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Found 87 Enz. Inhib. hit(s) with all data for entry = 50029719
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287241(CHEMBL285746 | N-[2-(2-Guanidino-thiazol-4-ylmethy...)
Affinity DataIC50:  3nMAssay Description:Inhibitory activity against gastrin receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50006878((R)-1-(1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benz...)
Affinity DataIC50:  4nMAssay Description:Inhibitory activity against gastrin receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287239(CHEMBL30656 | N-{[2-(2-Guanidino-thiazol-4-ylmethy...)
Affinity DataIC50:  12nMAssay Description:Inhibitory activity against gastrin receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287232(CHEMBL31726 | N-[2-(2-Guanidino-thiazol-4-ylmethyl...)
Affinity DataIC50:  14nMAssay Description:Inhibitory activity against gastrin receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287238(6-{2-[2-Oxo-5-phenyl-3-(3-m-tolyl-ureido)-2,3-dihy...)
Affinity DataIC50:  16nMAssay Description:Inhibitory activity against gastrin receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287245(CHEMBL285586 | N-[2-(2-Guanidino-thiazol-4-ylmethy...)
Affinity DataIC50:  25nMAssay Description:Inhibitory activity against gastrin receptorMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50006878((R)-1-(1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benz...)
Affinity DataIC50:  29nMAssay Description:Inhibitory activity against Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287240(6-(2-{3-[1-Methyl-2-oxo-3-(3-m-tolyl-ureido)-2,3-d...)
Affinity DataIC50:  32nMAssay Description:Inhibitory activity against gastrin receptorMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50287241(CHEMBL285746 | N-[2-(2-Guanidino-thiazol-4-ylmethy...)
Affinity DataIC50:  35nMAssay Description:Inhibitory activity against Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287253(6-(2-{3-[3-((R)-1-Methyl-2-oxo-5-phenyl-2,3-dihydr...)
Affinity DataIC50:  45nMAssay Description:Inhibitory activity against gastrin receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287235(4-(2-{3-[1-Methyl-2-oxo-3-(3-m-tolyl-ureido)-2,3-d...)
Affinity DataIC50:  60nMAssay Description:Inhibitory activity against gastrin receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287243(2-{3-[1-Methyl-2-oxo-3-(3-m-tolyl-ureido)-2,3-dihy...)
Affinity DataIC50:  63nMAssay Description:Inhibitory activity against gastrin receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287259(CHEMBL286908 | N-[2-(2-Guanidino-thiazol-4-ylmethy...)
Affinity DataIC50:  75nMAssay Description:Inhibitory activity against gastrin receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287255(CHEMBL30821 | N-[2-(2-Guanidino-thiazol-4-ylmethyl...)
Affinity DataIC50:  80nMAssay Description:Inhibitory activity against gastrin receptorMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50287256(6-(2-{3-[3-((R)-1-Methyl-2-oxo-5-phenyl-2,3-dihydr...)
Affinity DataIC50:  92nMAssay Description:Inhibitory activity against Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287256(6-(2-{3-[3-((R)-1-Methyl-2-oxo-5-phenyl-2,3-dihydr...)
Affinity DataIC50:  110nMAssay Description:Inhibitory activity against gastrin receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287250(4-(2-{3-[3-((R)-1-Methyl-2-oxo-5-phenyl-2,3-dihydr...)
Affinity DataIC50:  115nMAssay Description:Inhibitory activity against gastrin receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287255(CHEMBL30821 | N-[2-(2-Guanidino-thiazol-4-ylmethyl...)
Affinity DataIC50:  120nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287237(CHEMBL29888 | N-[2-(2-Guanidino-thiazol-4-ylmethyl...)
Affinity DataIC50:  135nMAssay Description:Inhibitory activity against gastrin receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287234(3-(2-{3-[3-((R)-1-Methyl-2-oxo-5-phenyl-2,3-dihydr...)
Affinity DataIC50:  136nMAssay Description:Inhibitory activity against gastrin receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287249(2-[2-Oxo-5-phenyl-3-(3-m-tolyl-ureido)-2,3-dihydro...)
Affinity DataIC50:  155nMAssay Description:Inhibitory activity against gastrin receptorMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50287257(2-{3-[3-((R)-1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1...)
Affinity DataIC50:  160nMAssay Description:Inhibitory activity against Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287248(CHEMBL30430 | N-[2-(2-Guanidino-thiazol-4-ylmethyl...)
Affinity DataIC50:  168nMAssay Description:Inhibitory activity against gastrin receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287252(3-{2-[2-Oxo-5-phenyl-3-(3-m-tolyl-ureido)-2,3-dihy...)
