Compile Data Set for Download or QSAR
maximum 50k data
Found 78 Enz. Inhib. hit(s) with all data for entry = 50029883
TargetSerine protease 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50063698(4-Guanidino-benzoic acid 6-carbamimidoyl-naphthale...)
Affinity DataIC50:  20nMAssay Description:Compound was evaluated for inhibitory activity against Trypsin.More data for this Ligand-Target Pair
In DepthDetails Article
TargetComplement C1s subcomponent(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50063698(4-Guanidino-benzoic acid 6-carbamimidoyl-naphthale...)
Affinity DataIC50:  140nMAssay Description:Compound was evaluated for inhibitory activity against C1s serine protease .More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlasminogen(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50063698(4-Guanidino-benzoic acid 6-carbamimidoyl-naphthale...)
Affinity DataIC50:  240nMAssay Description:Compound was evaluated for inhibitory activity against plasmin.More data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50063698(4-Guanidino-benzoic acid 6-carbamimidoyl-naphthale...)
Affinity DataIC50:  290nMAssay Description:Compound was evaluated for inhibitory activity against Thrombin.More data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50063703(2-(2-Iodo-phenyl)-benzo[d][1,3]oxazin-4-one | CHEM...)
Affinity DataIC50:  510nMAssay Description:Compound was evaluated for inhibitory activity against Thrombin.More data for this Ligand-Target Pair
In DepthDetails Article
TargetKallikrein-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50063698(4-Guanidino-benzoic acid 6-carbamimidoyl-naphthale...)
Affinity DataIC50:  650nMAssay Description:Compound was evaluated for inhibitory activity against Kallikrein.More data for this Ligand-Target Pair
In DepthDetails Article
TargetComplement C1r subcomponent(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289007(2-(2-Iodo-phenyl)-naphtho[2,3-d][1,3]oxazin-4-one ...)
Affinity DataIC50:  700nMAssay Description:Inhibition of C1r serine proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetComplement C1r subcomponent(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50063698(4-Guanidino-benzoic acid 6-carbamimidoyl-naphthale...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibitory activity against C1r serine proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetComplement C1r subcomponent(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50063698(4-Guanidino-benzoic acid 6-carbamimidoyl-naphthale...)
Affinity DataIC50:  1.04E+3nMAssay Description:Inhibitory activity against C1r serine proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetComplement C1s subcomponent(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50063703(2-(2-Iodo-phenyl)-benzo[d][1,3]oxazin-4-one | CHEM...)
Affinity DataIC50:  1.25E+3nMAssay Description:Compound was evaluated for inhibitory activity against C1s serine protease .More data for this Ligand-Target Pair
In DepthDetails Article
TargetComplement C1r subcomponent(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50063703(2-(2-Iodo-phenyl)-benzo[d][1,3]oxazin-4-one | CHEM...)
Affinity DataIC50:  1.37E+3nMAssay Description:Inhibitory activity against C1r serine proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetComplement C1r subcomponent(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50063703(2-(2-Iodo-phenyl)-benzo[d][1,3]oxazin-4-one | CHEM...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibitory activity against C1r serine proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetComplement C1r subcomponent(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288998(6,7-Dichloro-2-(2-iodo-phenyl)-benzo[d][1,3]oxazin...)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibitory activity against C1r serine proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetComplement C1r subcomponent(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289004(6-Chloro-2-(2-iodo-phenyl)-benzo[d][1,3]oxazin-4-o...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of C1r serine proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetComplement C1r subcomponent(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289016(5-Chloro-2-(2-iodo-phenyl)-benzo[d][1,3]oxazin-4-o...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibitory activity against C1r serine proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetComplement C1r subcomponent(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288996(2-(2-Trifluoromethyl-phenyl)-benzo[d][1,3]oxazin-4...)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibition of C1r serine proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetComplement C1r subcomponent(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289011(2-(2-Iodo-phenyl)-6-methoxy-benzo[d][1,3]oxazin-4-...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibitory activity against C1r serine proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetComplement C1r subcomponent(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289009(2-(2-Iodo-benzyl)-benzo[d][1,3]oxazin-4-one | CHEM...)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of C1r serine proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlasminogen(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50063703(2-(2-Iodo-phenyl)-benzo[d][1,3]oxazin-4-one | CHEM...)
