Compile Data Set for Download or QSAR
Report error Found 54 Enz. Inhib. hit(s) with all data for entry = 50029227
TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282470BDBM50282470(Quinazolinone Analog | CHEMBL353037)
Affinity DataIC50: 0.120nMAssay Description:Tested in vitro for binding affinity against Angiotensin II receptor, type 1 in rabbit aortic membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282468BDBM50282468(4'-[2-Butyl-6-(3-isopropyl-ureido)-4-oxo-4H-quinaz...)
Affinity DataIC50: 0.150nMAssay Description:Tested in vitro for binding affinity against Angiotensin II receptor, type 1 in rabbit aortic membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282453BDBM50282453(Quinazolinone Analog | CHEMBL353800)
Affinity DataIC50: 0.150nMAssay Description:Tested in vitro for binding affinity against Angiotensin II receptor, type 1 in rabbit aortic membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282466BDBM50282466(Quinazolinone Analog | CHEMBL354779)
Affinity DataIC50: 0.170nMAssay Description:Tested in vitro for binding affinity against Angiotensin II receptor, type 1 in rabbit aortic membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282472BDBM50282472(Quinazolinone Analog | CHEMBL169221)
Affinity DataIC50: 0.180nMAssay Description:Tested in vitro for binding affinity against Angiotensin II receptor, type 1 in rabbit aortic membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282464BDBM50282464(Quinazolinone Analog | CHEMBL169568)
Affinity DataIC50: 0.180nMAssay Description:Tested in vitro for binding affinity against Angiotensin II receptor, type 1 in rabbit aortic membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282462BDBM50282462(Quinazolinone Analog | CHEMBL352503)
Affinity DataIC50: 0.190nMAssay Description:Tested in vitro for binding affinity against Angiotensin II receptor, type 1 in rabbit aortic membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282455BDBM50282455(Quinazolinone Analog | CHEMBL169967)
Affinity DataIC50: 0.210nMAssay Description:Tested in vitro for binding affinity against Angiotensin II receptor, type 1 in rabbit aortic membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50049181BDBM50049181(2-Butyl-3-(2'-(butyloxycarbonylaminosulphonyl)-bip...)
Affinity DataIC50: 0.240nMAssay Description:Tested in vitro for binding affinity against Angiotensin II receptor, type 1 in rabbit aortic membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282452BDBM50282452(Quinazolinone Analog | CHEMBL169488)
Affinity DataIC50: 0.240nMAssay Description:Tested in vitro for binding affinity against Angiotensin II receptor, type 1 in rabbit aortic membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282460BDBM50282460(Quinazolinone Analog | CHEMBL169968)
Affinity DataIC50: 0.25nMAssay Description:Tested in vitro for binding affinity against Angiotensin II receptor, type 1 in rabbit aortic membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282465BDBM50282465(Quinazolinone Analog | CHEMBL353615)
Affinity DataIC50: 0.25nMAssay Description:Tested in vitro for binding affinity against Angiotensin II receptor, type 1 in rabbit aortic membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282477BDBM50282477(Quinazolinone Analog | CHEMBL168413)
Affinity DataIC50: 0.25nMAssay Description:Tested in vitro for binding affinity against Angiotensin II receptor, type 1 in rabbit aortic membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282461BDBM50282461(Quinazolinone Analog | CHEMBL168490)
Affinity DataIC50: 0.260nMAssay Description:Tested in vitro for binding affinity against Angiotensin II receptor, type 1 in rabbit aortic membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282467BDBM50282467(Quinazolinone Analog | CHEMBL352629)
Affinity DataIC50: 0.320nMAssay Description:Tested in vitro for binding affinity against Angiotensin II receptor, type 1 in rabbit aortic membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282458BDBM50282458(Quinazolinone Analog | CHEMBL352947)
Affinity DataIC50: 0.330nMAssay Description:Tested in vitro for binding affinity against Angiotensin II receptor, type 1 in rabbit aortic membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282469BDBM50282469(Quinazolinone Analog | CHEMBL352502)
