Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50028975
TargetDelta-type opioid receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50001468(deltorphin C | CHEMBL317956 | H-Tyr-D-Ala-Phe-Asp-...)
Affinity DataIC50: 0.110nMAssay Description:Inhibitory activity against Mouse vas deferens smooth muscleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetDelta-type opioid receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50280456({(4S,7R,10S,13R)-13-[(S)-2-Amino-3-(4-hydroxy-phen...)
Affinity DataIC50: 0.230nMAssay Description:Inhibitory activity against Mouse vas deferens smooth muscleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetDelta-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50001468(deltorphin C | CHEMBL317956 | H-Tyr-D-Ala-Phe-Asp-...)
Affinity DataIC50: 0.600nMAssay Description:Binding affinity against delta receptor with [3H][p-Cl-Phe4]-DPDPEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetDelta-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50280456({(4S,7R,10S,13R)-13-[(S)-2-Amino-3-(4-hydroxy-phen...)
Affinity DataIC50: 0.870nMAssay Description:Binding affinity against delta receptor with [3H][p-Cl-Phe4]-DPDPEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetMu-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50001468(deltorphin C | CHEMBL317956 | H-Tyr-D-Ala-Phe-Asp-...)
Affinity DataIC50: 2.90nMAssay Description:Inhibitory activity against Guinea pig ileum smooth muscleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetMu-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50280456({(4S,7R,10S,13R)-13-[(S)-2-Amino-3-(4-hydroxy-phen...)
Affinity DataIC50: 3nMAssay Description:Inhibitory activity against Guinea pig ileum smooth muscleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50280456({(4S,7R,10S,13R)-13-[(S)-2-Amino-3-(4-hydroxy-phen...)
Affinity DataIC50: 5.20nMAssay Description:Binding affinity against Opioid receptor mu 1 with [3H]CTOPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50001468(deltorphin C | CHEMBL317956 | H-Tyr-D-Ala-Phe-Asp-...)
Affinity DataIC50: 2.14E+3nMAssay Description:Binding affinity against Opioid receptor mu 1 with [3H]CTOPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article