Compile Data Set for Download or QSAR
maximum 50k data
Found 38 Enz. Inhib. hit(s) with all data for entry = 50029975
LigandPNGBDBM50449787(CHEMBL2062154 | PD-134308)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of binding of [125I]- Bolton-Hunter labeled CCK-8 to CCK-B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289877(CHEMBL62832 | [(S)-1-((1R,2R)-2-Hydroxy-1-hydroxym...)
Affinity DataIC50:  6.10nMAssay Description:Inhibition of binding of [125I]- Bolton-Hunter labeled CCK-8 to CCK-B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289871(CHEMBL262456 | N-{(R)-2-[2-(Adamantan-2-yloxycarbo...)
Affinity DataIC50:  8.20nMAssay Description:Inhibition of binding of [125I]- Bolton-Hunter labeled CCK-8 to CCK-B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289879(CHEMBL62205 | [(S)-2-(1H-Indol-3-yl)-1-methyl-1-ph...)
Affinity DataIC50:  32nMAssay Description:Inhibition of binding of [125I]- Bolton-Hunter labeled CCK-8 to CCK-B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289876(CHEMBL292194 | N-{(R)-2-[(R)-2-(Adamantan-2-yloxyc...)
Affinity DataIC50:  58nMAssay Description:Inhibition of binding of [125I]- Bolton-Hunter labeled CCK-8 to CCK-B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50289886(CHEMBL302194 | [2-(2-Dimethylcarbamoyl-benzofuran-...)
Affinity DataIC50:  65nMAssay Description:Inhibition of binding of [125I]- Bolton-Hunter labeled CCK-8 to CCK-A receptor in the rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289887(CHEMBL418464 | [1-((1R,2R)-2-Hydroxy-1-hydroxymeth...)
Affinity DataIC50:  68nMAssay Description:Inhibition of binding of [125I]- Bolton-Hunter labeled CCK-8 to CCK-B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289886(CHEMBL302194 | [2-(2-Dimethylcarbamoyl-benzofuran-...)
Affinity DataIC50:  125nMAssay Description:Inhibition of binding of [125I]- Bolton-Hunter labeled CCK-8 to CCK-B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289870(CHEMBL417412 | N-{2-[2-(Adamantan-2-yloxycarbonyla...)
Affinity DataIC50:  129nMAssay Description:Inhibition of binding of [125I]- Bolton-Hunter labeled CCK-8 to CCK-B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289872(CHEMBL60386 | [1-((1R,2R)-2-Hydroxy-1-hydroxymethy...)
Affinity DataIC50:  141nMAssay Description:Inhibition of binding of [125I]- Bolton-Hunter labeled CCK-8 to CCK-B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289888(CHEMBL292957 | [2-(2-Dimethylaminomethyl-benzofura...)
Affinity DataIC50:  171nMAssay Description:Inhibition of binding of [125I]- Bolton-Hunter labeled CCK-8 to CCK-B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289884(CHEMBL64770 | [1-((1R,2R)-2-Hydroxy-1-hydroxymethy...)
Affinity DataIC50:  200nMAssay Description:Inhibition of binding of [125I]- Bolton-Hunter labeled CCK-8 to CCK-B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50289873(CHEMBL64155 | N-{(R)-2-[2-(Adamantan-2-yloxycarbon...)
Affinity DataIC50:  583nMAssay Description:Inhibition of binding of [125I]- Bolton-Hunter labeled CCK-8 to CCK-A receptor in the rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50289872(CHEMBL60386 | [1-((1R,2R)-2-Hydroxy-1-hydroxymethy...)
Affinity DataIC50:  616nMAssay Description:Inhibition of binding of [125I]- Bolton-Hunter labeled CCK-8 to CCK-A receptor in the rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50289879(CHEMBL62205 | [(S)-2-(1H-Indol-3-yl)-1-methyl-1-ph...)
Affinity DataIC50:  650nMAssay Description:Inhibition of binding of [125I]- Bolton-Hunter labeled CCK-8 to CCK-A receptor in the rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50289877(CHEMBL62832 | [(S)-1-((1R,2R)-2-Hydroxy-1-hydroxym...)
Affinity DataIC50:  681nMAssay Description:Inhibition of binding of [125I]- Bolton-Hunter labeled CCK-8 to CCK-A receptor in the rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289880(CHEMBL303020 | N-{(R)-2-[2-(Adamantan-2-yloxycarbo...)
Affinity DataIC50:  693nMAssay Description:Inhibition of binding of [125I]- Bolton-Hunter labeled CCK-8 to CCK-B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289883(CHEMBL292422 | [2-(2-Acetylamino-thiazol-4-yl)-1-m...)
Affinity DataIC50:  877nMAssay Description:Inhibition of binding of [125I]- Bolton-Hunter labeled CCK-8 to CCK-B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50289874(CHEMBL434020 | N-(2-{[2-(Adamantan-2-yloxycarbonyl...)
Affinity DataIC50:  1.35E+3nMAssay Description:Inhibition of binding of [125I]- Bolton-Hunter labeled CCK-8 to CCK-A receptor in the rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289878(CHEMBL293178 | [1-((1R,2R)-2-Hydroxy-1-hydroxymeth...)
