Compile Data Set for Download or QSAR
maximum 50k data
Found 21 Enz. Inhib. hit(s) with all data for entry = 50029929
LigandPNGBDBM50083595(3-[3-((R)-2-Amino-3-mercapto-propylamino)-phenoxy]...)
Affinity DataIC50:  250nMAssay Description:Inhibition of the Farnesyltransferase catalyzed incorporation of [3H]-FPP into recombinant Ha-Ras by 50% in bovine brain at a concentration of ca. 1 ...More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289417((R)-2-Amino-3-(3-m-tolyloxy-phenylamino)-propane-1...)
Affinity DataIC50:  330nMAssay Description:Inhibition of the Farnesyltransferase catalyzed incorporation of [3H]-FPP into recombinant Ha-Ras by 50% in bovine brain at a concentration of ca. 1 ...More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289422(CHEMBL26314 | {3-[4-((R)-2-Amino-3-mercapto-propyl...)
Affinity DataIC50:  335nMAssay Description:Inhibition of the Farnesyltransferase catalyzed incorporation of [3H]-FPP into recombinant Ha-Ras by 50% in bovine brain at a concentration of ca. 1 ...More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289429(3-[4-((R)-2-Amino-3-mercapto-propylamino)-phenoxy]...)
Affinity DataIC50:  403nMAssay Description:Inhibition of the Farnesyltransferase catalyzed incorporation of [3H]-FPP into recombinant Ha-Ras by 50% in bovine brain at a concentration of ca. 1 ...More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289427((R)-2-Amino-3-(4-phenoxy-phenylamino)-propane-1-th...)
Affinity DataIC50:  460nMAssay Description:Inhibition of the Farnesyltransferase catalyzed incorporation of [3H]-FPP into recombinant Ha-Ras by 50% in bovine brain at a concentration of ca. 1 ...More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289420((R)-2-Amino-3-(4-m-tolyloxy-phenylamino)-propane-1...)
Affinity DataIC50:  615nMAssay Description:Inhibition of the Farnesyltransferase catalyzed incorporation of [3H]-FPP into recombinant Ha-Ras by 50% in bovine brain at a concentration of ca. 1 ...More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289425(3-[4-((R)-2-Amino-3-mercapto-propylamino)-phenoxy]...)
Affinity DataIC50:  650nMAssay Description:Inhibition of the Farnesyltransferase catalyzed incorporation of [3H]-FPP into recombinant Ha-Ras by 50% in bovine brain at a concentration of ca. 1 ...More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289431((R)-2-Amino-3-(3-phenoxy-phenylamino)-propane-1-th...)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of the Farnesyltransferase catalyzed incorporation of [3H]-FPP into recombinant Ha-Ras by 50% in bovine brain at a concentration of ca. 1 ...More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289425(3-[4-((R)-2-Amino-3-mercapto-propylamino)-phenoxy]...)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of Geranylgeranyl transferase type I, an enzyme that recognizes CaaX sequences containing leucine as the terminal residue.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289423(4-[4-((R)-2-Amino-3-mercapto-propylamino)-phenoxy]...)
Affinity DataIC50:  3.15E+3nMAssay Description:Inhibition of the Farnesyltransferase catalyzed incorporation of [3H]-FPP into recombinant Ha-Ras by 50% in bovine brain at a concentration of ca. 1 ...More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289428(4-[3-((R)-2-Amino-3-mercapto-propylamino)-phenoxy]...)
Affinity DataIC50:  3.80E+3nMAssay Description:Inhibition of the Farnesyltransferase catalyzed incorporation of [3H]-FPP into recombinant Ha-Ras by 50% in bovine brain at a concentration of ca. 1 ...More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289427((R)-2-Amino-3-(4-phenoxy-phenylamino)-propane-1-th...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of the Farnesyltransferase catalyzed incorporation of [3H]-FPP into recombinant Ha-Ras by 50% in bovine brain at a concentration of ca. 1 ...More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50083595(3-[3-((R)-2-Amino-3-mercapto-propylamino)-phenoxy]...)
Affinity DataIC50:  5.80E+3nMAssay Description:Inhibition of Geranylgeranyl transferase type I, an enzyme that recognizes CaaX sequences containing leucine as the terminal residue.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289426(3-[3-((R)-2-Amino-3-mercapto-propionylamino)-pheno...)
Affinity DataIC50:  6.90E+3nMAssay Description:Inhibition of the Farnesyltransferase catalyzed incorporation of [3H]-FPP into recombinant Ha-Ras by 50% in bovine brain at a concentration of ca. 1 ...More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289421(3-[4-((R)-2-Amino-3-mercapto-propionylamino)-pheno...)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of the Farnesyltransferase catalyzed incorporation of [3H]-FPP into recombinant Ha-Ras by 50% in bovine brain at a concentration of ca. 1 ...More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289424(4-[4-((R)-2-Amino-3-mercapto-propionylamino)-pheno...)
Affinity DataIC50:  3.90E+4nMAssay Description:Inhibition of Geranylgeranyl transferase type I, an enzyme that recognizes CaaX sequences containing leucine as the terminal residue.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289419(3-[3-((R)-2-Amino-3-mercapto-propionylamino)-pheno...)
Affinity DataIC50:  4.50E+4nMAssay Description:Inhibition of the Farnesyltransferase catalyzed incorporation of [3H]-FPP into recombinant Ha-Ras by 50% in bovine brain at a concentration of ca. 1 ...More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289416(3-[4-((R)-2-Amino-3-mercapto-propionylamino)-pheno...)
Affinity DataIC50:  4.50E+4nMAssay Description:Inhibition of the Farnesyltransferase catalyzed incorporation of [3H]-FPP into recombinant Ha-Ras by 50% in bovine brain at a concentration of ca. 1 ...More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289430(4-[4-((R)-2-Amino-3-mercapto-propionylamino)-pheno...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of the Farnesyltransferase catalyzed incorporation of [3H]-FPP into recombinant Ha-Ras by 50% in bovine brain at a concentration of ca. 1 ...More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289432(4-[3-((R)-2-Amino-3-mercapto-propionylamino)-pheno...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of the Farnesyltransferase catalyzed incorporation of [3H]-FPP into recombinant Ha-Ras by 50% in bovine brain at a concentration of ca. 1 ...More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289418(4-[3-((R)-2-Amino-3-mercapto-propionylamino)-pheno...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of the Farnesyltransferase catalyzed incorporation of [3H]-FPP into recombinant Ha-Ras by 50% in bovine brain at a concentration of ca. 1 ...More data for this Ligand-Target Pair
In DepthDetails Article