Compile Data Set for Download or QSAR
Report error Found 30 Enz. Inhib. hit(s) with all data for entry = 50023669
TargetBromodomain-containing protein 4(Human)
Chongqing University of Arts and Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 220447BDBM220447(US9296741, 36 | US10633379, Compound X)
Affinity DataIC50: 0.730nMAssay Description:Inhibition of His-tagged BRD4-BD1 (unknown origin) incubated for 30 mins in presence of ATP by Alphascreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Chongqing University of Arts and Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666503BDBM50666503(CHEMBL6169467)
Affinity DataIC50: 2nMAssay Description:Inhibition of His-tagged BRD4-BD2 (unknown origin) incubated for 30 mins in presence of ATP by Alphascreen assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Chongqing University of Arts and Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666499BDBM50666499(CHEMBL6170616)
Affinity DataIC50: 7.80nMAssay Description:Inhibition of His-tagged BRD4-BD1 (unknown origin) incubated for 30 mins in presence of ATP by Alphascreen assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Chongqing University of Arts and Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666501BDBM50666501(CHEMBL6177583)
Affinity DataIC50: 11nMAssay Description:Inhibition of His-tagged BRD4-BD1 (unknown origin) incubated for 30 mins in presence of ATP by Alphascreen assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Chongqing University of Arts and Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666502BDBM50666502(CHEMBL6177568)
Affinity DataIC50: 11nMAssay Description:Inhibition of His-tagged BRD4-BD1 (unknown origin) incubated for 30 mins in presence of ATP by Alphascreen assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Chongqing University of Arts and Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666500BDBM50666500(CHEMBL6177833)
Affinity DataIC50: 15nMAssay Description:Inhibition of His-tagged BRD4-BD1 (unknown origin) incubated for 30 mins in presence of ATP by Alphascreen assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetBromodomain-containing protein 2(Human)
Chongqing University of Arts and Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666503BDBM50666503(CHEMBL6169467)
Affinity DataIC50: 18nMAssay Description:Inhibition of His-tagged BRD2-BD1 (unknown origin) incubated for 30 mins in presence of ATP by Alphascreen assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Chongqing University of Arts and Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666503BDBM50666503(CHEMBL6169467)
Affinity DataIC50: 19nMAssay Description:Inhibition of His-tagged BRD4-BD1 (unknown origin) incubated for 30 mins in presence of ATP by Alphascreen assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50507818BDBM50507818(CHEMBL4450504)
Affinity DataIC50: 23nMAssay Description:Inhibition of p110delta/p85alpha (unknown origin) incubated for 2 hrs in presence of ATP by ADP-kinaseGlo reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetBromodomain-containing protein 3(Human)
Chongqing University of Arts and Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666503BDBM50666503(CHEMBL6169467)
Affinity DataIC50: 32nMAssay Description:Inhibition of His-tagged BRD3-BD1 (unknown origin) incubated for 30 mins in presence of ATP by Alphascreen assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetBromodomain testis-specific protein(Human)
Chongqing University of Arts and Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666503BDBM50666503(CHEMBL6169467)
Affinity DataIC50: 46nMAssay Description:Inhibition of His-tagged BRDT-BD1 (unknown origin) incubated for 30 mins in presence of ATP by Alphascreen assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50666500BDBM50666500(CHEMBL6177833)
Affinity DataIC50: 96nMAssay Description:Inhibition of p110delta/p85alpha (unknown origin) incubated for 2 hrs in presence of ATP by ADP-kinaseGlo reagent based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50427453BDBM50427453(CHEMBL2322228 | US9505780, 28 | US10308662, Compou...)
Affinity DataIC50: 106nMAssay Description:Inhibition of p110alpha/p85alpha (unknown origin) incubated for 2 hrs in presence of ATP by ADP-kinaseGlo reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50666501BDBM50666501(CHEMBL6177583)
Affinity DataIC50: 108nMAssay Description:Inhibition of p110delta/p85alpha (unknown origin) incubated for 2 hrs in presence of ATP by ADP-kinaseGlo reagent based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50666503BDBM50666503(CHEMBL6169467)
Affinity DataIC50: 112nMAssay Description:Inhibition of p110delta/p85alpha (unknown origin) incubated for 2 hrs in presence of ATP by ADP-kinaseGlo reagent based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Human)
Chongqing University of Arts and Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50427453BDBM50427453(CHEMBL2322228 | US9505780, 28 | US10308662, Compou...)