Affinity DataIC50:  6.68E+3nMAssay Description:Compound was evaluated for inhibitory activity against plasmin.More data for this Ligand-Target Pair
In DepthDetails Article
TargetComplement C1r subcomponent(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288997(2-(2-Iodo-phenyl)-5-methyl-benzo[d][1,3]oxazin-4-o...)
Affinity DataIC50:  7.50E+3nMAssay Description:Inhibitory activity against C1r serine proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetComplement C1r subcomponent(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289004(6-Chloro-2-(2-iodo-phenyl)-benzo[d][1,3]oxazin-4-o...)
Affinity DataIC50:  7.80E+3nMAssay Description:Inhibitory activity against C1r serine proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetComplement C1r subcomponent(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289006(2-(2-Bromo-phenyl)-benzo[d][1,3]oxazin-4-one | 2-(...)
Affinity DataIC50:  9.50E+3nMAssay Description:Inhibitory activity against C1r serine proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKallikrein-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50063703(2-(2-Iodo-phenyl)-benzo[d][1,3]oxazin-4-one | CHEM...)
Affinity DataIC50:  9.89E+3nMAssay Description:Compound was evaluated for inhibitory activity against Kallikrein.More data for this Ligand-Target Pair
In DepthDetails Article
TargetComplement C1r subcomponent(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289008(2-(2-Iodo-phenyl)-6-methyl-benzo[d][1,3]oxazin-4-o...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of C1r serine proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetComplement C1r subcomponent(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50063698(4-Guanidino-benzoic acid 6-carbamimidoyl-naphthale...)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibitory activity against C1r serine proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetComplement C1r subcomponent(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50063698(4-Guanidino-benzoic acid 6-carbamimidoyl-naphthale...)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibitory activity against C1r serine proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetComplement C1r subcomponent(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289012(2-(2-Fluoro-phenyl)-benzo[d][1,3]oxazin-4-one | 2-...)
Affinity DataIC50:  1.21E+4nMAssay Description:Inhibitory activity against C1r serine proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetComplement C1r subcomponent(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289016(5-Chloro-2-(2-iodo-phenyl)-benzo[d][1,3]oxazin-4-o...)
Affinity DataIC50:  1.35E+4nMAssay Description:Inhibitory activity against C1r serine proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetComplement C1r subcomponent(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM33703(2-(2-Nitro-phenyl)-benzo[d][1,3]oxazin-4-one | 2-(...)
Affinity DataIC50:  1.50E+4nMAssay Description:Compound was evaluated for inhibitory activity against C1r serine protease in assay 1More data for this Ligand-Target Pair
In DepthDetails Article
TargetSerine protease 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50063703(2-(2-Iodo-phenyl)-benzo[d][1,3]oxazin-4-one | CHEM...)
Affinity DataIC50:  1.53E+4nMAssay Description:Compound was evaluated for inhibitory activity against Trypsin.More data for this Ligand-Target Pair
In DepthDetails Article
TargetComplement C1r subcomponent(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50063703(2-(2-Iodo-phenyl)-benzo[d][1,3]oxazin-4-one | CHEM...)
Affinity DataIC50:  1.67E+4nMAssay Description:Inhibitory activity against C1r serine proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetComplement C1r subcomponent(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289010(2-(2-Chloro-phenyl)-benzo[d][1,3]oxazin-4-one | CH...)
Affinity DataIC50:  1.73E+4nMAssay Description:Inhibition of C1r serine proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetComplement C1r subcomponent(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289000(2-(2-Methoxy-phenyl)-benzo[d][1,3]oxazin-4-one | 2...)
Affinity DataIC50:  1.77E+4nMAssay Description:Inhibition of C1r serine proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetComplement C1r subcomponent(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289017(2-(2-Iodo-phenyl)-7-nitro-benzo[d][1,3]oxazin-4-on...)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibitory activity against C1r serine proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetComplement C1r subcomponent(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289009(2-(2-Iodo-benzyl)-benzo[d][1,3]oxazin-4-one | CHEM...)
