Compile Data Set for Download or QSAR
maximum 50k data
Found 10 Enz. Inhib. hit(s) with all data for entry = 50029152
TargetNeurotensin receptor type 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50281809((S)-2-{(2S,3S)-2-[(S)-2-{[(S)-1-((S)-6-Amino-2-ter...)
Affinity DataKi:  63nMAssay Description:Neurotensin receptor binding affinity by displacement of [3H]- neurotensinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50281812((S)-2-{(2S,3S)-2-[(S)-2-{[(S)-1-((S)-5-Amino-2-ter...)
Affinity DataKi:  82nMAssay Description:Neurotensin receptor binding affinity by displacement of [3H]- neurotensinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50281811((S)-2-{(2S,3S)-2-[(S)-2-[((S)-1-{(S)-2-[(Adamantan...)
Affinity DataKi:  117nMAssay Description:Neurotensin receptor binding affinity by displacement of [3H]- neurotensinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50281807((S)-2-{(2S,3S)-2-[(S)-2-{[(S)-1-((S)-2,6-Diamino-h...)
Affinity DataKi:  688nMAssay Description:Neurotensin receptor binding affinity by displacement of [3H]- neurotensinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50281806((S)-2-{(2S,3S)-2-[(S)-2-{N'-[2-((S)-1-{(S)-2-[(Ada...)
Affinity DataKi:  1.61E+3nMAssay Description:Neurotensin receptor binding affinity by displacement of [3H]- neurotensinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50281810((S)-2-{(2S,3S)-2-[(S)-2-{(E)-3-[(S)-1-((S)-6-Amino...)
Affinity DataKi:  1.63E+3nMAssay Description:Neurotensin receptor binding affinity by displacement of [3H]- neurotensinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50281804((S)-2-{(2S,3S)-2-[(S)-2-(N'-{2-[(S)-1-((S)-5-Amino...)
Affinity DataKi:  2.99E+3nMAssay Description:Neurotensin receptor binding affinity by displacement of [3H]- neurotensinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50281813((S)-2-((2S,3S)-2-{N'-[(S)-3-[((S)-1-{(S)-3-[(Adama...)
Affinity DataKi:  3.86E+3nMAssay Description:Neurotensin receptor binding affinity by displacement of [3H]- neurotensinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50281805((S)-2-((2S,3S)-2-{N'-[(S)-3-[((S)-1-{(S)-2-[(Adama...)
Affinity DataKi:  5.96E+3nMAssay Description:Neurotensin receptor binding affinity by displacement of [3H]- neurotensinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeurotensin receptor type 1(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50281808((S)-2-((2S,3S)-2-{N'-[(S)-3-{[(S)-1-((S)-5-Amino-2...)
Affinity DataKi: >1.00E+4nMAssay Description:Neurotensin receptor binding affinity by displacement of [3H]- neurotensinMore data for this Ligand-Target Pair
In DepthDetails Article