Compile Data Set for Download or QSAR
Report error Found 42 Enz. Inhib. hit(s) with all data for entry = 50029372
TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50283886BDBM50283886(18-hydroxy-3-methoxy-2-methyl-4-methylamino-(2R,3S...)
Affinity DataIC50: 17nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50283895BDBM50283895(3-methoxy-2-methyl-16-oxo-(2R,3S,4S,6S)-29-oxa-1,7...)
Affinity DataIC50: 19nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50283891BDBM50283891(2-[3-methoxy-2-methyl-16-oxo-(2R,3S,4S,6S)-29-oxa-...)
Affinity DataIC50: 31nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50283899BDBM50283899(ethyl[3-methoxy-2-methyl-16-oxo-(2R,3S,4S,6S)-29-o...)
Affinity DataIC50: 43nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 2579BDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 100nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50283888BDBM50283888(4-[3-methoxy-2-methyl-16-oxo-(2R,3S,4S,6S)-29-oxa-...)
Affinity DataIC50: 110nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50283892BDBM50283892(3-[3-methoxy-2-methyl-16-oxo-(2R,3S,4S,6S)-29-oxa-...)
Affinity DataIC50: 160nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50283901BDBM50283901(Staurosporine derivative | CHEMBL335931)
Affinity DataIC50: 160nMAssay Description:Inhibition of Src tyrosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50283894BDBM50283894(3-methoxy-2-methyl-4-methylamino-(2R,3S,4S,6S)-29-...)
Affinity DataIC50: 200nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50283892BDBM50283892(3-[3-methoxy-2-methyl-16-oxo-(2R,3S,4S,6S)-29-oxa-...)
Affinity DataIC50: 200nMAssay Description:Inhibition of Src tyrosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50283909BDBM50283909(1N-[3-methoxy-2-methyl-16-oxo-(2R,3S,4S,6S)-29-oxa...)
Affinity DataIC50: 220nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50283900BDBM50283900(4-ethyl(methyl)amino-3-methoxy-2-methyl-(2R,3S,4S,...)
Affinity DataIC50: 240nMAssay Description:Inhibition of Src tyrosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50283903BDBM50283903(18-hydroxy-5-methoxy-6-methyl-4-methylamino-(2S,4S...)
Affinity DataIC50: 260nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50283900BDBM50283900(4-ethyl(methyl)amino-3-methoxy-2-methyl-(2R,3S,4S,...)
Affinity DataIC50: 330nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 2579BDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 350nMAssay Description:Inhibition of Src tyrosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50283886BDBM50283886(18-hydroxy-3-methoxy-2-methyl-4-methylamino-(2R,3S...)
Affinity DataIC50: 600nMAssay Description:Inhibition of Src tyrosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50283894BDBM50283894(3-methoxy-2-methyl-4-methylamino-(2R,3S,4S,6S)-29-...)
Affinity DataIC50: 800nMAssay Description:Inhibition of Src tyrosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 31094BDBM31094(PKC-412 | cid_24202429)
Affinity DataIC50: 800nMAssay Description:Inhibition of Src tyrosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50283902BDBM50283902(4-benzyl(methyl)amino-3-methoxy-2-methyl-(2R,3S,4S...)
Affinity DataIC50: 910nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50283896BDBM50283896(N-[3-methoxy-2-methyl-16-oxo-(2R,3S,4S,6S)-29-oxa-...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50283906BDBM50283906(2-[3-methoxy-2-methyl-16-oxo-(2R,3S,4S,6S)-29-oxa-...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50283883BDBM50283883(methyl 2-[3-methoxy-2-methyl-16-oxo-(2R,3S,4S,6S)-...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50283887BDBM50283887(4-[2-hydroxyhexyl(methyl)amino]-3-methoxy-2-methyl...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50283903BDBM50283903(18-hydroxy-5-methoxy-6-methyl-4-methylamino-(2S,4S...)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of Src tyrosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 31094BDBM31094(PKC-412 | cid_24202429)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50283889BDBM50283889(Staurosporine derivative | CHEMBL130049)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50283893BDBM50283893(1N-[3-methoxy-2-methyl-16-oxo-(2R,3S,4S,6S)-29-oxa...)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50283901BDBM50283901(Staurosporine derivative | CHEMBL335931)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50283882BDBM50283882(3-methoxy-4-[4-methoxyphenyl(methyl)carboxamido]-2...)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50283898BDBM50283898(4-[3-chlorophenyl(methyl)carboxamido]-3-methoxy-2-...)
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50283897BDBM50283897(4-[2-chlorophenyl(methyl)carboxamido]-3-methoxy-2-...)
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50283904BDBM50283904(3-methoxy-2-methyl-4-methyl(3-nitrophenyl)carboxam...)
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50283912BDBM50283912(1N-[3-methoxy-2-methyl-16-oxo-(2R,3S,4S,6S)-29-oxa...)
Affinity DataIC50: 6.40E+3nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50283910BDBM50283910(4-[4-chlorophenyl(methyl)carboxamido]-3-methoxy-2-...)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50283878BDBM50283878(Staurosporine derivative | CHEMBL336192)
Affinity DataIC50: 7.40E+3nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50283881BDBM50283881(3-methoxy-2-methyl-4-methyl(3-pyridyl)carboxamido-...)
Affinity DataIC50: 8.18E+3nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50283905BDBM50283905(3-methoxy-2-methyl-4-methyl(2-pyrazinyl)carboxamid...)
Affinity DataIC50: 8.18E+3nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50283879BDBM50283879(3-methoxy-2-methyl-4-methyl[methylamino(thioxo)met...)
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50283884BDBM50283884(Staurosporine derivative | CHEMBL338449)
Affinity DataIC50: 1.35E+4nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50283880BDBM50283880(4-[3,5-dinitrophenyl(methyl)carboxamido]-3-methoxy...)
Affinity DataIC50: 7.00E+4nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50283911BDBM50283911(methyl 2-[3-methoxy-2-methyl-4-methyl(phenyl)carbo...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50283914BDBM50283914(17-benzyl-3-methoxy-2-methyl-4-methyl(phenyl)carbo...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against protein tyrosine kinase of Epidermal growth factor receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article