Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50022785
TargetHistone deacetylase 1(Human)
University of Kalyani

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654276BDBM50654276(CHEMBL6092022)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of chymotrypsin-like activity of proteasome beta-5 subunit in HEK293 cells using Suc-LLVY-Glo as substrate incubated for 2 hrs prior to su...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetHistone deacetylase 1(Human)
University of Kalyani

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654277BDBM50654277(CHEMBL6146119)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of chymotrypsin-like activity of proteasome beta-5 subunit in HEK293 cells using Suc-LLVY-Glo as substrate incubated for 2 hrs prior to su...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetHistone deacetylase 4(Human)
University of Kalyani

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50446481BDBM50446481(CHEMBL3110004 | US10011611, TMP269 | US10722597, C...)
Affinity DataIC50: 3.5nMAssay Description:Inhibition of DAAO (unknown origin) by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetHistone deacetylase 6(Human)
University of Kalyani

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50005711BDBM50005711(GNF-Pf-1011 | CHEBI:46024 | TRICHOSTATIN | Trichos...)
Affinity DataIC50: 4.70nMAssay Description:Antagonist activity at mouse urotensin2 receptor assessed as inhibition of urotensin2-stimulated Ca2+ mobilization by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetHistone deacetylase 1(Human)
University of Kalyani

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50005711BDBM50005711(GNF-Pf-1011 | CHEBI:46024 | TRICHOSTATIN | Trichos...)
Affinity DataIC50: 7.70nMAssay Description:Inhibition of chymotrypsin-like activity of proteasome beta-5 subunit in HEK293 cells using Suc-LLVY-Glo as substrate incubated for 2 hrs prior to su...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetHistone deacetylase 1(Human)
University of Kalyani

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654279BDBM50654279(CHEMBL6146427)
Affinity DataIC50: 12nMAssay Description:Displacement of [125I]-glucagon-cex from human glucagon receptor by cell based assay in presence of 0.2% bovine serum albuminMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetHistone deacetylase 1(Human)
University of Kalyani

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531377BDBM50531377(FR-235222 | CHEMBL513595)
Affinity DataIC50: 20nMAssay Description:Displacement of [125I]-glucagon-cex from human glucagon receptor by cell based assay in presence of 0.2% bovine serum albuminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetHistone deacetylase 1(Human)
University of Kalyani

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50588306BDBM50588306(CHEMBL474318)
Affinity DataIC50: 30nMAssay Description:Inhibition of DAAO (unknown origin) by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetHistone deacetylase 1(Human)
University of Kalyani

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50588310BDBM50588310(CHEMBL473512)
Affinity DataIC50: 330nMAssay Description:Inhibition of DAAO (unknown origin) by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetHistone deacetylase 6(Human)
University of Kalyani

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654276BDBM50654276(CHEMBL6092022)
Affinity DataIC50: 1.10E+3nMAssay Description:Antagonist activity at rat urotensin2 receptor assessed as inhibition of urotensin2-stimulated Ca2+ mobilization by cell-based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetHistone deacetylase 1(Human)
University of Kalyani

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654276BDBM50654276(CHEMBL6092022)
Affinity DataIC50: 1.10E+3nMAssay Description:Displacement of [125I]-glucagon-cex from human glucagon receptor by cell based assay in presence of 0.2% bovine serum albuminMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetHistone deacetylase 1(Human)
University of Kalyani

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654277BDBM50654277(CHEMBL6146119)
Affinity DataKi:  5.65E+3nMAssay Description:Antagonist activity at mouse urotensin2 receptor assessed as inhibition of urotensin2-stimulated Ca2+ mobilization by cell-based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetHistone deacetylase 1(Human)
University of Kalyani

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654278BDBM50654278(CHEMBL5180408)
Affinity DataKi:  1.12E+4nMAssay Description:Displacement of [125I]-glucagon-cex from human glucagon receptor by cell based assay in presence of 0.2% bovine serum albuminMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetHistone deacetylase 1(Human)
University of Kalyani

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654277BDBM50654277(CHEMBL6146119)
Affinity DataKi:  1.58E+4nMAssay Description:Displacement of [125I]-glucagon-cex from human glucagon receptor by cell based assay in presence of 0.2% bovine serum albuminMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetHistone deacetylase 1(Human)
University of Kalyani

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654278BDBM50654278(CHEMBL5180408)
Affinity DataKi:  2.21E+4nMAssay Description:Displacement of [125I]-glucagon-cex from human glucagon receptor by cell based assay in presence of 0.2% bovine serum albuminMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetHistone deacetylase 6(Human)
University of Kalyani

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654277BDBM50654277(CHEMBL6146119)
Affinity DataIC50: 3.19E+5nMAssay Description:Antagonist activity at rat urotensin2 receptor assessed as inhibition of urotensin2-stimulated Ca2+ mobilization by cell-based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed
TargetHistone deacetylase 4(Human)
University of Kalyani

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50654277BDBM50654277(CHEMBL6146119)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of DAAO (unknown origin) by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/4/2026
Entry Details PubMed