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Found 14 Enz. Inhib. hit(s) with all data for entry = 50029419
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284306(2-[(1E,3E)-4-(3,4-Dihydroxy-phenyl)-buta-1,3-dieny...)
Affinity DataIC50:  20nMAssay Description:Inhibition of 5-lipoxygenase of rat basophilic leukemia (RBL) cell cytosolic enzymesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284305(4-((1E,3E)-4-Benzooxazol-2-yl-buta-1,3-dienyl)-ben...)
Affinity DataIC50:  30nMAssay Description:Inhibition of 5-lipoxygenase of rat basophilic leukemia (RBL) cell cytosolic enzymesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284304(2-[(1E,3E)-4-(4-Hydroxy-3-methoxy-phenyl)-buta-1,3...)
Affinity DataIC50:  130nMAssay Description:Inhibition of 5-lipoxygenase of rat basophilic leukemia (RBL) cell cytosolic enzymesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284309((2E,4E)-5-(4-Hydroxy-3-methoxy-phenyl)-penta-2,4-d...)
Affinity DataIC50:  150nMAssay Description:Inhibition of 5-lipoxygenase of rat basophilic leukemia (RBL) cell cytosolic enzymesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284314(2-Methoxy-4-((1E,3E)-4-naphtho[1,2-d]oxazol-2-yl-b...)
Affinity DataIC50:  170nMAssay Description:Inhibition of 5-lipoxygenase of rat basophilic leukemia (RBL) cell cytosolic enzymesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284310(2-[(1E,3E)-4-(4-Hydroxy-3-methoxy-phenyl)-buta-1,3...)
Affinity DataIC50:  250nMAssay Description:Inhibition of 5-lipoxygenase of rat basophilic leukemia (RBL) cell cytosolic enzymesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284303(4-[(1E,3E)-4-(5-Hydroxymethyl-benzooxazol-2-yl)-bu...)
Affinity DataIC50:  260nMAssay Description:Inhibition of 5-lipoxygenase of rat basophilic leukemia (RBL) cell cytosolic enzymesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284311(2-Methoxy-4-[(1E,3E)-4-(5-methyl-benzooxazol-2-yl)...)
Affinity DataIC50:  290nMAssay Description:Inhibition of 5-lipoxygenase of rat basophilic leukemia (RBL) cell cytosolic enzymesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284315(4-[(1E,3E)-4-(6-Hydroxymethyl-benzooxazol-2-yl)-bu...)
Affinity DataIC50:  300nMAssay Description:Inhibition of 5-lipoxygenase of rat basophilic leukemia (RBL) cell cytosolic enzymesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284313(4-((1E,3E)-4-Benzooxazol-2-yl-buta-1,3-dienyl)-2-m...)
Affinity DataIC50:  330nMAssay Description:Inhibition of 5-lipoxygenase of rat basophilic leukemia (RBL) cell cytosolic enzymesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284308(2-Methoxy-4-((1E,3E)-4-oxazolo[4,5-b]pyridin-2-yl-...)
Affinity DataIC50:  370nMAssay Description:Inhibition of 5-lipoxygenase of rat basophilic leukemia (RBL) cell cytosolic enzymesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284307(4-[(1E,3E)-4-(5-Chloro-benzooxazol-2-yl)-buta-1,3-...)
Affinity DataIC50:  380nMAssay Description:Inhibition of 5-lipoxygenase of rat basophilic leukemia (RBL) cell cytosolic enzymesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50029196((E)-3-(3,4-Dihydroxy-phenyl)-acrylic acid ethyl es...)
Affinity DataIC50:  1.15E+3nMAssay Description:Inhibition of 5-lipoxygenase of rat basophilic leukemia (RBL) cell cytosolic enzymesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284312(2-[(1E,3E)-4-(4-Hydroxy-3-methoxy-phenyl)-buta-1,3...)
Affinity DataIC50:  5.80E+3nMAssay Description:Inhibition of 5-lipoxygenase of rat basophilic leukemia (RBL) cell cytosolic enzymesMore data for this Ligand-Target Pair
In DepthDetails Article