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Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50029378 Sort by
TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50283962((S)-1-Benzyl-3,5-bis-(1H-indol-3-ylmethyl)-piperid...)
Affinity DataIC50:  4.00E+3nMAssay Description:Binding affinity towards CCK-A receptor in rat pancreas using [125I]-Bolton-Hunter CCK-8 as radioligand; Value ranges from 3.5-4.6 uMMore data for this Ligand-Target Pair
In DepthDetails Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50283965((3R,5S)-1-Benzyl-3,5-bis-(1H-indol-3-ylmethyl)-pip...)
Affinity DataIC50:  4.10E+3nMAssay Description:Binding affinity towards CCK-A receptor in rat pancreas using [125I]-Bolton-Hunter CCK-8 as radioligand; Value ranges from 3.3-5.4 uMMore data for this Ligand-Target Pair
In DepthDetails Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50283963(3-(1-Benzyl-4-hydroxy-piperidin-3-ylmethyl)-indole...)
Affinity DataIC50:  5.20E+3nMAssay Description:Binding affinity towards CCK-A receptor in rat pancreas using [125I]-Bolton-Hunter CCK-8 as radioligand; Value ranges from 4.1-6.4 uMMore data for this Ligand-Target Pair
In DepthDetails Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50283961(3-[1-Benzyl-4-(diethoxy-phosphoryloxy)-1,2,3,6-tet...)
Affinity DataIC50:  5.50E+3nMAssay Description:Binding affinity towards CCK-A receptor in rat pancreas using [125I]-Bolton-Hunter CCK-8 as radioligand; Value ranges from 4.7-7.1 uMMore data for this Ligand-Target Pair
In DepthDetails Article

TargetSubstance-K receptor(Golden hamster)
TBA

Curated by ChEMBL
LigandPNGBDBM50283960(1-Benzyl-3-(1H-indol-3-ylmethyl)-piperidin-4-one |...)
Affinity DataIC50:  6.80E+3nMAssay Description:Binding affinity towards Tachykinin receptor 2 in hamster urinary bladder using [125I]-Neurokinin A as radioligand; Value ranges from 4.6-9.0 uMMore data for this Ligand-Target Pair
In DepthDetails Article

TargetSubstance-K receptor(Golden hamster)
TBA

Curated by ChEMBL
LigandPNGBDBM50283964(3-Benzyl-1-(3-1H-indol-3-yl-propionyl)-piperidin-4...)
Affinity DataIC50:  6.90E+3nMAssay Description:Binding affinity towards Tachykinin receptor 2 in hamster urinary bladder using [125I]-Neurokinin A as radioligand; Value ranges from 2.6-11 uMMore data for this Ligand-Target Pair
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TargetSubstance-P receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283959(3-Benzyl-4-oxo-piperidine-1-carboxylic acid benzyl...)
Affinity DataIC50:  8.10E+3nMAssay Description:Binding affinity towards NK-1 receptor in guinea pig cerebral cortex using [125I]-Bolton-Hunter substance P as radioligand; Value ranges from 7.3-8.8...More data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50283961(3-[1-Benzyl-4-(diethoxy-phosphoryloxy)-1,2,3,6-tet...)
Affinity DataIC50:  8.50E+3nMAssay Description:Binding affinity towards CCK-B receptor in mouse cerebral cortex using [125I]-Bolton-Hunter CCK-8 as radioligand; Value ranges from 7.8-9.3 uMMore data for this Ligand-Target Pair
In DepthDetails Article

TargetNeuromedin-K receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283966((S)-1-Benzyl-3-(1H-indol-3-ylmethyl)-piperidin-4-o...)
Affinity DataIC50:  8.80E+3nMAssay Description:Binding affinity towards Tachykinin receptor 3 in guinea pig cerebral cortex using [3H]-Senktide as radioligand; Value ranges from 8.2-9.4 uMMore data for this Ligand-Target Pair
In DepthDetails Article

TargetNeuromedin-K receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283960(1-Benzyl-3-(1H-indol-3-ylmethyl)-piperidin-4-one |...)
Affinity DataIC50:  1.00E+4nMAssay Description:Binding affinity towards Tachykinin receptor 3 in guinea pig cerebral cortex using [3H]-Senktide as radioligand; Value ranges from 5.8-14u MMore data for this Ligand-Target Pair
In DepthDetails Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50283959(3-Benzyl-4-oxo-piperidine-1-carboxylic acid benzyl...)
Affinity DataIC50:  1.30E+4nMAssay Description:Binding affinity towards CCK-A receptor in rat pancreas using [125I]-Bolton-Hunter CCK-8 as radioligand; Value ranges from 11-16 uMMore data for this Ligand-Target Pair
In DepthDetails Article

LigandPNGBDBM50283965((3R,5S)-1-Benzyl-3,5-bis-(1H-indol-3-ylmethyl)-pip...)
Affinity DataIC50:  1.50E+4nMAssay Description:Binding affinity towards CCK-B receptor in mouse cerebral cortex using [125I]-Bolton-Hunter CCK-8 as radioligand; Value ranges from 9.8-25 uMMore data for this Ligand-Target Pair
In DepthDetails Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50283960(1-Benzyl-3-(1H-indol-3-ylmethyl)-piperidin-4-one |...)
Affinity DataIC50:  1.60E+4nMAssay Description:Binding affinity towards CCK-A receptor in rat pancreas using [125I]-Bolton-Hunter CCK-8 as radioligand; Value ranges from 12-20 uMMore data for this Ligand-Target Pair
In DepthDetails Article