Compile Data Set for Download or QSAR
maximum 50k data
Found 26 Enz. Inhib. hit(s) with all data for entry = 50029541
TargetNeprilysin(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50064106(CGS-26303 | CHEMBL290698 | {[(R)-2-Biphenyl-4-yl-1...)
Affinity DataIC50:  0.930nMAssay Description:In vitro inhibitory activity against neutral endopeptidase (NEP)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeprilysin(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50285328(CHEMBL285747 | {[(S)-2-Biphenyl-4-yl-1-(1H-tetrazo...)
Affinity DataIC50:  1.40nMAssay Description:In vitro inhibitory activity against neutral endopeptidase (NEP)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeprilysin(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50285340(CHEMBL290285 | {[(S)-2-(2-Methoxy-biphenyl-4-yl)-1...)
Affinity DataIC50:  1.5nMAssay Description:In vitro inhibitory activity against neutral endopeptidase (NEP)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeprilysin(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50285327((S)-3-(2-Methoxy-biphenyl-4-yl)-2-(phosphonomethyl...)
Affinity DataIC50:  14nMAssay Description:In vitro inhibitory activity against neutral endopeptidase (NEP)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeprilysin(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50285343(CHEMBL288440 | {[(S)-2-(4-Isopropoxy-phenyl)-1-(1H...)
Affinity DataIC50:  15nMAssay Description:In vitro inhibitory activity against neutral endopeptidase (NEP)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeprilysin(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50285334((S)-3-Biphenyl-4-yl-2-(phosphonomethyl-amino)-prop...)
Affinity DataIC50:  15nMAssay Description:In vitro inhibitory activity against neutral endopeptidase (NEP)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeprilysin(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50285332((S)-4-Biphenyl-4-yl-3-(phosphonomethyl-amino)-buty...)
Affinity DataIC50:  15nMAssay Description:In vitro inhibitory activity against neutral endopeptidase (NEP)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeprilysin(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50285322(CHEMBL10164 | {[(S)-2-Phenyl-1-(1H-tetrazol-5-yl)-...)
Affinity DataIC50:  26nMAssay Description:In vitro inhibitory activity against neutral endopeptidase (NEP)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeprilysin(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50285325((E)-(S)-5-Biphenyl-4-yl-4-(phosphonomethyl-amino)-...)
Affinity DataIC50:  32nMAssay Description:In vitro inhibitory activity against neutral endopeptidase (NEP)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeprilysin(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50285326((S)-3-(4'-Methyl-biphenyl-4-yl)-2-(phosphonomethyl...)
Affinity DataIC50:  236nMAssay Description:In vitro inhibitory activity against neutral endopeptidase (NEP)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeprilysin(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50285338(CHEMBL36036 | [((S)-1-Benzylcarbamoyl-2-biphenyl-4...)
Affinity DataIC50:  308nMAssay Description:In vitro inhibitory activity against neutral endopeptidase (NEP)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeprilysin(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50285339(CHEMBL275317 | {[(S)-2-Naphthalen-2-yl-1-(1H-tetra...)
Affinity DataIC50:  364nMAssay Description:In vitro inhibitory activity against neutral endopeptidase (NEP)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeprilysin(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50285331(({[(S)-2-Biphenyl-4-yl-1-(1H-tetrazol-5-yl)-ethyl]...)
Affinity DataIC50:  530nMAssay Description:In vitro inhibitory activity against neutral endopeptidase (NEP)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeprilysin(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50285324((R)-5-Biphenyl-4-yl-4-(phosphonomethyl-amino)-pent...)
Affinity DataIC50:  643nMAssay Description:In vitro inhibitory activity against neutral endopeptidase (NEP)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeprilysin(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50285336(3-Biphenyl-2-yl-2-(phosphonomethyl-amino)-propioni...)
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibitory activity against neutral endopeptidase (NEP)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeprilysin(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50285333(CHEMBL291081 | {[2,2-Diphenyl-1-(1H-tetrazol-5-yl)...)
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibitory activity against neutral endopeptidase (NEP)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeprilysin(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50285330(3-Biphenyl-3-yl-2-(phosphonomethyl-amino)-propioni...)
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibitory activity against neutral endopeptidase (NEP)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeprilysin(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50285329(CHEMBL290792 | {[(S)-1-(1-Benzyl-1H-tetrazol-5-yl)...)
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibitory activity against neutral endopeptidase (NEP)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeprilysin(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50403483(CHEMBL273461)
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibitory activity against neutral endopeptidase (NEP)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeprilysin(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50285321((R)-3-Biphenyl-4-yl-2-(phosphonomethyl-amino)-prop...)
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibitory activity against neutral endopeptidase (NEP)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeprilysin(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50285342((S)-2-(Phosphonomethyl-amino)-3-(4-pyridin-3-yl-ph...)
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibitory activity against neutral endopeptidase (NEP)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeprilysin(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50285341((S)-3-Phenyl-2-(phosphonomethyl-amino)-propionic a...)
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibitory activity against neutral endopeptidase (NEP)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeprilysin(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50285323(CHEMBL288034 | [((S)-2-Biphenyl-4-yl-1-carbamoyl-e...)
Affinity DataIC50:  1.30E+3nMAssay Description:In vitro inhibitory activity against neutral endopeptidase (NEP)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeprilysin(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50034851(3-[(S)-3-Biphenyl-4-yl-2-(phosphonomethyl-amino)-p...)
Affinity DataIC50:  1.90E+3nMAssay Description:In vitro inhibitory activity against neutral endopeptidase (NEP)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeprilysin(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50285335((S)-3-Biphenyl-4-yl-2-(2-phosphono-ethylamino)-pro...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibitory activity against neutral endopeptidase (NEP)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeprilysin(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50285337(CHEMBL10384 | {[(S)-3-Phenyl-1-(1H-tetrazol-5-yl)-...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibitory activity against neutral endopeptidase (NEP)More data for this Ligand-Target Pair
In DepthDetails Article