Compile Data Set for Download or QSAR
Report error Found 72 Enz. Inhib. hit(s) with all data for entry = 50022773
TargetNAD-dependent protein deacylase sirtuin-6(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654151BDBM50654151(CHEMBL6120377)
Affinity DataIC50: 5.68E+3nMAssay Description:Inhibition of Nav1.5 by cell based whole-cell voltage clamp electrophysiology assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654151BDBM50654151(CHEMBL6120377)
Affinity DataIC50: 5.81E+3nMAssay Description:Agonist activity at human ghrelin receptor by cell based BACMAM FLIPR assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654146BDBM50654146(CHEMBL6103529)
Affinity DataIC50: 6.74E+3nMAssay Description:Agonist activity at human ghrelin receptor by cell based BACMAM FLIPR assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654138BDBM50654138(CHEMBL6151119)
Affinity DataIC50: 7.51E+3nMAssay Description:Agonist activity at human ghrelin receptor by cell based BACMAM FLIPR assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50005711BDBM50005711(GNF-Pf-1011 | CHEBI:46024 | TRICHOSTATIN | Trichos...)
Affinity DataIC50: 7.88E+3nMAssay Description:Agonist activity at human ghrelin receptor by cell based BACMAM FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654127BDBM50654127(CHEMBL6144963)
Affinity DataIC50: 7.97E+3nMAssay Description:Agonist activity at mu1-opioid receptor (unknown origin) by cell-based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654158BDBM50654158(CHEMBL6146343)
Affinity DataIC50: 8.85E+3nMAssay Description:Agonist activity at human ghrelin receptor by cell based BACMAM FLIPR assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654154BDBM50654154(CHEMBL6148720)
Affinity DataIC50: 9.05E+3nMAssay Description:Agonist activity at human ghrelin receptor by cell based BACMAM FLIPR assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654143BDBM50654143(CHEMBL6102875)
Affinity DataIC50: 9.47E+3nMAssay Description:Agonist activity at human ghrelin receptor by cell based BACMAM FLIPR assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654152BDBM50654152(CHEMBL6091963)
Affinity DataIC50: 1.11E+4nMAssay Description:Agonist activity at human ghrelin receptor by cell based BACMAM FLIPR assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654159BDBM50654159(CHEMBL6132631)
Affinity DataIC50: 1.11E+4nMAssay Description:Agonist activity at human ghrelin receptor by cell based BACMAM FLIPR assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654145BDBM50654145(CHEMBL6133480)
Affinity DataIC50: 1.14E+4nMAssay Description:Agonist activity at human ghrelin receptor by cell based BACMAM FLIPR assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654117BDBM50654117(CHEMBL6146976)
Affinity DataIC50: 1.25E+4nMAssay Description:Agonist activity at GAL4-fused PPARalpha assessed as transcriptional activity by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654122BDBM50654122(CHEMBL6133554)
Affinity DataIC50: 1.34E+4nMAssay Description:Inhibition of human thrombin-mediated platelet aggregation in cell-based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654140BDBM50654140(CHEMBL6150337)
Affinity DataIC50: 1.37E+4nMAssay Description:Agonist activity at human ghrelin receptor by cell based BACMAM FLIPR assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654153BDBM50654153(CHEMBL6150689)
Affinity DataIC50: 1.43E+4nMAssay Description:Agonist activity at human ghrelin receptor by cell based BACMAM FLIPR assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654139BDBM50654139(CHEMBL6146266)
Affinity DataIC50: 1.51E+4nMAssay Description:Agonist activity at human ghrelin receptor by cell based BACMAM FLIPR assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetNAD-dependent protein deacylase sirtuin-6(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654151BDBM50654151(CHEMBL6120377)
Affinity DataKd:  1.65E+4nMAssay Description:Inhibition of Nav1.5 by cell based whole-cell voltage clamp electrophysiology assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654141BDBM50654141(CHEMBL6151291)
Affinity DataIC50: 1.70E+4nMAssay Description:Agonist activity at human ghrelin receptor by cell based BACMAM FLIPR assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654112BDBM50654112(CHEMBL6134211)
Affinity DataIC50: 1.95E+4nMAssay Description:Agonist activity at GAL4-fused PPARalpha assessed as transcriptional activity by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654142BDBM50654142(CHEMBL6133031)
Affinity DataIC50: 2.26E+4nMAssay Description:Agonist activity at human ghrelin receptor by cell based BACMAM FLIPR assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654160BDBM50654160(CHEMBL6103342)
Affinity DataIC50: 2.43E+4nMAssay Description:Antagonist activity at human adrenergic alpha1A receptor assessed as intracellular calcium luminescence by cell based aequorin assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654155BDBM50654155(CHEMBL6101858)
Affinity DataIC50: 2.52E+4nMAssay Description:Agonist activity at human ghrelin receptor by cell based BACMAM FLIPR assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654150BDBM50654150(CHEMBL6103351)
Affinity DataIC50: 3.63E+4nMAssay Description:Agonist activity at human ghrelin receptor by cell based BACMAM FLIPR assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654136BDBM50654136(CHEMBL6102224)
