Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50029140
LigandChemical structure of BindingDB Monomer ID 50062005BDBM50062005(PD-135666 | 3-[2-(2-Adamantan-2-yl-acetylamino)-3-...)
Affinity DataIC50: 0.150nMAssay Description:Inhibition of [125I]CCK-8 to Cholecystokinin type B receptor in the mouse cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50449787BDBM50449787(PD-134308 | CHEMBL2062154)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of [125I]CCK-8 to Cholecystokinin type B receptor in the mouse cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50073729BDBM50073729((R)-3-[(S)-2-(Adamantan-2-yloxycarbonylamino)-3-(1...)
Affinity DataIC50: 2.80nMAssay Description:Inhibition of [125I]CCK-8 binding to Cholecystokinin type A receptor of rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50007446BDBM50007446(CHEMBL335914 | N-{2-[2-(Adamantan-2-yloxycarbonyla...)
Affinity DataIC50: 4.20nMAssay Description:Inhibition of [125I]CCK-8 to Cholecystokinin type B receptor in the mouse cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50061990BDBM50061990((R)-3-[(R)-2-(Adamantan-2-yloxycarbonylamino)-3-(1...)
Affinity DataIC50: 9.30nMAssay Description:Inhibition of [125I]CCK-8 to Cholecystokinin type B receptor in the mouse cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50073727BDBM50073727((S)-3-[(S)-2-(Adamantan-2-yloxycarbonylamino)-3-(1...)
Affinity DataIC50: 13nMAssay Description:Inhibition of [125I]CCK-8 to Cholecystokinin type B receptor in the mouse cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50007442BDBM50007442(CHEMBL337661 | N-{2-[2-(Adamantan-2-yloxycarbonyla...)
Affinity DataIC50: 23nMAssay Description:Inhibition of [125I]CCK-8 to Cholecystokinin type B receptor in the mouse cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50062005BDBM50062005(PD-135666 | 3-[2-(2-Adamantan-2-yl-acetylamino)-3-...)
Affinity DataIC50: 26nMAssay Description:Inhibition of [125I]CCK-8 binding to Cholecystokinin type A receptor of rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50006875BDBM50006875(N-{(S)-2-[(R)-2-(Adamantan-2-yloxycarbonylamino)-3...)
Affinity DataIC50: 43nMAssay Description:Inhibition of [125I]CCK-8 to Cholecystokinin type B receptor in the mouse cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50422043BDBM50422043(CI-988 | PD-137342 | CHEMBL2062144)
Affinity DataIC50: 63nMAssay Description:Inhibition of [125I]CCK-8 to Cholecystokinin type B receptor in the mouse cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50281735BDBM50281735(PD-137337 | N-{(S)-2-[(S)-2-(Adamantan-2-yloxycarb...)
Affinity DataIC50: 160nMAssay Description:Inhibition of [125I]CCK-8 to Cholecystokinin type B receptor in the mouse cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50281734BDBM50281734(PD-138915 | N-{(R)-2-[(S)-2-(Adamantan-2-yloxycarb...)
Affinity DataIC50: 170nMAssay Description:Inhibition of [125I]CCK-8 to Cholecystokinin type B receptor in the mouse cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50281733BDBM50281733(PD-138917 | N-{(S)-2-[(S)-2-(Adamantan-2-yloxycarb...)
Affinity DataIC50: 180nMAssay Description:Inhibition of [125I]CCK-8 to Cholecystokinin type B receptor in the mouse cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50061990BDBM50061990((R)-3-[(R)-2-(Adamantan-2-yloxycarbonylamino)-3-(1...)
Affinity DataIC50: 186nMAssay Description:Inhibition of [125I]CCK-8 binding to Cholecystokinin type A receptor of rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50073729BDBM50073729((R)-3-[(S)-2-(Adamantan-2-yloxycarbonylamino)-3-(1...)
Affinity DataIC50: 259nMAssay Description:Inhibition of [125I]CCK-8 to Cholecystokinin type B receptor in the mouse cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50073727BDBM50073727((S)-3-[(S)-2-(Adamantan-2-yloxycarbonylamino)-3-(1...)
Affinity DataIC50: 539nMAssay Description:Inhibition of [125I]CCK-8 binding to Cholecystokinin type A receptor of rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50281734BDBM50281734(PD-138915 | N-{(R)-2-[(S)-2-(Adamantan-2-yloxycarb...)
Affinity DataIC50: 580nMAssay Description:Inhibition of [125I]CCK-8 binding to Cholecystokinin type A receptor of rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50007442BDBM50007442(CHEMBL337661 | N-{2-[2-(Adamantan-2-yloxycarbonyla...)
Affinity DataIC50: 850nMAssay Description:Inhibition of [125I]CCK-8 binding to Cholecystokinin type A receptor of rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50007446BDBM50007446(CHEMBL335914 | N-{2-[2-(Adamantan-2-yloxycarbonyla...)
Affinity DataIC50: 950nMAssay Description:Inhibition of [125I]CCK-8 binding to Cholecystokinin type A receptor of rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50281735BDBM50281735(PD-137337 | N-{(S)-2-[(S)-2-(Adamantan-2-yloxycarb...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of [125I]CCK-8 binding to Cholecystokinin type A receptor of rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50006875BDBM50006875(N-{(S)-2-[(R)-2-(Adamantan-2-yloxycarbonylamino)-3...)
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of [125I]CCK-8 binding to Cholecystokinin type A receptor of rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50449787BDBM50449787(PD-134308 | CHEMBL2062154)
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of [125I]CCK-8 binding to Cholecystokinin type A receptor of rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50281733BDBM50281733(PD-138917 | N-{(S)-2-[(S)-2-(Adamantan-2-yloxycarb...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of [125I]CCK-8 binding to Cholecystokinin type A receptor of rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50422043BDBM50422043(CI-988 | PD-137342 | CHEMBL2062144)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of [125I]CCK-8 binding to Cholecystokinin type A receptor of rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article