Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50029522
TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50285198BDBM50285198([(5S,11S,14S)-21-Fluoro-11-(3-guanidino-propyl)-14...)
Affinity DataIC50: 4nMAssay Description:Inhibition of platelet aggregation in vitro using fibrinogen binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50285199BDBM50285199(DMP-757 | [(5S,11S,14S)-11-(3-Guanidino-propyl)-14...)
Affinity DataIC50: 6nMAssay Description:Inhibition of platelet aggregation in vitro using fibrinogen binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50285198BDBM50285198([(5S,11S,14S)-21-Fluoro-11-(3-guanidino-propyl)-14...)
Affinity DataIC50: 20nMAssay Description:Inhibition of platelet aggregation using human platelet rich plasma (hPRP) assay (200microL, 2-3 x 10e 8 platelets/mL, n=1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50285199BDBM50285199(DMP-757 | [(5S,11S,14S)-11-(3-Guanidino-propyl)-14...)
Affinity DataIC50: 20nMAssay Description:Inhibition of platelet aggregation using human platelet rich plasma (hPRP) assay (200microL, 2-3 x 10e 8 platelets/mL, n=1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50285196BDBM50285196([(5S,11S,14S)-11-(3-Guanidino-propyl)-14-isopropyl...)
Affinity DataIC50: 50nMAssay Description:Inhibition of platelet aggregation using human platelet rich plasma (hPRP) assay (200microL, 2-3 x 10e 8 platelets/mL, n=1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50285201BDBM50285201([(5S,11S,14S)-11-(3-Guanidino-propyl)-14-isopropyl...)
Affinity DataIC50: 100nMAssay Description:Inhibition of platelet aggregation using human platelet rich plasma (hPRP) assay (200microL, 2-3 x 10e 8 platelets/mL, n=1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50285194BDBM50285194([(5S,11S,14S)-11-(3-Guanidino-propyl)-14-isopropyl...)
Affinity DataIC50: 100nMAssay Description:Inhibition of platelet aggregation using human platelet rich plasma (hPRP) assay (200microL, 2-3 x 10e 8 platelets/mL, n=1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50285195BDBM50285195([(Z)-(3R,9R,12R)-9-(3-Guanidino-propyl)-12-isoprop...)
Affinity DataIC50: 200nMAssay Description:Inhibition of platelet aggregation using human platelet rich plasma (hPRP) assay (200microL, 2-3 x 10e 8 platelets/mL, n=1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50285200BDBM50285200([(Z)-(3R,9R,12R)-9-(3-Guanidino-propyl)-12-isoprop...)
Affinity DataIC50: 200nMAssay Description:Inhibition of platelet aggregation using human platelet rich plasma (hPRP) assay (200microL, 2-3 x 10e 8 platelets/mL, n=1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50285197BDBM50285197([(4S,10S,13S)-10-(3-Guanidino-propyl)-13-isopropyl...)
Affinity DataIC50: 400nMAssay Description:Inhibition of platelet aggregation using human platelet rich plasma (hPRP) assay (200microL, 2-3 x 10e 8 platelets/mL, n=1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50285202BDBM50285202([(5S,11S,14S)-11-(3-Guanidino-propyl)-14-isopropyl...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of platelet aggregation using human platelet rich plasma (hPRP) assay (200microL, 2-3 x 10e 8 platelets/mL, n=1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article