Compile Data Set for Download or QSAR
Report error Found 68 Enz. Inhib. hit(s) with all data for entry = 50029444
TargetD(2) dopamine receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  1.5nMAssay Description:Ability to displace [3H]spiperone from D2 dopamine receptor isolated from the striata of male Wistar ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetD(2) dopamine receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50001885(3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin...)
Affinity DataKi:  1.80nMAssay Description:Ability to displace [3H]spiperone from D2 dopamine receptor isolated from the striata of male Wistar ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetD(2) dopamine receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284595(4-Methyl-6-methylsulfanyl-3,4-dihydro-2H-benzo[1,4...)
Affinity DataKi:  3.60nMAssay Description:Ability to displace [3H]spiperone from D2 dopamine receptor isolated from the striata of male Wistar ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetD(2) dopamine receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284598(5-Chloro-2,3-dihydro-benzofuran-7-carboxylic acid ...)
Affinity DataKi:  3.80nMAssay Description:Ability to displace [3H]spiperone from D2 dopamine receptor isolated from the striata of male Wistar ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetD(2) dopamine receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284608(4-Methyl-6-methylsulfanyl-3,4-dihydro-2H-benzo[1,4...)
Affinity DataKi:  4.20nMAssay Description:Ability to displace [3H]spiperone from D2 dopamine receptor isolated from the striata of male Wistar ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetD(2) dopamine receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284589(5-Chloro-2,3-dihydro-benzofuran-7-carboxylic acid ...)
Affinity DataKi:  6.5nMAssay Description:Ability to displace [3H]spiperone from D2 dopamine receptor isolated from the striata of male Wistar ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

Target5-hydroxytryptamine receptor 1A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50086858(6-Chloro-4-methyl-3,4-dihydro-2H-benzo[1,4]oxazine...)
Affinity DataKi:  10nMAssay Description:Ability to displace [3H]-8-OH-DPAT from serotonergic 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetD(2) dopamine receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50086852(6-Chloro-4-methyl-3,4-dihydro-2H-benzo[1,4]oxazine...)
Affinity DataKi:  12nMAssay Description:Compound was evaluated for its ability to displace [3H]spiperone from D2 dopamine receptor isolated from the striata of male Wistar ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetD(2) dopamine receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284593(6-Chloro-4-methyl-3,4-dihydro-2H-benzo[1,4]oxazine...)
Affinity DataKi:  16nMAssay Description:Ability to displace [3H]spiperone from D2 dopamine receptor isolated from the striata of male Wistar ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

Target5-hydroxytryptamine receptor 1A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284607(2-Methoxy-N-((R)-1-nonyl-pyrrolidin-2-ylmethyl)-5-...)
Affinity DataKi:  16nMAssay Description:Ability to displace [3H]-8-OH-DPAT from serotonergic 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetD(2) dopamine receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284611(4-Methyl-6-methylsulfanyl-3,4-dihydro-2H-benzo[1,4...)
Affinity DataKi:  17nMAssay Description:Ability to displace [3H]spiperone from D2 dopamine receptor isolated from the striata of male Wistar ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

Target5-hydroxytryptamine receptor 1A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284608(4-Methyl-6-methylsulfanyl-3,4-dihydro-2H-benzo[1,4...)
Affinity DataKi:  17nMAssay Description:Ability to displace [3H]-8-OH-DPAT from serotonergic 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

Target5-hydroxytryptamine receptor 1A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284598(5-Chloro-2,3-dihydro-benzofuran-7-carboxylic acid ...)
Affinity DataKi:  18nMAssay Description:Ability to displace [3H]-8-OH-DPAT from serotonergic 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetD(2) dopamine receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284590(5-Chloro-2,3-dihydro-benzofuran-7-carboxylic acid ...)
Affinity DataKi:  19nMAssay Description:Ability to displace [3H]spiperone from D2 dopamine receptor isolated from the striata of male Wistar ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

Target5-hydroxytryptamine receptor 1A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284595(4-Methyl-6-methylsulfanyl-3,4-dihydro-2H-benzo[1,4...)
Affinity DataKi:  19nMAssay Description:Ability to displace [3H]-8-OH-DPAT from serotonergic 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

Target5-hydroxytryptamine receptor 1A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284602(6-Chloro-4-methyl-3,4-dihydro-2H-benzo[1,4]oxazine...)
Affinity DataKi:  21nMAssay Description:Ability to displace [3H]-8-OH-DPAT from serotonergic 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

Target5-hydroxytryptamine receptor 1A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50086852(6-Chloro-4-methyl-3,4-dihydro-2H-benzo[1,4]oxazine...)
Affinity DataKi:  34nMAssay Description:Compound was evaluated for its ability to displace [3H]8-OH-DPAT from serotonergic 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

Target5-hydroxytryptamine receptor 1A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50086862(6-Chloro-4-methyl-3,4-dihydro-2H-benzo[1,4]oxazine...)
Affinity DataKi:  35nMAssay Description:Ability to displace [3H]-8-OH-DPAT from serotonergic 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetD(2) dopamine receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284586(N-((S)-1-Butyl-pyrrolidin-2-ylmethyl)-2-methoxy-5-...)
Affinity DataKi:  51nMAssay Description:Compound was evaluated for its ability to displace [3H]spiperone from D2 dopamine receptor isolated from the striata of male Wistar ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetD(2) dopamine receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50086862(6-Chloro-4-methyl-3,4-dihydro-2H-benzo[1,4]oxazine...)
Affinity DataKi:  57nMAssay Description:Ability to displace [3H]spiperone from D2 dopamine receptor isolated from the striata of male Wistar ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

Target5-hydroxytryptamine receptor 1A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284597(2-Methoxy-N-((S)-1-nonyl-pyrrolidin-2-ylmethyl)-5-...)
Affinity DataKi:  81nMAssay Description:Ability to displace [3H]-8-OH-DPAT from serotonergic 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetD(2) dopamine receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284591(5-Chloro-2,3-dihydro-benzofuran-7-carboxylic acid ...)
Affinity DataKi:  84nMAssay Description:Ability to displace [3H]spiperone from D2 dopamine receptor isolated from the striata of male Wistar ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetD(2) dopamine receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284607(2-Methoxy-N-((R)-1-nonyl-pyrrolidin-2-ylmethyl)-5-...)
Affinity DataKi:  92nMAssay Description:Ability to displace [3H]spiperone from D2 dopamine receptor isolated from the striata of male Wistar ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

Target5-hydroxytryptamine receptor 1A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284611(4-Methyl-6-methylsulfanyl-3,4-dihydro-2H-benzo[1,4...)
Affinity DataKi:  120nMAssay Description:Ability to displace [3H]-8-OH-DPAT from serotonergic 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

Target5-hydroxytryptamine receptor 1A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50001885(3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin...)
Affinity DataKi:  130nMAssay Description:Ability to displace [3H]-8-OH-DPAT from serotonergic 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

Target5-hydroxytryptamine receptor 1A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284606(4-Methyl-3,4-dihydro-2H-benzo[1,4]oxazine-8-carbox...)
Affinity DataKi:  170nMAssay Description:Compound was evaluated for its ability to displace [3H]8-OH-DPAT from serotonergic 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetD(2) dopamine receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284597(2-Methoxy-N-((S)-1-nonyl-pyrrolidin-2-ylmethyl)-5-...)
Affinity DataKi:  180nMAssay Description:Ability to displace [3H]spiperone from D2 dopamine receptor isolated from the striata of male Wistar ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetD(2) dopamine receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284602(6-Chloro-4-methyl-3,4-dihydro-2H-benzo[1,4]oxazine...)
Affinity DataKi:  210nMAssay Description:Ability to displace [3H]spiperone from D2 dopamine receptor isolated from the striata of male Wistar ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

Target5-hydroxytryptamine receptor 1A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284604(6-Chloro-4-methyl-3,4-dihydro-2H-benzo[1,4]oxazine...)
Affinity DataKi:  220nMAssay Description:Ability to displace [3H]-8-OH-DPAT from serotonergic 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetD(2) dopamine receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284609(N-((R)-1-Butyl-pyrrolidin-2-ylmethyl)-2-methoxy-5-...)
Affinity DataKi:  230nMAssay Description:Compound was evaluated for its ability to displace [3H]spiperone from D2 dopamine receptor isolated from the striata of male Wistar ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetD(2) dopamine receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284606(4-Methyl-3,4-dihydro-2H-benzo[1,4]oxazine-8-carbox...)
Affinity DataKi:  270nMAssay Description:Compound was evaluated for its ability to displace [3H]spiperone from D2 dopamine receptor isolated from the striata of male Wistar ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetD(2) dopamine receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284592(4-Methyl-6-methylsulfanyl-3,4-dihydro-2H-benzo[1,4...)
Affinity DataKi:  270nMAssay Description:Ability to displace [3H]spiperone from D2 dopamine receptor isolated from the striata of male Wistar ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

Target5-hydroxytryptamine receptor 1A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284587(6-Chloro-4-methyl-3,4-dihydro-2H-benzo[1,4]oxazine...)
Affinity DataKi:  280nMAssay Description:Compound was evaluated for its ability to displace [3H]8-OH-DPAT from serotonergic 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetD(2) dopamine receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284604(6-Chloro-4-methyl-3,4-dihydro-2H-benzo[1,4]oxazine...)
Affinity DataKi:  310nMAssay Description:Ability to displace [3H]spiperone from D2 dopamine receptor isolated from the striata of male Wistar ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

