Report error Found 117 Enz. Inhib. hit(s) with all data for entry = 50022903
TargetEpidermal growth factor receptor(Human)
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 0.0100nMAssay Description:Inhibition of wild type EGFR (unknown origin)More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 0.0200nMAssay Description:Inhibition of wild type EGFR (unknown origin)More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 0.0300nMAssay Description:Inhibition of EGFR L858R/T790M/C797S triple mutant (unknown origin)More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 0.0500nMAssay Description:Inhibition of wild type EGFR (unknown origin)More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 0.0600nMAssay Description:Inhibition of EGFR del19/T790M/C797S triple mutant (unknown origin) in presence of ATP by FRET assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 0.0600nMAssay Description:Inhibition of human recombinant EGFR L858R/T790M/C797S triple mutant by TR-FRET assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 0.0600nMAssay Description:Inhibition of EGFR del19/T790M/C797S triple mutant (unknown origin) in presence of ATP by FRET assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 0.0700nMAssay Description:Inhibition of EGFR del19/T790M/C797S triple mutant (unknown origin) in presence of ATP by FRET assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 0.0800nMAssay Description:Inhibition of human recombinant EGFR L858R/T790M/C797S triple mutant by TR-FRET assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 0.0800nMAssay Description:Inhibition of EGFR del19/T790M/C797S triple mutant (unknown origin) in presence of ATP by FRET assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 0.0800nMAssay Description:Inhibition of EGFR L858R/T790M/C797S triple mutant (unknown origin)More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 0.0900nMAssay Description:Inhibition of EGFR del19/T790M/C797S triple mutant (unknown origin) in presence of ATP by FRET assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 0.0900nMAssay Description:Inhibition of human recombinant EGFR L858R/T790M/C797S triple mutant by TR-FRET assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 0.100nMAssay Description:Inhibition of EGFR L858R/T790M/C797S triple mutant (unknown origin)More data for this Ligand-Target Pair
Ligand Info
TargetEpidermal growth factor receptor(Human)
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 0.100nMAssay Description:Inhibition of wild type EGFR (unknown origin)More data for this Ligand-Target Pair
Ligand Info
TargetEpidermal growth factor receptor(Human)
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 0.110nMAssay Description:Inhibition of EGFR del19/T790M/C797S triple mutant (unknown origin) in presence of ATP by FRET assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 0.120nMAssay Description:Inhibition of human recombinant EGFR L858R/T790M/C797S triple mutant by TR-FRET assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 0.150nMAssay Description:Inhibition of EGFR del19/T790M/C797S triple mutant (unknown origin) in presence of ATP by FRET assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 0.150nMAssay Description:Inhibition of human recombinant EGFR L858R/T790M/C797S triple mutant by TR-FRET assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 0.150nMAssay Description:Inhibition of human recombinant EGFR L858R/T790M/C797S triple mutant by TR-FRET assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 0.190nMAssay Description:Inhibition of EGFR del19/T790M/C797S triple mutant (unknown origin) in presence of ATP by FRET assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Inhibition of EGFR del19/T790M/C797S triple mutant (unknown origin) in presence of ATP by FRET assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Inhibition of EGFR del19/T790M/C797S triple mutant (unknown origin) in presence of ATP by FRET assayMore data for this Ligand-Target Pair
Ligand Info
TargetEpidermal growth factor receptor(Human)
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Inhibition of EGFR del19/T790M/C797S triple mutant (unknown origin) in presence of ATP by FRET assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 0.210nMAssay Description:Inhibition of EGFR del19/T790M/C797S triple mutant (unknown origin) in presence of ATP by FRET assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 0.230nMAssay Description:Inhibition of EGFR del19/T790M/C797S triple mutant (unknown origin) in presence of ATP by FRET assayMore data for this Ligand-Target Pair
Ligand Info
TargetEpidermal growth factor receptor(Human)
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 0.280nMAssay Description:Inhibition of EGFR L858R/T790M/C797S triple mutant (unknown origin)More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:Inhibition of EGFR L858R/T790M/C797S triple mutant (unknown origin)More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:Inhibition of EGFR del19/T790M/C797S triple mutant (unknown origin) in presence of ATP by FRET assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 0.310nMAssay Description:Inhibition of human recombinant EGFR L858R/T790M/C797S triple mutant by TR-FRET assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 0.320nMAssay Description:Inhibition of EGFR del19/T790M/C797S triple mutant (unknown origin) in presence of ATP by FRET assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 0.330nMAssay Description:Inhibition of EGFR del19/T790M/C797S triple mutant (unknown origin) in presence of ATP by FRET assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 0.340nMAssay Description:Inhibition of human recombinant EGFR L858R/T790M/C797S triple mutant by TR-FRET assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 0.350nMAssay Description:Inhibition of wild type EGFR (unknown origin)More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 0.400nMAssay Description:Inhibition of EGFR L858R/T790M/C797S triple mutant (unknown origin)More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 0.430nMAssay Description:Inhibition of human recombinant EGFR L858R/T790M/C797S triple mutant by TR-FRET assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Inhibition of EGFR L858R/T790M/C797S triple mutant (unknown origin)More data for this Ligand-Target Pair
Ligand Info
TargetEpidermal growth factor receptor(Human)
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Inhibition of EGFR L858R/T790M/C797S triple mutant (unknown origin)More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Inhibition of wild type EGFR (unknown origin)More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 0.570nMAssay Description:Inhibition of EGFR del19/T790M/C797S triple mutant (unknown origin) in presence of ATP by FRET assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 0.600nMAssay Description:Inhibition of EGFR L858R/T790M/C797S triple mutant (unknown origin)More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 0.610nMAssay Description:Inhibition of wild type EGFR (unknown origin)More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 0.640nMAssay Description:Inhibition of EGFR L858R/T790M/C797S triple mutant (unknown origin)More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 0.650nMAssay Description:Inhibition of EGFR del19/T790M/C797S triple mutant (unknown origin) in presence of ATP by FRET assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 0.700nMAssay Description:Inhibition of EGFR del19/T790M/C797S triple mutant (unknown origin) in presence of ATP by FRET assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 0.700nMAssay Description:Inhibition of EGFR L858R/T790M/C797S triple mutant (unknown origin)More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 0.700nMAssay Description:Inhibition of EGFR L858R/T790M/C797S triple mutant (unknown origin)More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 0.810nMAssay Description:Inhibition of human recombinant EGFR L858R/T790M/C797S triple mutant by TR-FRET assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of wild type EGFR (unknown origin)More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
R. C. Patel Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of wild type EGFR (unknown origin)More data for this Ligand-Target Pair

3D Structure (crystal)
































