PubMed
TargetFibroblast growth factor receptor 4(Human)
The Second Affiliated Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50483566BDBM50483566(CHEMBL6078359)
Affinity DataIC50: 840nMAssay Description:Inhibition of VEGFR2 by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details PubMed
TargetFibroblast growth factor receptor 1(Human)
The Second Affiliated Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50483568BDBM50483568(CHEMBL6102515)
Affinity DataIC50: 850nMAssay Description:Antagonist activity at human estrogen receptor beta assessed as inhibition of agonist-induced protein interaction with steroid receptor co-activator ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details PubMed
TargetFibroblast growth factor receptor 3(Human)
The Second Affiliated Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50483573BDBM50483573(CHEMBL6077990)
Affinity DataIC50: 880nMAssay Description:Inhibition of VEGFR2 by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details PubMed
TargetFibroblast growth factor receptor 2(Human)
The Second Affiliated Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50483564BDBM50483564(CHEMBL6083029)
Affinity DataIC50: 960nMAssay Description:Inhibition of human ACAT1 expressed in AC29 cells by cell-based fluorescent assay systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details PubMed
TargetFibroblast growth factor receptor 3(Human)
The Second Affiliated Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50483564BDBM50483564(CHEMBL6083029)
Affinity DataIC50: 1.04E+3nMAssay Description:Inhibition of VEGFR2 by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details PubMed
TargetFibroblast growth factor receptor 3(Human)
The Second Affiliated Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50483572BDBM50483572(CHEMBL6078007)
Affinity DataIC50: 1.07E+3nMAssay Description:Inhibition of VEGFR2 by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details PubMed
TargetFibroblast growth factor receptor 2(Human)
The Second Affiliated Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50483572BDBM50483572(CHEMBL6078007)
Affinity DataIC50: 1.09E+3nMAssay Description:Inhibition of VEGFR2 by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details PubMed
TargetFibroblast growth factor receptor 2(Human)
The Second Affiliated Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50483567BDBM50483567(CHEMBL6096594)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of VEGFR2 by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details PubMed
TargetFibroblast growth factor receptor 4(Human)
The Second Affiliated Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50483570BDBM50483570(CHEMBL6074472)
Affinity DataIC50: 1.17E+3nMAssay Description:Inhibition of VEGFR2 by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details PubMed
TargetFibroblast growth factor receptor 1(Human)
The Second Affiliated Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50483573BDBM50483573(CHEMBL6077990)
Affinity DataIC50: 1.18E+3nMAssay Description:Inhibition of human DP receptor assessed as LTD4-mediated intracellular calcium mobilization by cell-based aequorin luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details PubMed
TargetFibroblast growth factor receptor 1(Human)
The Second Affiliated Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50483572BDBM50483572(CHEMBL6078007)
Affinity DataIC50: 1.45E+3nMAssay Description:Inhibition of human IP receptor assessed as LTD4-mediated intracellular calcium mobilization by cell-based aequorin luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details PubMed
TargetFibroblast growth factor receptor 1(Human)
The Second Affiliated Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50483565BDBM50483565(CHEMBL6078164)
Affinity DataIC50: 1.50E+3nMAssay Description:Antagonist activity at human estrogen receptor beta assessed as inhibition of agonist-induced protein interaction with steroid receptor co-activator ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details PubMed
TargetFibroblast growth factor receptor 4(Human)
The Second Affiliated Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50483573BDBM50483573(CHEMBL6077990)
Affinity DataIC50: 1.61E+3nMAssay Description:Inhibition of VEGFR2 by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details PubMed
TargetFibroblast growth factor receptor 1(Human)
The Second Affiliated Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50483564BDBM50483564(CHEMBL6083029)
Affinity DataIC50: 1.72E+3nMAssay Description:Antagonist activity at human estrogen receptor beta assessed as inhibition of agonist-induced protein interaction with steroid receptor co-activator ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details PubMed
TargetFibroblast growth factor receptor 4(Human)
The Second Affiliated Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50483572BDBM50483572(CHEMBL6078007)
Affinity DataIC50: 1.74E+3nMAssay Description:Inhibition of VEGFR2 by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2026
Entry Details PubMed
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