Compile Data Set for Download or QSAR
maximum 50k data
Found 6 Enz. Inhib. hit(s) with all data for entry = 50029735
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50073850((S)-2-((S)-2-Benzyloxycarbonylamino-3-methyl-butyr...)
Affinity DataIC50:  17nMAssay Description:Inhibitory activity of compound against recombinant human Calpain 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287391((R)-4-Methyl-2-[2-oxo-2-(9H-xanthen-9-yl)-ethyl]-p...)
Affinity DataIC50:  25nMAssay Description:Inhibitory activity of compound against recombinant human Calpain 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287394((R)-2-Isobutyl-4-oxo-5,5-diphenyl-pentanoic acid (...)
Affinity DataIC50:  50nMAssay Description:Inhibitory activity of compound against recombinant human Calpain 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287392((R)-4-Methyl-2-[2-oxo-2-(9H-xanthen-9-yl)-ethyl]-p...)
Affinity DataIC50:  130nMAssay Description:Inhibitory activity of compound against recombinant human Calpain 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287390((R)-2-Isobutyl-4-oxo-8-phenyl-octanoic acid ((S)-1...)
Affinity DataIC50:  138nMAssay Description:Inhibitory activity of compound against recombinant human Calpain 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287393(CHEMBL296285 | [(S)-1-(1-Ethylaminooxalyl-propylca...)
Affinity DataIC50:  240nMAssay Description:Inhibitory activity of compound against recombinant human Calpain 1More data for this Ligand-Target Pair
In DepthDetails Article