Affinity DataIC50: 129nMAssay Description:Inhibition of PI3Kbeta (unknown origin) incubated for 2 hrs in presence of ATP by ADP-kinaseGlo reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50427453BDBM50427453(CHEMBL2322228 | US9505780, 28 | US10308662, Compou...)
Affinity DataIC50: 158nMAssay Description:Inhibition of p110delta/p85alpha (unknown origin) incubated for 2 hrs in presence of ATP by ADP-kinaseGlo reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50666502BDBM50666502(CHEMBL6177568)
Affinity DataIC50: 206nMAssay Description:Inhibition of p110delta/p85alpha (unknown origin) incubated for 2 hrs in presence of ATP by ADP-kinaseGlo reagent based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Chongqing University of Arts and Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50427453BDBM50427453(CHEMBL2322228 | US9505780, 28 | US10308662, Compou...)
Affinity DataIC50: 235nMAssay Description:Inhibition of His-tagged BRD4-BD2 (unknown origin) incubated for 30 mins in presence of ATP by Alphascreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Human)
Chongqing University of Arts and Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50427453BDBM50427453(CHEMBL2322228 | US9505780, 28 | US10308662, Compou...)
Affinity DataIC50: 251nMAssay Description:Inhibition of PI3Kgamma (unknown origin) incubated for 2 hrs in presence of ATP by ADP-kinaseGlo reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetBromodomain-containing protein 3(Human)
Chongqing University of Arts and Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50427453BDBM50427453(CHEMBL2322228 | US9505780, 28 | US10308662, Compou...)
Affinity DataIC50: 303nMAssay Description:Inhibition of His-tagged BRD3-BD1 (unknown origin) incubated for 30 mins in presence of ATP by Alphascreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Chongqing University of Arts and Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50427453BDBM50427453(CHEMBL2322228 | US9505780, 28 | US10308662, Compou...)
Affinity DataIC50: 312nMAssay Description:Inhibition of His-tagged BRD4-BD1 (unknown origin) incubated for 30 mins in presence of ATP by Alphascreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetBromodomain-containing protein 2(Human)
Chongqing University of Arts and Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50427453BDBM50427453(CHEMBL2322228 | US9505780, 28 | US10308662, Compou...)
Affinity DataIC50: 383nMAssay Description:Inhibition of His-tagged BRD2-BD1 (unknown origin) incubated for 30 mins in presence of ATP by Alphascreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50666499BDBM50666499(CHEMBL6170616)
Affinity DataIC50: 464nMAssay Description:Inhibition of p110delta/p85alpha (unknown origin) incubated for 2 hrs in presence of ATP by ADP-kinaseGlo reagent based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Chongqing University of Arts and Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50427453BDBM50427453(CHEMBL2322228 | US9505780, 28 | US10308662, Compou...)
Affinity DataIC50: 599nMAssay Description:Inhibition of mTOR (unknown origin) incubated for 2 hrs in presence of ATP by ADP-kinaseGlo reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Human)
Chongqing University of Arts and Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666503BDBM50666503(CHEMBL6169467)
Affinity DataIC50: 915nMAssay Description:Inhibition of PI3Kgamma (unknown origin) incubated for 2 hrs in presence of ATP by ADP-kinaseGlo reagent based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetBromodomain testis-specific protein(Human)
Chongqing University of Arts and Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50427453BDBM50427453(CHEMBL2322228 | US9505780, 28 | US10308662, Compou...)
Affinity DataIC50: 1.23E+3nMAssay Description:Inhibition of His-tagged BRDT-BD1 (unknown origin) incubated for 30 mins in presence of ATP by Alphascreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Human)
Chongqing University of Arts and Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666503BDBM50666503(CHEMBL6169467)
Affinity DataIC50: 4.75E+3nMAssay Description:Inhibition of PI3Kbeta (unknown origin) incubated for 2 hrs in presence of ATP by ADP-kinaseGlo reagent based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50666503BDBM50666503(CHEMBL6169467)
Affinity DataIC50: 6.13E+3nMAssay Description:Inhibition of p110alpha/p85alpha (unknown origin) incubated for 2 hrs in presence of ATP by ADP-kinaseGlo reagent based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Chongqing University of Arts and Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666503BDBM50666503(CHEMBL6169467)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of mTOR (unknown origin) incubated for 2 hrs in presence of ATP by ADP-kinaseGlo reagent based assayMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed