Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50029473
TargetAcyl-CoA:cholesterol acyltransferase(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50284874(1-(2,6-Diisopropyl-phenyl)-3-((4R,5R)-4,5-dimethyl...)
Affinity DataIC50: 24nMAssay Description:Inhibitory activity against acyl-CoA: cholesterol acyltransferase (ACAT) in microsomes from monkey liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetAcyl-CoA:cholesterol acyltransferase(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50284874(1-(2,6-Diisopropyl-phenyl)-3-((4R,5R)-4,5-dimethyl...)
Affinity DataIC50: 27nMAssay Description:Inhibitory activity against acyl-CoA: cholesterol acyltransferase (ACAT) in microsomes from cholesterol-fed rabbit intestinal mucosaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetAcyl-CoA:cholesterol acyltransferase(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50284873(1-(2,6-Diisopropyl-phenyl)-3-[(4R,5R)-2-(4-hydroxy...)
Affinity DataIC50: 27nMAssay Description:Inhibitory activity against acyl-CoA: cholesterol acyltransferase (ACAT) in microsomes from cholesterol-fed rabbit intestinal mucosaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetSterol O-acyltransferase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50284874(1-(2,6-Diisopropyl-phenyl)-3-((4R,5R)-4,5-dimethyl...)
Affinity DataIC50: 63nMAssay Description:Inhibitory activity against acyl-CoA: cholesterol acyltransferase (ACAT) in microsomes from monkey liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetSterol O-acyltransferase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50284873(1-(2,6-Diisopropyl-phenyl)-3-[(4R,5R)-2-(4-hydroxy...)
Affinity DataIC50: 119nMAssay Description:Inhibitory activity against acyl-CoA: cholesterol acyltransferase (ACAT) in microsomes from monkey liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetAcyl-CoA:cholesterol acyltransferase(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50284873(1-(2,6-Diisopropyl-phenyl)-3-[(4R,5R)-2-(4-hydroxy...)
Affinity DataIC50: 119nMAssay Description:Inhibitory activity against acyl-CoA: cholesterol acyltransferase (ACAT) in microsomes from monkey liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetAcyl-CoA:cholesterol acyltransferase(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50284875(Phosphoric acid mono-(4-{(4R,5R)-2-[3-(2,6-diisopr...)
Affinity DataIC50: 1.08E+3nMAssay Description:Inhibitory activity against acyl-CoA: cholesterol acyltransferase (ACAT) in microsomes from cholesterol-fed rabbit intestinal mucosaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetAcyl-CoA:cholesterol acyltransferase(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50284875(Phosphoric acid mono-(4-{(4R,5R)-2-[3-(2,6-diisopr...)
Affinity DataIC50: 2.55E+3nMAssay Description:Inhibitory activity against acyl-CoA: cholesterol acyltransferase (ACAT) in microsomes from monkey liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetSterol O-acyltransferase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50284875(Phosphoric acid mono-(4-{(4R,5R)-2-[3-(2,6-diisopr...)
Affinity DataIC50: 2.55E+3nMAssay Description:Inhibitory activity against acyl-CoA: cholesterol acyltransferase (ACAT) in microsomes from monkey liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article