Report error Found 40 Enz. Inhib. hit(s) with all data for entry = 50023432
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKd: 7.30nMAssay Description:Binding affinity to PDK1 (unknown origin) assessed as dissociation constant by surface plasmon resonance assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 40nMAssay Description:Inhibition of 14-3-3beta (unknown origin) extracted from Escherichia coli BL21 (DE3) incubated for 60 mins by fluorescence based analysisMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 430nMAssay Description:Inhibition of 14-3-3beta (unknown origin) extracted from Escherichia coli BL21 (DE3) incubated for 60 mins by fluorescence based analysisMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of ERalpha (unknown origin)More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of ERalpha (unknown origin)More data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKd: 1.40E+3nMAssay Description:Binding affinity to PDK1 (unknown origin) assessed as dissociation constant by surface plasmon resonance assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of 14-3-3beta (unknown origin) extracted from Escherichia coli BL21 (DE3) incubated for 60 mins by fluorescence based analysisMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of ERalpha (unknown origin)More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of ERalpha (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPDB
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of ERalpha (unknown origin)More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of ERalpha (unknown origin)More data for this Ligand-Target Pair
Ligand Info
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKd: 6.00E+3nMAssay Description:Binding affinity to PDK1 (unknown origin) assessed as dissociation constant by surface plasmon resonance assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 6.20E+3nMAssay Description:Inhibition of 14-3-3beta (unknown origin) extracted from Escherichia coli BL21 (DE3) incubated for 60 mins by fluorescence based analysisMore data for this Ligand-Target Pair
Ligand Info
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKd: 6.40E+3nMAssay Description:Binding affinity to PDK1 (unknown origin) assessed as dissociation constant by surface plasmon resonance assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of human full length 14-3-3beta expressed in Escherichia coli BL21 (DE3) by fluorescence based analysisMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of ERalpha (unknown origin)More data for this Ligand-Target Pair
Ligand Info
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKd: 9.30E+3nMAssay Description:Binding affinity to PDK1 (unknown origin) assessed as dissociation constant by surface plasmon resonance assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of 14-3-3beta (unknown origin) extracted from Escherichia coli BL21 (DE3) incubated for 60 mins by fluorescence based analysisMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.46E+4nMAssay Description:Inhibition of 14-3-3beta (unknown origin) extracted from Escherichia coli BL21 (DE3) incubated for 60 mins by fluorescence based analysisMore data for this Ligand-Target Pair
Ligand Info
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKd: 1.50E+4nMAssay Description:Binding affinity to PDK1 (unknown origin) assessed as dissociation constant by surface plasmon resonance assayMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKd: 1.60E+4nMAssay Description:Binding affinity to PDK1 (unknown origin) assessed as dissociation constant by surface plasmon resonance assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of ERalpha (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPDB
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of ERalpha (unknown origin)More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibition of ERalpha (unknown origin)More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 3.61E+4nMAssay Description:Inhibition of 14-3-3beta (unknown origin) extracted from Escherichia coli BL21 (DE3) incubated for 60 mins by fluorescence based analysisMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 3.70E+4nMAssay Description:Inhibition of human full length 14-3-3beta expressed in Escherichia coli BL21 (DE3) by fluorescence based analysisMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of ERalpha (unknown origin)More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 6.50E+4nMAssay Description:Inhibition of human full length 14-3-3beta expressed in Escherichia coli BL21 (DE3) by fluorescence based analysisMore data for this Ligand-Target Pair
Ligand InfoPDB
Affinity DataIC50: 7.70E+4nMAssay Description:Inhibition of ERalpha (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPDB
TargetRAF proto-oncogene serine/threonine-protein kinase(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 7.70E+4nMAssay Description:Inhibition of C-RAF (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPDB
Affinity DataIC50: 8.00E+4nMAssay Description:Inhibition of ERalpha (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPDB
Affinity DataIC50: 8.10E+4nMAssay Description:Inhibition of human full length 14-3-3beta expressed in Escherichia coli BL21 (DE3) by fluorescence based analysisMore data for this Ligand-Target Pair
Ligand InfoPDB
TargetRAF proto-oncogene serine/threonine-protein kinase(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 8.10E+4nMAssay Description:Inhibition of C-RAF (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPDB
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of 14-3-3beta (unknown origin) extracted from Escherichia coli BL21 (DE3) incubated for 60 mins by fluorescence based analysisMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.16E+5nMAssay Description:Inhibition of ERalpha (unknown origin)More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.51E+5nMAssay Description:Inhibition of 14-3-3beta (unknown origin) extracted from Escherichia coli BL21 (DE3) incubated for 60 mins by fluorescence based analysisMore data for this Ligand-Target Pair
Ligand Info
TargetRAF proto-oncogene serine/threonine-protein kinase(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 2.46E+5nMAssay Description:Inhibition of C-RAF (unknown origin)More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 2.50E+5nMAssay Description:Inhibition of human full length 14-3-3beta expressed in Escherichia coli BL21 (DE3) by fluorescence based analysisMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 4.26E+5nMAssay Description:Inhibition of ERalpha (unknown origin)More data for this Ligand-Target Pair
Ligand Info
TargetRAF proto-oncogene serine/threonine-protein kinase(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 4.26E+5nMAssay Description:Inhibition of C-RAF (unknown origin)More data for this Ligand-Target Pair
Ligand Info


































