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Found 7 Enz. Inhib. hit(s) with all data for entry = 50029847
TargetChymotrypsin-like protease CTRL-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50031442(1N-[4-amino(nitroimino)methylamino-1-(1-formyl-3-m...)
Affinity DataIC50:  2nMAssay Description:Compound was tested for inhibition of chymotrypsin-like protease of proteasome from postmortem human liver and brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetChymotrypsin-like protease CTRL-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50031440(1N-[4-amino(nitroimino)methylamino-1-(1-formyl-3-m...)
Affinity DataIC50:  6nMAssay Description:Compound was tested for inhibition of chymotrypsin-like protease of proteasome from postmortem human liver and brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetChymotrypsin-like protease CTRL-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288611(Alpha-ketocarbonyl boronic ester derivative | CHEM...)
Affinity DataIC50:  8nMAssay Description:Compound was tested for inhibition of chymotrypsin-like protease of proteasome from postmortem human liver and brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetChymotrypsin-like protease CTRL-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288609(Alpha-ketocarbonyl derivative | CHEMBL317337)
Affinity DataIC50:  22nMAssay Description:Compound was tested for inhibition of chymotrypsin-like protease of proteasome from postmortem human liver and brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetChymotrypsin-like protease CTRL-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288609(Alpha-ketocarbonyl derivative | CHEMBL317337)
Affinity DataIC50:  22nMAssay Description:Compound was tested for inhibition of chymotrypsin-like protease of proteasome from postmortem human liver and brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetChymotrypsin-like protease CTRL-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288610(Alpha-ketocarbonyl derivative | CHEMBL98937)
Affinity DataIC50: >1.00E+3nMAssay Description:Compound was tested for thromboxane TXA2 synthase inhibitory activity using human plateletMore data for this Ligand-Target Pair
In DepthDetails Article
TargetChymotrypsin-like protease CTRL-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288610(Alpha-ketocarbonyl derivative | CHEMBL98937)
Affinity DataIC50: >1.00E+3nMAssay Description:Compound was tested for inhibition of chymotrypsin-like protease of proteasome from postmortem human liver and brainMore data for this Ligand-Target Pair
In DepthDetails Article