Compile Data Set for Download or QSAR
maximum 50k data
Found 58 Enz. Inhib. hit(s) with all data for entry = 50029368
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50283831(CHEMBL319986 | N-tert-Butyl-2-[(3R,5S,7R)-7-(3-flu...)
Affinity DataIC50:  1nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50283845(2-[(3R,5S,7R)-2-Oxo-7-phenyl-5-o-tolyl-3-(3-m-toly...)
Affinity DataIC50:  1.10nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50283832(CHEMBL319504 | N-tert-Butyl-2-[(3R,5S,7R)-2-oxo-7-...)
Affinity DataIC50:  1.10nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50283843(CHEMBL320821 | N-(2-Chloro-phenyl)-2-[(3R,5S,7R)-2...)
Affinity DataIC50:  1.10nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50283842(CHEMBL316619 | N-tert-Butyl-2-[(3R,5S,7R)-2-oxo-7-...)
Affinity DataIC50:  1.30nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50283838(CHEMBL316504 | N-tert-Butyl-2-[(3R,5S,7R)-2-oxo-5-...)
Affinity DataIC50:  1.60nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50283826(CHEMBL327496 | N-tert-Butyl-2-{(3R,5S,7R)-3-[3-(3-...)
Affinity DataIC50:  1.80nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50283827(CHEMBL329286 | N-tert-Butyl-2-{(3R,5S,7R)-3-[3-(4-...)
Affinity DataIC50:  2.20nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50283839(CHEMBL330197 | N-tert-Butyl-2-[(3R,5S,7R)-7-(4-flu...)
Affinity DataIC50:  2.80nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50283824(CHEMBL329735 | N-(1-Methyl-cyclohexyl)-2-[(3R,5S,7...)
Affinity DataIC50:  4.40nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283825(CHEMBL96970 | N-tert-Butyl-2-[(3R,5S,7R)-2-oxo-7-p...)
Affinity DataIC50:  7.80nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50006878((R)-1-(1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benz...)
Affinity DataIC50:  8.10nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50283830(2-{(3R,5S,7R)-3-[3-(3-Ethyl-phenyl)-ureido]-2-oxo-...)
Affinity DataIC50: >10nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50283836(2-[(3R,5S,7R)-2-Oxo-7-phenyl-5-o-tolyl-3-(3-m-toly...)
Affinity DataIC50: >10nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50283829(CHEMBL99311 | N-tert-Butyl-2-{(3R,5S,7R)-3-[3-(4-c...)
Affinity DataIC50: >10nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50283823(CHEMBL321752 | N-(1-tert-Butyl-2,2-dimethyl-propyl...)
Affinity DataIC50: >10nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50283847(CHEMBL319882 | N-tert-Butyl-2-{(3R,5S,7R)-3-[3-(3-...)
Affinity DataIC50: >10nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50283840(CHEMBL319749 | N-tert-Butyl-2-[(3S,5S,7R)-2-oxo-5,...)
Affinity DataIC50:  10nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50283828(CHEMBL414223 | N-(3-Chloro-phenyl)-2-[(3R,5S,7R)-2...)
Affinity DataIC50: >10nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50283841(CHEMBL317366 | N-(4-Chloro-phenyl)-2-[(3R,5S,7R)-2...)
Affinity DataIC50: >10nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283847(CHEMBL319882 | N-tert-Butyl-2-{(3R,5S,7R)-3-[3-(3-...)
Affinity DataIC50:  10nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283833(CHEMBL327526 | N-tert-Butyl-2-[(3R,5S,7R)-2-oxo-5,...)
Affinity DataIC50:  16nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283822(CHEMBL97133 | N-tert-Butyl-2-[(3R,5S,7R)-5-(2-ethy...)
Affinity DataIC50:  25nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283843(CHEMBL320821 | N-(2-Chloro-phenyl)-2-[(3R,5S,7R)-2...)
Affinity DataIC50:  28nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283834(CHEMBL319748 | N-tert-Butyl-2-{(3R,5S,7R)-2-oxo-7-...)