Affinity DataIC50:  185nMAssay Description:Inhibitory activity against gastrin receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287234(3-(2-{3-[3-((R)-1-Methyl-2-oxo-5-phenyl-2,3-dihydr...)
Affinity DataIC50:  190nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287236(CHEMBL286907 | N-[2-(2-Guanidino-thiazol-4-ylmethy...)
Affinity DataIC50:  190nMAssay Description:Inhibitory activity against gastrin receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287253(6-(2-{3-[3-((R)-1-Methyl-2-oxo-5-phenyl-2,3-dihydr...)
Affinity DataIC50:  190nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50287255(CHEMBL30821 | N-[2-(2-Guanidino-thiazol-4-ylmethyl...)
Affinity DataIC50:  200nMAssay Description:Inhibitory activity against Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287242(3-(2-{3-[1-Methyl-2-oxo-3-(3-m-tolyl-ureido)-2,3-d...)
Affinity DataIC50:  200nMAssay Description:Inhibitory activity against gastrin receptorMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50287250(4-(2-{3-[3-((R)-1-Methyl-2-oxo-5-phenyl-2,3-dihydr...)
Affinity DataIC50:  205nMAssay Description:Inhibitory activity against Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287246(4-{2-[2-Oxo-5-phenyl-3-(3-m-tolyl-ureido)-2,3-dihy...)
Affinity DataIC50:  210nMAssay Description:Inhibitory activity against gastrin receptorMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50287232(CHEMBL31726 | N-[2-(2-Guanidino-thiazol-4-ylmethyl...)
Affinity DataIC50:  215nMAssay Description:Inhibitory activity against Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287257(2-{3-[3-((R)-1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1...)
Affinity DataIC50:  230nMAssay Description:Inhibitory activity against gastrin receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287251(CHEMBL262125 | N-[2-(2-Guanidino-thiazol-4-ylmethy...)
Affinity DataIC50:  240nMAssay Description:Inhibitory activity against gastrin receptorMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50287253(6-(2-{3-[3-((R)-1-Methyl-2-oxo-5-phenyl-2,3-dihydr...)
Affinity DataIC50:  255nMAssay Description:Inhibitory activity against Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50287234(3-(2-{3-[3-((R)-1-Methyl-2-oxo-5-phenyl-2,3-dihydr...)
Affinity DataIC50:  290nMAssay Description:Inhibitory activity against Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50287235(4-(2-{3-[1-Methyl-2-oxo-3-(3-m-tolyl-ureido)-2,3-d...)
Affinity DataIC50:  290nMAssay Description:Inhibitory activity against Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50287239(CHEMBL30656 | N-{[2-(2-Guanidino-thiazol-4-ylmethy...)
Affinity DataIC50:  310nMAssay Description:Inhibitory activity against Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50287240(6-(2-{3-[1-Methyl-2-oxo-3-(3-m-tolyl-ureido)-2,3-d...)
Affinity DataIC50:  320nMAssay Description:Inhibitory activity against Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287250(4-(2-{3-[3-((R)-1-Methyl-2-oxo-5-phenyl-2,3-dihydr...)
Affinity DataIC50:  330nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50287251(CHEMBL262125 | N-[2-(2-Guanidino-thiazol-4-ylmethy...)
Affinity DataIC50:  330nMAssay Description:Inhibitory activity against Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287251(CHEMBL262125 | N-[2-(2-Guanidino-thiazol-4-ylmethy...)
Affinity DataIC50:  330nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287256(6-(2-{3-[3-((R)-1-Methyl-2-oxo-5-phenyl-2,3-dihydr...)
Affinity DataIC50:  340nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50287237(CHEMBL29888 | N-[2-(2-Guanidino-thiazol-4-ylmethyl...)
Affinity DataIC50:  350nMAssay Description:Inhibitory activity against Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287254(CHEMBL281082 | N-{[2-(2-Guanidino-thiazol-4-ylmeth...)
Affinity DataIC50:  370nMAssay Description:Inhibitory activity against gastrin receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287233(CHEMBL280980 | N-[2-(2-Guanidino-thiazol-4-ylmethy...)
Affinity DataIC50:  380nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287233(CHEMBL280980 | N-[2-(2-Guanidino-thiazol-4-ylmethy...)
Affinity DataIC50:  380nMAssay Description:Inhibitory activity against gastrin receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287259(CHEMBL286908 | N-[2-(2-Guanidino-thiazol-4-ylmethy...)
Affinity DataIC50:  390nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50287245(CHEMBL285586 | N-[2-(2-Guanidino-thiazol-4-ylmethy...)
Affinity DataIC50:  400nMAssay Description:Inhibitory activity against Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287244(2-[2-Oxo-5-phenyl-3-(3-m-tolyl-ureido)-2,3-dihydro...)
Affinity DataIC50:  430nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
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