Compile Data Set for Download or QSAR
maximum 50k data
Found 8 Enz. Inhib. hit(s) with all data for entry = 50029218
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50282359(4'-(2-Ethyl-6,8-dimethyl-imidazo[1,2-b]pyridazin-3...)
Affinity DataIC50:  0.800nMAssay Description:In vitro binding affinity of the compound evaluated by its ability to displace the specific binding ligand 125I-SAR1, Ile8-AII from Angiotensin II re...More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50282358(CHEMBL432734 | N-[4'-(2-Ethyl-6,8-dimethyl-imidazo...)
Affinity DataIC50:  1.70nMAssay Description:In vitro binding affinity of the compound evaluated by its ability to displace the specific binding ligand 125I-SAR1, Ile8-AII from Angiotensin II re...More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50282360(2-Ethyl-6,8-dimethyl-3-[2'-(2H-tetrazol-5-yl)-biph...)
Affinity DataIC50:  5.70nMAssay Description:In vitro binding affinity of the compound evaluated by its ability to displace the specific binding ligand 125I-SAR1, Ile8-AII from Angiotensin II re...More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50282361(4'-(2-Ethyl-6,8-dimethyl-imidazo[1,2-b]pyridazin-3...)
Affinity DataIC50: >10nMAssay Description:In vitro binding affinity to AT2 receptor determined by its ability to displace the specific binding ligand [125I]-Sar1, Ile8-AII from AT2 receptor i...More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50282358(CHEMBL432734 | N-[4'-(2-Ethyl-6,8-dimethyl-imidazo...)
Affinity DataIC50: >10nMAssay Description:In vitro binding affinity to AT2 receptor determined by its ability to displace the specific binding ligand [125I]-Sar1, Ile8-AII from AT2 receptor i...More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50282359(4'-(2-Ethyl-6,8-dimethyl-imidazo[1,2-b]pyridazin-3...)
Affinity DataIC50: >10nMAssay Description:In vitro binding affinity to AT2 receptor determined by its ability to displace the specific binding ligand [125I]-Sar1, Ile8-AII from AT2 receptor i...More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50282360(2-Ethyl-6,8-dimethyl-3-[2'-(2H-tetrazol-5-yl)-biph...)
Affinity DataIC50: >10nMAssay Description:In vitro binding affinity at AT2 receptor determined by its ability to displace the specific binding ligand [125I]-Sar1, Ile8-AII from rat brain memb...More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50282361(4'-(2-Ethyl-6,8-dimethyl-imidazo[1,2-b]pyridazin-3...)
Affinity DataIC50:  83nMAssay Description:In vitro binding affinity of the compound evaluated by its ability to displace the specific binding ligand 125I-SAR1, Ile8-AII from Angiotensin II re...More data for this Ligand-Target Pair
In DepthDetails Article