Affinity DataIC50: 0.350nMAssay Description:Tested in vitro for binding affinity against Angiotensin II receptor, type 1 in rabbit aortic membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282476BDBM50282476(Quinazolinone Analog | CHEMBL352458)
Affinity DataIC50: 0.360nMAssay Description:Tested in vitro for binding affinity against Angiotensin II receptor, type 1 in rabbit aortic membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282457BDBM50282457(Quinazolinone Analog | CHEMBL169279)
Affinity DataIC50: 0.390nMAssay Description:Tested in vitro for binding affinity against Angiotensin II receptor, type 1 in rabbit aortic membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282463BDBM50282463(Quinazolinone Analog | CHEMBL354080)
Affinity DataIC50: 0.430nMAssay Description:Tested in vitro for binding affinity against Angiotensin II receptor, type 1 in rabbit aortic membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282454BDBM50282454(Quinazolinone Analog | CHEMBL353980)
Affinity DataIC50: 0.550nMAssay Description:Tested in vitro for binding affinity against Angiotensin II receptor, type 1 in rabbit aortic membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282459BDBM50282459(Quinazolinone Analog | CHEMBL169009)
Affinity DataIC50: 0.860nMAssay Description:Tested in vitro for binding affinity against Angiotensin II receptor, type 1 in rabbit aortic membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282471BDBM50282471(N-[3-(2'-Benzoylsulfamoyl-biphenyl-4-ylmethyl)-4-o...)
Affinity DataIC50: 0.990nMAssay Description:Tested in vitro for binding affinity against Angiotensin II receptor, type 1 in rabbit aortic membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282473BDBM50282473(Quinazolinone Analog | CHEMBL354298)
Affinity DataIC50: 1.10nMAssay Description:Tested in vitro for binding affinity against Angiotensin II receptor, type 1 in rabbit aortic membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282458BDBM50282458(Quinazolinone Analog | CHEMBL352947)
Affinity DataIC50: 1.60nMAssay Description:In vitro for binding affinity against angiotensin II receptor type 2 in rat midbrain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282469BDBM50282469(Quinazolinone Analog | CHEMBL352502)
Affinity DataIC50: 2.10nMAssay Description:In vitro for binding affinity against angiotensin II receptor type 2 in rat midbrain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50049181BDBM50049181(2-Butyl-3-(2'-(butyloxycarbonylaminosulphonyl)-bip...)
Affinity DataIC50: 2.40nMAssay Description:In vitro for binding affinity against angiotensin II receptor type 2 in rat midbrain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282460BDBM50282460(Quinazolinone Analog | CHEMBL169968)
Affinity DataIC50: 2.80nMAssay Description:In vitro for binding affinity against angiotensin II receptor type 2 in rat midbrain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282466BDBM50282466(Quinazolinone Analog | CHEMBL354779)
Affinity DataIC50: 2.90nMAssay Description:In vitro for binding affinity against angiotensin II receptor type 2 in rat midbrain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282455BDBM50282455(Quinazolinone Analog | CHEMBL169967)
Affinity DataIC50: 3.20nMAssay Description:In vitro for binding affinity against angiotensin II receptor type 2 in rat midbrain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282453BDBM50282453(Quinazolinone Analog | CHEMBL353800)
Affinity DataIC50: 3.30nMAssay Description:In vitro for binding affinity against angiotensin II receptor type 2 in rat midbrain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282464BDBM50282464(Quinazolinone Analog | CHEMBL169568)
Affinity DataIC50: 3.60nMAssay Description:In vitro for binding affinity against angiotensin II receptor type 2 in rat midbrain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282470BDBM50282470(Quinazolinone Analog | CHEMBL353037)
Affinity DataIC50: 3.60nMAssay Description:In vitro for binding affinity against angiotensin II receptor type 2 in rat midbrain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282463BDBM50282463(Quinazolinone Analog | CHEMBL354080)
