Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50023756
TargetGTPase KRas(Human)
Risen (Shanghai) Pharma Tech Co., Ltd.

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50579601BDBM50579601(CHEMBL4858364 | US11453683, Example 252 | US202302...)
Affinity DataIC50: 2.30nMAssay Description:Binding affinity to 6 His-tagged GDP-loaded human KRAS G12D mutant assessed as GDP-GTP exchange preincubated for 30 mins followed by GTP addition for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetGTPase KRas(Human)
Risen (Shanghai) Pharma Tech Co., Ltd.

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50667829BDBM50667829(CHEMBL6190724)
Affinity DataIC50: 4nMAssay Description:Binding affinity to 6 His-tagged GDP-loaded human KRAS G12D mutant assessed as GDP-GTP exchange preincubated for 30 mins followed by GTP addition for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetGTPase KRas(Human)
Risen (Shanghai) Pharma Tech Co., Ltd.

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50667830BDBM50667830(CHEMBL6189990)
Affinity DataIC50: 6.30nMAssay Description:Binding affinity to 6 His-tagged GDP-loaded human KRAS G12D mutant assessed as GDP-GTP exchange preincubated for 30 mins followed by GTP addition for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed