Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50023554
TargetUbiquitin carboxyl-terminal hydrolase 7(Human)
Shanghai Institute of Materia Medica
Curated by ChEMBL
Shanghai Institute of Materia Medica
Curated by ChEMBL
Affinity DataKd: 2.42E+4nMAssay Description:Activation of USP7 C223S mutant catalytic domain (unknown origin) assessed as Kd of K48-linked di-ubiquitin at 0.5 mM by isothermal titration calorim...More data for this Ligand-Target Pair
TargetUbiquitin carboxyl-terminal hydrolase 7(Human)
Shanghai Institute of Materia Medica
Curated by ChEMBL
Shanghai Institute of Materia Medica
Curated by ChEMBL
Affinity DataEC50: 3.22E+4nMAssay Description:Activation of USP7 catalytic domain (208 to 560 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) assessed as Ub-AMC hydrolysis prei...More data for this Ligand-Target Pair
TargetUbiquitin carboxyl-terminal hydrolase 7(Human)
Shanghai Institute of Materia Medica
Curated by ChEMBL
Shanghai Institute of Materia Medica
Curated by ChEMBL
Affinity DataEC50: 6.10E+4nMAssay Description:Activation of USP7 catalytic domain (208 to 560 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) assessed as Ub-AMC hydrolysis prei...More data for this Ligand-Target Pair
TargetUbiquitin carboxyl-terminal hydrolase 7(Human)
Shanghai Institute of Materia Medica
Curated by ChEMBL
Shanghai Institute of Materia Medica
Curated by ChEMBL
Affinity DataKd: 4.91E+5nMAssay Description:Binding affinity to [15N,2H]-labeled USP7 catalytic domain (208 to 560 residues) (unknown origin) by [1H,15N] TROSY-HSQC titration based NMR spectros...More data for this Ligand-Target Pair


3D Structure (crystal)