Affinity DataIC50:  1.54E+3nMAssay Description:Inhibition of binding of [125I]- Bolton-Hunter labeled CCK-8 to CCK-B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289878(CHEMBL293178 | [1-((1R,2R)-2-Hydroxy-1-hydroxymeth...)
Affinity DataIC50:  1.54E+3nMAssay Description:Inhibition of binding of [125I]- Bolton-Hunter labeled CCK-8 to CCK-B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289881(CHEMBL59985 | [1-Methyl-1-phenethylcarbamoyl-2-(5,...)
Affinity DataIC50:  1.56E+3nMAssay Description:Inhibition of binding of [125I]- Bolton-Hunter labeled CCK-8 to CCK-B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50289880(CHEMBL303020 | N-{(R)-2-[2-(Adamantan-2-yloxycarbo...)
Affinity DataIC50:  1.91E+3nMAssay Description:Inhibition of binding of [125I]- Bolton-Hunter labeled CCK-8 to CCK-A receptor in the rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289874(CHEMBL434020 | N-(2-{[2-(Adamantan-2-yloxycarbonyl...)
Affinity DataIC50:  1.91E+3nMAssay Description:Inhibition of binding of [125I]- Bolton-Hunter labeled CCK-8 to CCK-B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289882((2-Benzotriazol-1-yl-1-methyl-1-phenethylcarbamoyl...)
Affinity DataIC50:  2.17E+3nMAssay Description:Inhibition of binding of [125I]- Bolton-Hunter labeled CCK-8 to CCK-B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50289871(CHEMBL262456 | N-{(R)-2-[2-(Adamantan-2-yloxycarbo...)
Affinity DataIC50:  2.19E+3nMAssay Description:Inhibition of binding of [125I]- Bolton-Hunter labeled CCK-8 to CCK-A receptor in the rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289889(CHEMBL64623 | [2-(3,5-Dimethyl-isoxazol-4-yl)-1-me...)
Affinity DataIC50:  2.28E+3nMAssay Description:Inhibition of binding of [125I]- Bolton-Hunter labeled CCK-8 to CCK-B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50289870(CHEMBL417412 | N-{2-[2-(Adamantan-2-yloxycarbonyla...)
Affinity DataIC50:  2.65E+3nMAssay Description:Inhibition of binding of [125I]- Bolton-Hunter labeled CCK-8 to CCK-A receptor in the rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289873(CHEMBL64155 | N-{(R)-2-[2-(Adamantan-2-yloxycarbon...)
Affinity DataIC50:  2.82E+3nMAssay Description:Inhibition of binding of [125I]- Bolton-Hunter labeled CCK-8 to CCK-B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50289876(CHEMBL292194 | N-{(R)-2-[(R)-2-(Adamantan-2-yloxyc...)
Affinity DataIC50:  2.86E+3nMAssay Description:Inhibition of binding of [125I]- Bolton-Hunter labeled CCK-8 to CCK-A receptor in the rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50289882((2-Benzotriazol-1-yl-1-methyl-1-phenethylcarbamoyl...)
Affinity DataIC50:  3.62E+3nMAssay Description:Inhibition of binding of [125I]- Bolton-Hunter labeled CCK-8 to CCK-A receptor in the rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50449787(CHEMBL2062154 | PD-134308)
Affinity DataIC50:  4.30E+3nMAssay Description:Inhibition of binding of [125I]- Bolton-Hunter labeled CCK-8 to CCK-A receptor in the rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50289883(CHEMBL292422 | [2-(2-Acetylamino-thiazol-4-yl)-1-m...)
Affinity DataIC50:  5.35E+3nMAssay Description:Inhibition of binding of [125I]- Bolton-Hunter labeled CCK-8 to CCK-A receptor in the rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289875((1-Phenethylcarbamoyl-3-spiro[cyclobutane-1,2'-(2'...)
Affinity DataIC50:  6.78E+3nMAssay Description:Inhibition of binding of [125I]- Bolton-Hunter labeled CCK-8 to CCK-B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50289889(CHEMBL64623 | [2-(3,5-Dimethyl-isoxazol-4-yl)-1-me...)
Affinity DataIC50:  6.94E+3nMAssay Description:Inhibition of binding of [125I]- Bolton-Hunter labeled CCK-8 to CCK-A receptor in the rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50289875((1-Phenethylcarbamoyl-3-spiro[cyclobutane-1,2'-(2'...)
Affinity DataIC50:  7.22E+3nMAssay Description:Inhibition of binding of [125I]- Bolton-Hunter labeled CCK-8 to CCK-A receptor in the rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50289881(CHEMBL59985 | [1-Methyl-1-phenethylcarbamoyl-2-(5,...)
Affinity DataIC50:  1.98E+4nMAssay Description:Inhibition of binding of [125I]- Bolton-Hunter labeled CCK-8 to CCK-A receptor in the rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289885((2-Phenethylcarbamoyl-indan-2-yl)-carbamic acid ad...)
Affinity DataIC50:  2.04E+4nMAssay Description:Inhibition of binding of [125I]- Bolton-Hunter labeled CCK-8 to CCK-B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails Article