Affinity DataIC50:  2.60E+4nMAssay Description:Inhibitory activity against C1r serine proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetComplement C1r subcomponent(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289004(6-Chloro-2-(2-iodo-phenyl)-benzo[d][1,3]oxazin-4-o...)
Affinity DataIC50:  2.73E+4nMAssay Description:Inhibition of C1r serine proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetComplement C1r subcomponent(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289006(2-(2-Bromo-phenyl)-benzo[d][1,3]oxazin-4-one | 2-(...)
Affinity DataIC50:  3.20E+4nMAssay Description:Inhibitory activity against C1r serine proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetComplement C1r subcomponent(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288996(2-(2-Trifluoromethyl-phenyl)-benzo[d][1,3]oxazin-4...)
Affinity DataIC50:  3.54E+4nMAssay Description:Inhibitory activity against C1r serine proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetComplement C1r subcomponent(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM33703(2-(2-Nitro-phenyl)-benzo[d][1,3]oxazin-4-one | 2-(...)
Affinity DataIC50:  3.63E+4nMAssay Description:Inhibition of C1r serine proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetComplement C1r subcomponent(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289009(2-(2-Iodo-benzyl)-benzo[d][1,3]oxazin-4-one | CHEM...)
Affinity DataIC50:  4.00E+4nMAssay Description:Inhibitory activity against C1r serine proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetComplement C1r subcomponent(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289010(2-(2-Chloro-phenyl)-benzo[d][1,3]oxazin-4-one | CH...)
Affinity DataIC50:  4.50E+4nMAssay Description:Inhibitory activity against C1r serine proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetComplement C1r subcomponent(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289006(2-(2-Bromo-phenyl)-benzo[d][1,3]oxazin-4-one | 2-(...)
Affinity DataIC50:  4.60E+4nMAssay Description:Compound was evaluated for inhibitory activity against C1r serine protease in assay 2 at t=60 min.More data for this Ligand-Target Pair
In DepthDetails Article
TargetComplement C1r subcomponent(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50063703(2-(2-Iodo-phenyl)-benzo[d][1,3]oxazin-4-one | CHEM...)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibitory activity against C1r serine proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetComplement C1r subcomponent(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289008(2-(2-Iodo-phenyl)-6-methyl-benzo[d][1,3]oxazin-4-o...)
Affinity DataIC50:  5.10E+4nMAssay Description:Inhibitory activity against C1r serine proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetComplement C1r subcomponent(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289016(5-Chloro-2-(2-iodo-phenyl)-benzo[d][1,3]oxazin-4-o...)
Affinity DataIC50:  5.70E+4nMAssay Description:Compound was evaluated for percentage inhibitory activity against C1r serine protease in assay 1.More data for this Ligand-Target Pair
In DepthDetails Article
TargetComplement C1r subcomponent(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289010(2-(2-Chloro-phenyl)-benzo[d][1,3]oxazin-4-one | CH...)
Affinity DataIC50: >6.25E+4nMAssay Description:Inhibition of C1r serine proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetComplement C1r subcomponent(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289017(2-(2-Iodo-phenyl)-7-nitro-benzo[d][1,3]oxazin-4-on...)
Affinity DataIC50: >6.25E+4nMAssay Description:Inhibitory activity against C1r serine proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetComplement C1r subcomponent(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289013(2-(3-Iodo-phenyl)-benzo[d][1,3]oxazin-4-one | CHEM...)
Affinity DataIC50: >6.25E+4nMAssay Description:Inhibitory activity against C1r serine proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetComplement C1r subcomponent(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289005(2-(2-Hydroxy-phenyl)-benzo[d][1,3]oxazin-4-one | C...)
Affinity DataIC50: >6.25E+4nMAssay Description:Inhibitory activity against C1r serine proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetComplement C1r subcomponent(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288999(2-(2-Iodo-phenyl)-7-methyl-benzo[d][1,3]oxazin-4-o...)
Affinity DataIC50: >6.25E+4nMAssay Description:Inhibitory activity against C1r serine proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
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