Target5-hydroxytryptamine receptor 1A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284591(5-Chloro-2,3-dihydro-benzofuran-7-carboxylic acid ...)
Affinity DataKi:  330nMAssay Description:Ability to displace [3H]-8-OH-DPAT from serotonergic 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

Target5-hydroxytryptamine receptor 1A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284590(5-Chloro-2,3-dihydro-benzofuran-7-carboxylic acid ...)
Affinity DataKi:  330nMAssay Description:Ability to displace [3H]-8-OH-DPAT from serotonergic 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

Target5-hydroxytryptamine receptor 1A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50086863(6-Chloro-4-methyl-3,4-dihydro-2H-benzo[1,4]oxazine...)
Affinity DataKi:  430nMAssay Description:Compound was evaluated for its ability to displace [3H]8-OH-DPAT from serotonergic 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

Target5-hydroxytryptamine receptor 1A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284588(4-Methyl-6-sulfamoyl-3,4-dihydro-2H-benzo[1,4]oxaz...)
Affinity DataKi:  450nMAssay Description:Compound was evaluated for its ability to displace [3H]8-OH-DPAT from serotonergic 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

Target5-hydroxytryptamine receptor 1A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284612(5-Chloro-2,3-dihydro-benzofuran-7-carboxylic acid ...)
Affinity DataKi:  570nMAssay Description:Ability to displace [3H]-8-OH-DPAT from serotonergic 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetD(2) dopamine receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50086863(6-Chloro-4-methyl-3,4-dihydro-2H-benzo[1,4]oxazine...)
Affinity DataKi:  630nMAssay Description:Compound was evaluated for its ability to displace [3H]spiperone from D2 dopamine receptor isolated from the striata of male Wistar ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetD(2) dopamine receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284588(4-Methyl-6-sulfamoyl-3,4-dihydro-2H-benzo[1,4]oxaz...)
Affinity DataKi:  670nMAssay Description:Compound was evaluated for its ability to displace [3H]spiperone from D2 dopamine receptor isolated from the striata of male Wistar ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetD(2) dopamine receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284603(6-Chloro-4-methyl-3,4-dihydro-2H-benzo[1,4]oxazine...)
Affinity DataKi:  690nMAssay Description:Compound was evaluated for its ability to displace [3H]spiperone from D2 dopamine receptor isolated from the striata of male Wistar ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetD(2) dopamine receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284587(6-Chloro-4-methyl-3,4-dihydro-2H-benzo[1,4]oxazine...)
Affinity DataKi:  750nMAssay Description:Compound was evaluated for its ability to displace [3H]spiperone from D2 dopamine receptor isolated from the striata of male Wistar ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetD(2) dopamine receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50086858(6-Chloro-4-methyl-3,4-dihydro-2H-benzo[1,4]oxazine...)
Affinity DataKi:  800nMAssay Description:Ability to displace [3H]spiperone from D2 dopamine receptor isolated from the striata of male Wistar ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

Target5-hydroxytryptamine receptor 1A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284592(4-Methyl-6-methylsulfanyl-3,4-dihydro-2H-benzo[1,4...)
Affinity DataKi:  880nMAssay Description:Ability to displace [3H]-8-OH-DPAT from serotonergic 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetD(2) dopamine receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284600(6-Chloro-4-methyl-3-oxo-3,4-dihydro-2H-benzo[1,4]o...)
Affinity DataKi: >1.00E+3nMAssay Description:Ability to displace [3H]spiperone from D2 dopamine receptor isolated from the striata of male Wistar ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

Target5-hydroxytryptamine receptor 1A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284589(5-Chloro-2,3-dihydro-benzofuran-7-carboxylic acid ...)
Affinity DataKi: >1.00E+3nMAssay Description:Ability to displace [3H]-8-OH-DPAT from serotonergic 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetD(2) dopamine receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284613(6-Chloro-4-methyl-3-oxo-3,4-dihydro-2H-benzo[1,4]o...)
Affinity DataKi: >1.00E+3nMAssay Description:Ability to displace [3H]spiperone from D2 dopamine receptor isolated from the striata of male Wistar ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetD(2) dopamine receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284601(6-Chloro-4-methyl-3-oxo-3,4-dihydro-2H-benzo[1,4]o...)
Affinity DataKi: >1.00E+3nMAssay Description:Ability to displace [3H]spiperone from D2 dopamine receptor isolated from the striata of male Wistar ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetD(2) dopamine receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284612(5-Chloro-2,3-dihydro-benzofuran-7-carboxylic acid ...)
Affinity DataKi: >1.00E+3nMAssay Description:Ability to displace [3H]spiperone from D2 dopamine receptor isolated from the striata of male Wistar ratsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

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