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Report error Found 58 Enz. Inhib. hit(s) with all data for entry = 50026802
TargetCoagulation factor VII(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272503((2R,3S)-3-Methyl-2-phenylmethanesulfonylamino-pent...)
Affinity DataKi:  15nMAssay Description:Inhibition of human factor 7a-tissue factor complexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCoagulation factor XI(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272558(4-({(1S,2S)-1-[(S)-1-(4-Carbamimidoyl-benzylcarbam...)
Affinity DataKi:  17nMAssay Description:Inhibition of human factor 11aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCoagulation factor VII(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272539(3-({(1S,2S)-1-[(S)-1-(4-Carbamimidoyl-benzylcarbam...)
Affinity DataKi:  18nMAssay Description:Inhibition of human factor 7a-tissue factor complexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCoagulation factor VII(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272576(3-({(1S,2S)-1-[(S)-1-(4-Carbamimidoyl-benzylcarbam...)
Affinity DataKi:  20nMAssay Description:Inhibition of human factor 7a-tissue factor complexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCoagulation factor VII(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272480((S)-2-((2R,3S)-3-Methyl-2-phenylmethanesulfonylami...)
Affinity DataKi:  25nMAssay Description:Inhibition of human factor 7a-tissue factor complexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCoagulation factor VII(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272560(3-({(1S,2R)-1-[(S)-1-(4-Carbamimidoyl-benzylcarbam...)
Affinity DataKi:  30nMAssay Description:Inhibition of human factor 7a-tissue factor complexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCoagulation factor XI(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272539(3-({(1S,2S)-1-[(S)-1-(4-Carbamimidoyl-benzylcarbam...)
Affinity DataKi:  33nMAssay Description:Inhibition of human factor 11aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCoagulation factor VII(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272502((2R,3S)-3-Methyl-2-(propane-1-sulfonylamino)-penta...)
Affinity DataKi:  35nMAssay Description:Inhibition of human factor 7a-tissue factor complexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCoagulation factor VII(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272558(4-({(1S,2S)-1-[(S)-1-(4-Carbamimidoyl-benzylcarbam...)
Affinity DataKi:  35nMAssay Description:Inhibition of human factor 7a-tissue factor complexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCoagulation factor VII(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272537((2R,3R)-N-[(S)-1-(4-Carbamimidoyl-benzylcarbamoyl)...)
Affinity DataKi:  42nMAssay Description:Inhibition of human factor 7a-tissue factor complexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCoagulation factor VII(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272538(2-({(1S,2S)-1-[(S)-1-(4-Carbamimidoyl-benzylcarbam...)
Affinity DataKi:  43nMAssay Description:Inhibition of human factor 7a-tissue factor complexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272503((2R,3S)-3-Methyl-2-phenylmethanesulfonylamino-pent...)
Affinity DataKi:  55nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCoagulation factor VII(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272479((S)-2-[(2R,3S)-3-Methyl-2-(propane-1-sulfonylamino...)
Affinity DataKi:  69nMAssay Description:Inhibition of human factor 7a-tissue factor complexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCoagulation factor VII(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272559(3-({(1S,2R)-1-[(S)-1-(4-Carbamimidoyl-benzylcarbam...)
Affinity DataKi:  74nMAssay Description:Inhibition of human factor 7a-tissue factor complexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCoagulation factor XI(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272538(2-({(1S,2S)-1-[(S)-1-(4-Carbamimidoyl-benzylcarbam...)
Affinity DataKi:  113nMAssay Description:Inhibition of human factor 11aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCoagulation factor VII(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272501((S)-2-((2R,3R)-3-Hydroxy-2-phenylmethanesulfonylam...)
Affinity DataKi:  114nMAssay Description:Inhibition of human factor 7a-tissue factor complexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCoagulation factor XI(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272576(3-({(1S,2S)-1-[(S)-1-(4-Carbamimidoyl-benzylcarbam...)
Affinity DataKi:  115nMAssay Description:Inhibition of human factor 11aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCoagulation factor VII(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272536((2R,3R)-N-[(S)-1-(4-Carbamimidoyl-benzylcarbamoyl)...)
Affinity DataKi:  130nMAssay Description:Inhibition of human factor 7a-tissue factor complexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272480((S)-2-((2R,3S)-3-Methyl-2-phenylmethanesulfonylami...)
Affinity DataKi:  150nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCoagulation factor X(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272503((2R,3S)-3-Methyl-2-phenylmethanesulfonylamino-pent...)
Affinity DataKi:  160nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCoagulation factor VII(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272500((S)-2-[(2R,3R)-3-Hydroxy-2-(propane-1-sulfonylamin...)
Affinity DataKi:  198nMAssay Description:Inhibition of human factor 7a-tissue factor complexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272502((2R,3S)-3-Methyl-2-(propane-1-sulfonylamino)-penta...)
