Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50022727
LigandChemical structure of BindingDB Monomer ID 50653638BDBM50653638(CHEMBL6078250)
Affinity DataIC50: 150nMAssay Description:Displacement of [3H]-N-methyl-scopolamine from human muscarinic M3 receptor after 6 hrs by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50653630BDBM50653630(CHEMBL6091763)
Affinity DataIC50: 160nMAssay Description:Antagonist activity at human mGlu5 receptor assessed as inhibition of glutamate-induced calcium flux by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50653635BDBM50653635(CHEMBL6101903)
Affinity DataIC50: 260nMAssay Description:Antagonist activity at human mGlu5 receptor assessed as inhibition of glutamate-induced calcium flux by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50653634BDBM50653634(CHEMBL6101800)
Affinity DataIC50: 380nMAssay Description:Antagonist activity at human mGlu5 receptor assessed as inhibition of glutamate-induced calcium flux by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50653636BDBM50653636(CHEMBL6120267)
Affinity DataIC50: 480nMAssay Description:Antagonist activity at human mGlu5 receptor assessed as inhibition of glutamate-induced calcium flux by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50653632BDBM50653632(CHEMBL6102809)
Affinity DataIC50: 490nMAssay Description:Antagonist activity at human mGlu5 receptor assessed as inhibition of glutamate-induced calcium flux by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50653637BDBM50653637(CHEMBL6142517)
Affinity DataIC50: 560nMAssay Description:Displacement of [3H]-N-methyl-scopolamine from human muscarinic M3 receptor after 6 hrs by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50653640BDBM50653640(CHEMBL6078142)
Affinity DataIC50: 890nMAssay Description:Displacement of [3H]-N-methyl-scopolamine from human muscarinic M3 receptor after 6 hrs by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50653639BDBM50653639(CHEMBL6134377)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [3H]-N-methyl-scopolamine from human muscarinic M3 receptor after 6 hrs by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50653631BDBM50653631(CHEMBL6082935)
Affinity DataIC50: 1.43E+3nMAssay Description:Antagonist activity at human mGlu5 receptor assessed as inhibition of glutamate-induced calcium flux by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50653641BDBM50653641(CHEMBL6078466)
Affinity DataIC50: 1.93E+3nMAssay Description:Displacement of [3H]-N-methyl-scopolamine from human muscarinic M3 receptor after 6 hrs by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50653633BDBM50653633(CHEMBL6134131)
Affinity DataIC50: 2.60E+3nMAssay Description:Antagonist activity at human mGlu5 receptor assessed as inhibition of glutamate-induced calcium flux by cell based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/3/2026
Entry Details
PubMed