Affinity DataIC50: 4.40nMAssay Description:In vitro for binding affinity against angiotensin II receptor type 2 in rat midbrain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282465BDBM50282465(Quinazolinone Analog | CHEMBL353615)
Affinity DataIC50: 4.60nMAssay Description:In vitro for binding affinity against angiotensin II receptor type 2 in rat midbrain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282476BDBM50282476(Quinazolinone Analog | CHEMBL352458)
Affinity DataIC50: 5nMAssay Description:In vitro for binding affinity against angiotensin II receptor type 2 in rat midbrain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282462BDBM50282462(Quinazolinone Analog | CHEMBL352503)
Affinity DataIC50: 5.30nMAssay Description:In vitro for binding affinity against angiotensin II receptor type 2 in rat midbrain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282472BDBM50282472(Quinazolinone Analog | CHEMBL169221)
Affinity DataIC50: 6.30nMAssay Description:In vitro for binding affinity against angiotensin II receptor type 2 in rat midbrain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282452BDBM50282452(Quinazolinone Analog | CHEMBL169488)
Affinity DataIC50: 7.40nMAssay Description:In vitro for binding affinity against angiotensin II receptor type 2 in rat midbrain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282457BDBM50282457(Quinazolinone Analog | CHEMBL169279)
Affinity DataIC50: 8nMAssay Description:In vitro for binding affinity against angiotensin II receptor type 2 in rat midbrain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282473BDBM50282473(Quinazolinone Analog | CHEMBL354298)
Affinity DataIC50: 8.90nMAssay Description:In vitro for binding affinity against angiotensin II receptor type 2 in rat midbrain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282461BDBM50282461(Quinazolinone Analog | CHEMBL168490)
Affinity DataIC50: 10nMAssay Description:In vitro for binding affinity against angiotensin II receptor type 2 in rat midbrain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282468BDBM50282468(4'-[2-Butyl-6-(3-isopropyl-ureido)-4-oxo-4H-quinaz...)
Affinity DataIC50: 12nMAssay Description:In vitro for binding affinity against angiotensin II receptor type 2 in rat midbrain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282467BDBM50282467(Quinazolinone Analog | CHEMBL352629)
Affinity DataIC50: 13nMAssay Description:In vitro for binding affinity against angiotensin II receptor type 2 in rat midbrain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282475BDBM50282475(Quinazolinone Analog | CHEMBL168346)
Affinity DataIC50: 15nMAssay Description:Tested in vitro for binding affinity against Angiotensin II receptor, type 1 in rabbit aortic membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282454BDBM50282454(Quinazolinone Analog | CHEMBL353980)
Affinity DataIC50: 15nMAssay Description:In vitro for binding affinity against angiotensin II receptor type 2 in rat midbrain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282471BDBM50282471(N-[3-(2'-Benzoylsulfamoyl-biphenyl-4-ylmethyl)-4-o...)
Affinity DataIC50: 16nMAssay Description:In vitro for binding affinity against angiotensin II receptor type 2 in rat midbrain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282474BDBM50282474(N-[3-(2'-Acetylsulfamoyl-biphenyl-4-ylmethyl)-4-ox...)
Affinity DataIC50: 16nMAssay Description:Tested in vitro for binding affinity against Angiotensin II receptor, type 1 in rabbit aortic membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282477BDBM50282477(Quinazolinone Analog | CHEMBL168413)
Affinity DataIC50: 20nMAssay Description:In vitro for binding affinity against angiotensin II receptor type 2 in rat midbrain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282459BDBM50282459(Quinazolinone Analog | CHEMBL169009)
Affinity DataIC50: 170nMAssay Description:In vitro for binding affinity against angiotensin II receptor type 2 in rat midbrain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

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