Affinity DataKi:  220nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCoagulation factor XI(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272559(3-({(1S,2R)-1-[(S)-1-(4-Carbamimidoyl-benzylcarbam...)
Affinity DataKi:  259nMAssay Description:Inhibition of human factor 11aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCoagulation factor XI(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272560(3-({(1S,2R)-1-[(S)-1-(4-Carbamimidoyl-benzylcarbam...)
Affinity DataKi:  323nMAssay Description:Inhibition of human factor 11aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCoagulation factor X(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272480((S)-2-((2R,3S)-3-Methyl-2-phenylmethanesulfonylami...)
Affinity DataKi:  330nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272479((S)-2-[(2R,3S)-3-Methyl-2-(propane-1-sulfonylamino...)
Affinity DataKi:  500nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272558(4-({(1S,2S)-1-[(S)-1-(4-Carbamimidoyl-benzylcarbam...)
Affinity DataKi:  680nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCoagulation factor X(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272539(3-({(1S,2S)-1-[(S)-1-(4-Carbamimidoyl-benzylcarbam...)
Affinity DataKi:  685nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272537((2R,3R)-N-[(S)-1-(4-Carbamimidoyl-benzylcarbamoyl)...)
Affinity DataKi:  760nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCoagulation factor X(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272576(3-({(1S,2S)-1-[(S)-1-(4-Carbamimidoyl-benzylcarbam...)
Affinity DataKi:  920nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCoagulation factor X(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272502((2R,3S)-3-Methyl-2-(propane-1-sulfonylamino)-penta...)
Affinity DataKi:  1.50E+3nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCoagulation factor X(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272537((2R,3R)-N-[(S)-1-(4-Carbamimidoyl-benzylcarbamoyl)...)
Affinity DataKi:  1.80E+3nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCoagulation factor X(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272558(4-({(1S,2S)-1-[(S)-1-(4-Carbamimidoyl-benzylcarbam...)
Affinity DataKi:  2.48E+3nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCoagulation factor X(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272479((S)-2-[(2R,3S)-3-Methyl-2-(propane-1-sulfonylamino...)
Affinity DataKi:  2.70E+3nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCoagulation factor X(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272538(2-({(1S,2S)-1-[(S)-1-(4-Carbamimidoyl-benzylcarbam...)
Affinity DataKi:  3.13E+3nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272501((S)-2-((2R,3R)-3-Hydroxy-2-phenylmethanesulfonylam...)
Affinity DataKi:  3.36E+3nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272536((2R,3R)-N-[(S)-1-(4-Carbamimidoyl-benzylcarbamoyl)...)
Affinity DataKi:  3.40E+3nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272576(3-({(1S,2S)-1-[(S)-1-(4-Carbamimidoyl-benzylcarbam...)
Affinity DataKi:  3.85E+3nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272538(2-({(1S,2S)-1-[(S)-1-(4-Carbamimidoyl-benzylcarbam...)
Affinity DataKi:  5.49E+3nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCoagulation factor X(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272560(3-({(1S,2R)-1-[(S)-1-(4-Carbamimidoyl-benzylcarbam...)
Affinity DataKi:  5.70E+3nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272539(3-({(1S,2S)-1-[(S)-1-(4-Carbamimidoyl-benzylcarbam...)
Affinity DataKi:  5.73E+3nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272500((S)-2-[(2R,3R)-3-Hydroxy-2-(propane-1-sulfonylamin...)
Affinity DataKi:  1.33E+4nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCoagulation factor X(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272559(3-({(1S,2R)-1-[(S)-1-(4-Carbamimidoyl-benzylcarbam...)
Affinity DataKi:  1.47E+4nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCoagulation factor X(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272536((2R,3R)-N-[(S)-1-(4-Carbamimidoyl-benzylcarbamoyl)...)
Affinity DataKi:  2.50E+4nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272560(3-({(1S,2R)-1-[(S)-1-(4-Carbamimidoyl-benzylcarbam...)
Affinity DataKi:  2.53E+4nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProthrombin(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272559(3-({(1S,2R)-1-[(S)-1-(4-Carbamimidoyl-benzylcarbam...)
Affinity DataKi:  4.55E+4nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCoagulation factor IX(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272538(2-({(1S,2S)-1-[(S)-1-(4-Carbamimidoyl-benzylcarbam...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human factor 9aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCoagulation factor IX(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272560(3-({(1S,2R)-1-[(S)-1-(4-Carbamimidoyl-benzylcarbam...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human factor 9aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCoagulation factor XII(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272538(2-({(1S,2S)-1-[(S)-1-(4-Carbamimidoyl-benzylcarbam...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human factor 12aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCoagulation factor XII(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272576(3-({(1S,2S)-1-[(S)-1-(4-Carbamimidoyl-benzylcarbam...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human factor 12aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

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