Report error Found 64 Enz. Inhib. hit(s) with all data for entry = 50023307
Affinity DataIC50: 10nMAssay Description:Inhibition of human NETMore data for this Ligand-Target Pair
Ligand InfoPDB
Affinity DataIC50: 60nMAssay Description:Inhibition of DAT (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPDB
Affinity DataIC50: 280nMAssay Description:Inhibition of human GluN1/GluN2A NMDA receptor expressed in HEK293 cells assessed as reduction in glutamate induced current at -70 mV holding potenti...More data for this Ligand-Target Pair
Affinity DataIC50: 280nMAssay Description:Inhibition of human GluN1/GluN2A NMDA receptor expressed in HEK293 cells assessed as reduction in glutamate induced current at -70 mV holding potenti...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 280nMAssay Description:Inhibition of human GluN1/GluN2A NMDA receptor expressed in HEK293 cells assessed as reduction in glutamate induced current at -70 mV holding potenti...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 300nMAssay Description:Inhibition of human GluN1/GluN2A NMDA receptor expressed in HEK293 cells assessed as reduction in glutamate induced current at -70 mV holding potenti...More data for this Ligand-Target Pair
Affinity DataIC50: 340nMAssay Description:Inhibition of human GluN1/GluN2A NMDA receptor expressed in HEK293 cells assessed as reduction in glutamate induced current at -70 mV holding potenti...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 430nMAssay Description:Antagonist activity at human GluN1/GluN2A NMDA receptor expressed in HEK293 cells assessed as reduction in glutamate induced current at -70 mV holdin...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 500nMAssay Description:Inhibition of human GluN1/GluN2A NMDA receptor expressed in HEK293 cells assessed as reduction in glutamate induced current at -70 mV holding potenti...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.04E+3nMAssay Description:Antagonist activity at human GluN1/GluN2A NMDA receptor expressed in HEK293 cells assessed as reduction in glutamate induced current at -70 mV holdin...More data for this Ligand-Target Pair
Affinity DataIC50: 1.22E+3nMAssay Description:Inhibition of human NETMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of human GluN1/GluN2A NMDA receptor expressed in HEK293 cells assessed as reduction in glutamate induced current at -70 mV holding potenti...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.81E+3nMAssay Description:Inhibition of human GluN1/GluN2A NMDA receptor expressed in HEK293 cells assessed as reduction in glutamate induced current at -70 mV holding potenti...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 2.17E+3nMAssay Description:Inhibition of human GluN1/GluN2A NMDA receptor expressed in HEK293 cells assessed as reduction in glutamate induced current at -70 mV holding potenti...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of human GluN1/GluN2A NMDA receptor expressed in HEK293 cells assessed as reduction in glutamate induced current at -70 mV holding potenti...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 2.84E+3nMAssay Description:Inhibition of human NETMore data for this Ligand-Target Pair
Affinity DataIC50: 2.96E+3nMAssay Description:Inhibition of human GluN1/GluN2A NMDA receptor expressed in HEK293 cells assessed as reduction in glutamate induced current at -70 mV holding potenti...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 2.96E+3nMAssay Description:Inhibition of human GluN1/GluN2A NMDA receptor expressed in HEK293 cells assessed as reduction in glutamate induced current at -70 mV holding potenti...More data for this Ligand-Target Pair
Affinity DataIC50: 3.01E+3nMAssay Description:Inhibition of human GluN1/GluN2A NMDA receptor expressed in HEK293 cells assessed as reduction in glutamate induced current at -70 mV holding potenti...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 3.07E+3nMAssay Description:Inhibition of human GluN1/GluN2A NMDA receptor expressed in HEK293 cells assessed as reduction in glutamate induced current at -70 mV holding potenti...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 3.50E+3nMAssay Description:Antagonist activity at human GluN1/GluN2A NMDA receptor expressed in HEK293 cells assessed as reduction in glutamate induced current at -70 mV holdin...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 4.71E+3nMAssay Description:Inhibition of human NETMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 4.77E+3nMAssay Description:Inhibition of human GluN1/GluN2A NMDA receptor expressed in HEK293 cells assessed as reduction in glutamate induced current at -70 mV holding potenti...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of human NETMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 4.92E+3nMAssay Description:Inhibition of human GluN1/GluN2A NMDA receptor expressed in HEK293 cells assessed as reduction in glutamate induced current at -70 mV holding potenti...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 5.18E+3nMAssay Description:Inhibition of human GluN1/GluN2A NMDA receptor expressed in HEK293 cells assessed as reduction in glutamate induced current at -70 mV holding potenti...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 5.72E+3nMAssay Description:Inhibition of human NETMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 6.23E+3nMAssay Description:Inhibition of human GluN1/GluN2A NMDA receptor expressed in HEK293 cells assessed as reduction in glutamate induced current at -70 mV holding potenti...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 9.23E+3nMAssay Description:Inhibition of human GluN1/GluN2A NMDA receptor expressed in HEK293 cells assessed as reduction in glutamate induced current at -70 mV holding potenti...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 9.87E+3nMAssay Description:Inhibition of human GluN1/GluN2A NMDA receptor expressed in HEK293 cells assessed as reduction in glutamate induced current at -70 mV holding potenti...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.06E+4nMAssay Description:Inhibition of human NETMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of human SERTMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.65E+4nMAssay Description:Inhibition of human NETMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of human SERTMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.73E+4nMAssay Description:Inhibition of human NETMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.99E+4nMAssay Description:Inhibition of human GluN1/GluN2A NMDA receptor expressed in HEK293 cells assessed as reduction in glutamate induced current at -70 mV holding potenti...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibition of human SERTMore data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of human GluN1/GluN2A NMDA receptor expressed in HEK293 cells assessed as reduction in glutamate induced current at -70 mV holding potenti...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of human GluN1/GluN2A NMDA receptor expressed in HEK293 cells assessed as reduction in glutamate induced current at -70 mV holding potenti...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 9.00E+4nMAssay Description:Inhibition of human SERTMore data for this Ligand-Target Pair
Ligand InfoPDB
Affinity DataIC50: 1.23E+5nMAssay Description:Inhibition of human SERTMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.30E+5nMAssay Description:Inhibition of human SERTMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.48E+5nMAssay Description:Inhibition of human SERTMore data for this Ligand-Target Pair
Affinity DataIC50: 2.38E+5nMAssay Description:Inhibition of human SERTMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 2.70E+5nMAssay Description:Inhibition of human SERTMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 3.33E+5nMAssay Description:Inhibition of human SERTMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 3.35E+5nMAssay Description:Inhibition of human SERTMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 4.35E+5nMAssay Description:Inhibition of human SERTMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 4.63E+5nMAssay Description:Inhibition of human SERTMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 5.77E+5nMAssay Description:Inhibition of human SERTMore data for this Ligand-Target Pair
Ligand Info

3D Structure (crystal)
