Affinity DataIC50:  28nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283844(CHEMBL99289 | N-tert-Butyl-2-[(3R,5S,7R)-5-(2-meth...)
Affinity DataIC50:  28nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283831(CHEMBL319986 | N-tert-Butyl-2-[(3R,5S,7R)-7-(3-flu...)
Affinity DataIC50:  31nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283826(CHEMBL327496 | N-tert-Butyl-2-{(3R,5S,7R)-3-[3-(3-...)
Affinity DataIC50:  36nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283830(2-{(3R,5S,7R)-3-[3-(3-Ethyl-phenyl)-ureido]-2-oxo-...)
Affinity DataIC50:  38nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283836(2-[(3R,5S,7R)-2-Oxo-7-phenyl-5-o-tolyl-3-(3-m-toly...)
Affinity DataIC50:  40nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283837(CHEMBL95209 | N-tert-Butyl-2-[(3R,5S,7R)-5-(4-fluo...)
Affinity DataIC50:  65nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283842(CHEMBL316619 | N-tert-Butyl-2-[(3R,5S,7R)-2-oxo-7-...)
Affinity DataIC50:  66nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283845(2-[(3R,5S,7R)-2-Oxo-7-phenyl-5-o-tolyl-3-(3-m-toly...)
Affinity DataIC50:  71nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283828(CHEMBL414223 | N-(3-Chloro-phenyl)-2-[(3R,5S,7R)-2...)
Affinity DataIC50:  79nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283835(CHEMBL319569 | N-Isopropyl-2-[(3R,5S,7R)-2-oxo-7-p...)
Affinity DataIC50:  80nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50006878((R)-1-(1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benz...)
Affinity DataIC50:  86nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283827(CHEMBL329286 | N-tert-Butyl-2-{(3R,5S,7R)-3-[3-(4-...)
Affinity DataIC50:  87nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283829(CHEMBL99311 | N-tert-Butyl-2-{(3R,5S,7R)-3-[3-(4-c...)
Affinity DataIC50:  117nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283824(CHEMBL329735 | N-(1-Methyl-cyclohexyl)-2-[(3R,5S,7...)
Affinity DataIC50:  134nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283838(CHEMBL316504 | N-tert-Butyl-2-[(3R,5S,7R)-2-oxo-5-...)
Affinity DataIC50:  141nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283832(CHEMBL319504 | N-tert-Butyl-2-[(3R,5S,7R)-2-oxo-7-...)
Affinity DataIC50:  190nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283839(CHEMBL330197 | N-tert-Butyl-2-[(3R,5S,7R)-7-(4-flu...)
Affinity DataIC50:  203nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283841(CHEMBL317366 | N-(4-Chloro-phenyl)-2-[(3R,5S,7R)-2...)
Affinity DataIC50:  278nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283840(CHEMBL319749 | N-tert-Butyl-2-[(3S,5S,7R)-2-oxo-5,...)
Affinity DataIC50:  450nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283823(CHEMBL321752 | N-(1-tert-Butyl-2,2-dimethyl-propyl...)
Affinity DataIC50:  453nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283825(CHEMBL96970 | N-tert-Butyl-2-[(3R,5S,7R)-2-oxo-7-p...)
Affinity DataIC50:  527nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283825(CHEMBL96970 | N-tert-Butyl-2-[(3R,5S,7R)-2-oxo-7-p...)
Affinity DataIC50:  527nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50283835(CHEMBL319569 | N-Isopropyl-2-[(3R,5S,7R)-2-oxo-7-p...)
Affinity DataIC50:  560nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283846(CHEMBL95369 | N-tert-Butyl-2-[(3R,5S,7R)-2-oxo-5-p...)
Affinity DataIC50:  560nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50283825(CHEMBL96970 | N-tert-Butyl-2-[(3R,5S,7R)-2-oxo-7-p...)
Affinity DataIC50:  580nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In DepthDetails Article
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