Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50023205
TargetHistone acetyltransferase p300/Hypoxia-inducible factor 1-alpha(Human)
Institute of Science Tokyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50524839BDBM50524839(CHEMBL4466328)
Affinity DataIC50: 51nMAssay Description:Inhibition of HIF-1alpha(unknown origin)/human p300 CH1 domain (323 to 423 residues) PPI extracted from Escherichia coli incubated for 1 hr by Spectr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetHistone acetyltransferase p300(Human)
Institute of Science Tokyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50524839BDBM50524839(CHEMBL4466328)
Affinity DataIC50: 530nMAssay Description:Inhibition of p300 CH1 domain (unknown origin) by tryptophan fluorescence spectroscopy analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetHistone acetyltransferase p300/Hypoxia-inducible factor 1-alpha(Human)
Institute of Science Tokyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50447758BDBM50447758(CHEBI:9287 | NSC-45383 | Nigrin | Rufocromomycin |...)
Affinity DataIC50: 1.38E+3nMAssay Description:Inhibition of HIF-1alpha(unknown origin)/human p300 CH1 domain (323 to 423 residues) PPI extracted from Escherichia coli incubated for 1 hr by Spectr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetHistone acetyltransferase p300/Hypoxia-inducible factor 1-alpha(Human)
Institute of Science Tokyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50400094BDBM50400094(CHEMBL427092)
Affinity DataIC50: 4.40E+3nMAssay Description:Inhibition of HIF-1alpha/p300 PPI (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed