Report error Found 193 Enz. Inhib. hit(s) with all data for entry = 50023357
Affinity DataIC50: 4nMAssay Description:Inhibition of JNK2 (unknown origin) using ATF2 as substrate incubated for 60 mins by PamQuinase assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 10(Human)
Eberhard Karls Universitat Tubingen
Curated by ChEMBL
Eberhard Karls Universitat Tubingen
Curated by ChEMBL
Affinity DataKd: 5.5nMAssay Description:Binding affinity to JNK3 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 10(Human)
Eberhard Karls Universitat Tubingen
Curated by ChEMBL
Eberhard Karls Universitat Tubingen
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibition of JNK3 (unknown origin)More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 10(Human)
Eberhard Karls Universitat Tubingen
Curated by ChEMBL
Eberhard Karls Universitat Tubingen
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibition of JNK3 (unknown origin) using ATF2 as substrate incubated for 60 mins by PamQuinase assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 10(Human)
Eberhard Karls Universitat Tubingen
Curated by ChEMBL
Eberhard Karls Universitat Tubingen
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibition of JNK3 (unknown origin) using ATF2 as substrate incubated for 60 mins by PamQuinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Inhibition of JNK2 (unknown origin) using ATF2 as substrate incubated for 60 mins by PamQuinase assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 10(Human)
Eberhard Karls Universitat Tubingen
Curated by ChEMBL
Eberhard Karls Universitat Tubingen
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Inhibition of JNK3 (unknown origin) using ATF2 as substrate incubated for 60 mins by PamQuinase assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 10(Human)
Eberhard Karls Universitat Tubingen
Curated by ChEMBL
Eberhard Karls Universitat Tubingen
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Inhibition of JNK3 (unknown origin) using ATF2 as substrate incubated for 60 mins by PamQuinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibition of JNK2 (unknown origin) using ATF2 as substrate incubated for 60 mins by PamQuinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inhibition of JNK2 (unknown origin) using ATF2 as substrate incubated for 60 mins by PamQuinase assayMore data for this Ligand-Target Pair
Affinity DataKd: 15nMAssay Description:Binding affinity to JNK2 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 10(Human)
Eberhard Karls Universitat Tubingen
Curated by ChEMBL
Eberhard Karls Universitat Tubingen
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Inhibition of JNK3 (unknown origin) using ATF2 as substrate incubated for 60 mins by PamQuinase assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 10(Human)
Eberhard Karls Universitat Tubingen
Curated by ChEMBL
Eberhard Karls Universitat Tubingen
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Inhibition of JNK3 (unknown origin) using ATF2 as substrate incubated for 60 mins by PamQuinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Inhibition of JNK2 (unknown origin) using ATF2 as substrate incubated for 60 mins by PamQuinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Time dependent inhibition of JNK2 (unknown origin) using sulfonamido-oxine fluorophore as substrate preincubated for 60 mins in presence of ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:Inhibition of JNK2 (unknown origin) using ATF2 as substrate incubated for 60 mins by PamQuinase assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 10(Human)
Eberhard Karls Universitat Tubingen
Curated by ChEMBL
Eberhard Karls Universitat Tubingen
Curated by ChEMBL
Affinity DataIC50: 29nMAssay Description:Inhibition of JNK3 (unknown origin) using ATF2 as substrate incubated for 60 mins by PamQuinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 31nMAssay Description:Inhibition of JNK2 (unknown origin) using ATF2 as substrate incubated for 60 mins by PamQuinase assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 10(Human)
Eberhard Karls Universitat Tubingen
Curated by ChEMBL
Eberhard Karls Universitat Tubingen
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Inhibition of JNK3 (unknown origin) using ATF2 as substrate incubated for 60 mins by PamQuinase assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 10(Human)
Eberhard Karls Universitat Tubingen
Curated by ChEMBL
Eberhard Karls Universitat Tubingen
Curated by ChEMBL
Affinity DataIC50: 38nMAssay Description:Inhibition of JNK3 (unknown origin) using ATF2 as substrate incubated for 60 mins by PamQuinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 38nMAssay Description:Inhibition of JNK2 (unknown origin) using ATF2 as substrate incubated for 60 mins by PamQuinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 38nMAssay Description:Inhibition of JNK2 (unknown origin) using ATF2 as substrate incubated for 60 mins by PamQuinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 38nMAssay Description:Inhibition of JNK2 (unknown origin) using ATF2 as substrate incubated for 60 mins by PamQuinase assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 10(Human)
Eberhard Karls Universitat Tubingen
Curated by ChEMBL
Eberhard Karls Universitat Tubingen
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Time dependent inhibition of JNK3 (unknown origin) using sulfonamido-oxine fluorophore as substrate preincubated for 60 mins in presence of ATPMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 10(Human)
Eberhard Karls Universitat Tubingen
Curated by ChEMBL
Eberhard Karls Universitat Tubingen
Curated by ChEMBL
Affinity DataIC50: 45nMAssay Description:Inhibition of JNK3 (unknown origin) using ATF2 as substrate incubated for 60 mins by PamQuinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 49nMAssay Description:Inhibition of JNK1 (unknown origin) using ATF2 as substrate incubated for 60 mins by PamQuinase assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 10(Human)
Eberhard Karls Universitat Tubingen
Curated by ChEMBL
Eberhard Karls Universitat Tubingen
Curated by ChEMBL
Affinity DataIC50: 52nMAssay Description:Inhibition of JNK3 (unknown origin) using ATF2 as substrate incubated for 60 mins by PamQuinase assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 10(Human)
Eberhard Karls Universitat Tubingen
Curated by ChEMBL
Eberhard Karls Universitat Tubingen
Curated by ChEMBL
Affinity DataIC50: 54nMAssay Description:Inhibition of JNK3 (unknown origin) using ATF2 as substrate incubated for 60 mins by PamQuinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 59nMAssay Description:Inhibition of JNK2 (unknown origin) using ATF2 as substrate incubated for 60 mins by PamQuinase assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 10(Human)
Eberhard Karls Universitat Tubingen
Curated by ChEMBL
Eberhard Karls Universitat Tubingen
Curated by ChEMBL
Affinity DataIC50: 61nMAssay Description:Inhibition of JNK3 (unknown origin) using ATF2 as substrate incubated for 60 mins by PamQuinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 64nMAssay Description:Inhibition of JNK2 (unknown origin) using ATF2 as substrate incubated for 60 mins by PamQuinase assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 10(Human)
Eberhard Karls Universitat Tubingen
Curated by ChEMBL
Eberhard Karls Universitat Tubingen
Curated by ChEMBL
Affinity DataIC50: 64nMAssay Description:Inhibition of JNK3 (unknown origin) using ATF2 as substrate incubated for 60 mins by PamQuinase assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 10(Human)
Eberhard Karls Universitat Tubingen
Curated by ChEMBL
Eberhard Karls Universitat Tubingen
Curated by ChEMBL
Affinity DataIC50: 64nMAssay Description:Inhibition of JNK3 (unknown origin) using ATF2 as substrate incubated for 60 mins by PamQuinase assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 10(Human)
Eberhard Karls Universitat Tubingen
Curated by ChEMBL
Eberhard Karls Universitat Tubingen
Curated by ChEMBL
Affinity DataIC50: 65nMAssay Description:Inhibition of JNK3 (unknown origin) using ATF2 as substrate incubated for 60 mins by PamQuinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Inhibition of JNK2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 73nMAssay Description:Inhibition of JNK2 (unknown origin) using ATF2 as substrate incubated for 60 mins by PamQuinase assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 10(Human)
Eberhard Karls Universitat Tubingen
Curated by ChEMBL
Eberhard Karls Universitat Tubingen
Curated by ChEMBL
Affinity DataIC50: 84nMAssay Description:Inhibition of JNK3 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 87nMAssay Description:Inhibition of JNK2 (unknown origin) using ATF2 as substrate incubated for 60 mins by PamQuinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 88nMAssay Description:Inhibition of JNK2 (unknown origin) using ATF2 as substrate incubated for 60 mins by PamQuinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 102nMAssay Description:Inhibition of JNK2 (unknown origin) using ATF2 as substrate incubated for 60 mins by PamQuinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 111nMAssay Description:Inhibition of JNK1 (unknown origin) using ATF2 as substrate incubated for 60 mins by PamQuinase assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 10(Human)
Eberhard Karls Universitat Tubingen
Curated by ChEMBL
Eberhard Karls Universitat Tubingen
Curated by ChEMBL
Affinity DataIC50: 118nMAssay Description:Inhibition of JNK3 (unknown origin) using ATF2 as substrate incubated for 60 mins by PamQuinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 126nMAssay Description:Inhibition of JNK2 (unknown origin) using ATF2 as substrate incubated for 60 mins by PamQuinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 132nMAssay Description:Inhibition of JNK1 (unknown origin) using ATF2 as substrate incubated for 60 mins by PamQuinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 136nMAssay Description:Inhibition of JNK1 (unknown origin) using ATF2 as substrate incubated for 60 mins by PamQuinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 138nMAssay Description:Inhibition of JNK2 (unknown origin) using ATF2 as substrate incubated for 60 mins by PamQuinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 156nMAssay Description:Inhibition of JNK2 (unknown origin) using ATF2 as substrate incubated for 60 mins by PamQuinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 157nMAssay Description:Inhibition of JNK2 (unknown origin) using ATF2 as substrate incubated for 60 mins by PamQuinase assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 10(Human)
Eberhard Karls Universitat Tubingen
Curated by ChEMBL
Eberhard Karls Universitat Tubingen
Curated by ChEMBL
Affinity DataIC50: 158nMAssay Description:Inhibition of JNK3 (unknown origin) using ATF2 as substrate incubated for 60 mins by PamQuinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 170nMAssay Description:Inhibition of JNK1 (unknown origin) using ATF2 as substrate incubated for 60 mins by PamQuinase assayMore data for this Ligand-Target Pair






















