Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50029011
TargetThromboxane-A synthase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50280723({6-Fluoro-9-[3-(6-pyridin-3-yl-hex-5-ynyloxy)-benz...)
Affinity DataIC50: 40nMAssay Description:Human microsomal Thromboxane synthase inhibition was determined by inhibiting TXB2 formation from [14C]- labelled arachidonic acidMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetThromboxane-A synthase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50280719({6-Fluoro-9-[3-(5-pyridin-3-yl-pent-4-ynyloxy)-ben...)
Affinity DataIC50: 50nMAssay Description:Human microsomal Thromboxane synthase inhibition was determined by inhibiting TXB2 formation from [14C]- labelled arachidonic acidMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetThromboxane-A synthase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50280720({6-Fluoro-9-[3-(4-pyridin-3-yl-butoxy)-benzyl]-2,3...)
Affinity DataIC50: 100nMAssay Description:Human microsomal Thromboxane synthase inhibition was determined by inhibiting TXB2 formation from [14C]- labelled arachidonic acidMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetThromboxane-A synthase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50280724({6-Fluoro-9-[3-((Z)-5-pyridin-3-yl-pent-4-enyloxy)...)
Affinity DataIC50: 200nMAssay Description:Human microsomal Thromboxane synthase inhibition was determined by inhibiting TXB2 formation from [14C]- labelled arachidonic acidMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetThromboxane-A synthase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50280721({6-Fluoro-9-[3-(5-pyridin-3-yl-pentyloxy)-benzyl]-...)
Affinity DataIC50: 300nMAssay Description:Human microsomal Thromboxane synthase inhibition was determined by inhibiting TXB2 formation from [14C]- labelled arachidonic acidMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetThromboxane-A synthase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50280722({6-Fluoro-9-[4-(6-pyridin-3-yl-hex-5-ynyloxy)-benz...)
Affinity DataIC50: 400nMAssay Description:Human microsomal Thromboxane synthase inhibition was determined by inhibiting TXB2 formation from [14C]- labelled arachidonic acidMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetThromboxane-A synthase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50280726({6-Fluoro-9-[3-(5-pyridin-3-yl-pentyl)-benzyl]-2,3...)
Affinity DataIC50: 500nMAssay Description:Human microsomal Thromboxane synthase inhibition was determined by inhibiting TXB2 formation from [14C]- labelled arachidonic acidMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetThromboxane-A synthase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50280725({6-Fluoro-9-[4-(5-pyridin-3-yl-pent-4-ynyloxy)-ben...)
Affinity DataIC50: 600nMAssay Description:Human microsomal Thromboxane synthase inhibition was determined by inhibiting TXB2 formation from [14C]- labelled arachidonic acidMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article