Affinity DataIC50: 3.99E+4nMAssay Description:Agonist activity at human ghrelin receptor by cell based BACMAM FLIPR assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654135BDBM50654135(CHEMBL6134080)
Affinity DataIC50: 4.36E+4nMAssay Description:Agonist activity at human ghrelin receptor by cell based BACMAM FLIPR assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654137BDBM50654137(CHEMBL6144261)
Affinity DataIC50: 4.63E+4nMAssay Description:Agonist activity at human ghrelin receptor by cell based BACMAM FLIPR assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654148BDBM50654148(CHEMBL6141774)
Affinity DataIC50: 5.25E+4nMAssay Description:Agonist activity at human ghrelin receptor by cell based BACMAM FLIPR assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654149BDBM50654149(CHEMBL6134149)
Affinity DataIC50: 5.45E+4nMAssay Description:Agonist activity at human ghrelin receptor by cell based BACMAM FLIPR assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654157BDBM50654157(CHEMBL6102959)
Affinity DataIC50: 5.62E+4nMAssay Description:Agonist activity at human ghrelin receptor by cell based BACMAM FLIPR assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654128BDBM50654128(CHEMBL6102927)
Affinity DataIC50: 5.62E+4nMAssay Description:Agonist activity at FXR (unknown origin) measured after 16 hrs in presence of CCF4-AM dye by cell-based GeneBlazer FRET assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50017342BDBM50017342(CHEMBL1588664)
Affinity DataIC50: 9.17E+4nMAssay Description:Agonist activity at human ghrelin receptor by cell based BACMAM FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654170BDBM50654170(CHEMBL6102062)
Affinity DataIC50: 1.00E+5nMAssay Description:Positive allosteric modulation of calcium sensing receptor by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654171BDBM50654171(CHEMBL6109006)
Affinity DataIC50: 1.00E+5nMAssay Description:Positive allosteric modulation of calcium sensing receptor by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654168BDBM50654168(CHEMBL6149946)
Affinity DataIC50: 1.00E+5nMAssay Description:Positive allosteric modulation of calcium sensing receptor by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654169BDBM50654169(CHEMBL6151062)
Affinity DataIC50: 1.00E+5nMAssay Description:Positive allosteric modulation of calcium sensing receptor by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654156BDBM50654156(CHEMBL6120526)
Affinity DataIC50: 1.00E+5nMAssay Description:Agonist activity at human ghrelin receptor by cell based BACMAM FLIPR assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654172BDBM50654172(CHEMBL6101841)
Affinity DataIC50: 1.00E+5nMAssay Description:Positive allosteric modulation of calcium sensing receptor by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654162BDBM50654162(CHEMBL6148242)
Affinity DataIC50: 1.00E+5nMAssay Description:Positive allosteric modulation of calcium sensing receptor by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654163BDBM50654163(CHEMBL6096611)
Affinity DataIC50: 1.00E+5nMAssay Description:Positive allosteric modulation of calcium sensing receptor by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654166BDBM50654166(CHEMBL6103275)
Affinity DataIC50: 1.00E+5nMAssay Description:Positive allosteric modulation of calcium sensing receptor by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654167BDBM50654167(CHEMBL6102100)
Affinity DataIC50: 1.00E+5nMAssay Description:Positive allosteric modulation of calcium sensing receptor by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654164BDBM50654164(CHEMBL6134349)
Affinity DataIC50: 1.00E+5nMAssay Description:Positive allosteric modulation of calcium sensing receptor by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654147BDBM50654147(CHEMBL6114895)
Affinity DataIC50: 1.00E+5nMAssay Description:Agonist activity at human ghrelin receptor by cell based BACMAM FLIPR assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654165BDBM50654165(CHEMBL6150316)
Affinity DataIC50: 1.00E+5nMAssay Description:Positive allosteric modulation of calcium sensing receptor by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654115BDBM50654115(CHEMBL6147923)
Affinity DataIC50: 1.00E+5nMAssay Description:Agonist activity at GAL4-fused PPARalpha assessed as transcriptional activity by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654124BDBM50654124(CHEMBL6149278)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of PI3Kdelta by cell-based proliferation assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654114BDBM50654114(CHEMBL6142966)
Affinity DataIC50: 1.00E+5nMAssay Description:Agonist activity at GAL4-fused PPARalpha assessed as transcriptional activity by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654116BDBM50654116(CHEMBL6149372)
Affinity DataIC50: 1.00E+5nMAssay Description:Agonist activity at GAL4-fused PPARalpha assessed as transcriptional activity by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654119BDBM50654119(CHEMBL6103485)
Affinity DataIC50: 1.00E+5nMAssay Description:Agonist activity at GAL4-fused PPARalpha assessed as transcriptional activity by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
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