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Report error Found 32 Enz. Inhib. hit(s) with all data for entry = 50030049
TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290631((6,7-Dimethoxy-quinazolin-4-yl)-isoquinolin-4-yl-a...)
Affinity DataIC50:  6.40nMAssay Description:Tested for inhibition of Epidermal growth factor receptor from A431 vulval squamous carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM4626(Anilinoquinazoline deriv. 9 | CHEMBL301018 | N-(3-...)
Affinity DataIC50:  9nMAssay Description:Inhibition of EGF-stimulated proliferation of KB cells in cultureMore data for this Ligand-Target Pair
In DepthDetails Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290640((6,7-Dimethoxy-quinazolin-4-yl)-(2-phenyl-cyclopro...)
Affinity DataIC50:  10nMAssay Description:Tested for inhibition of Epidermal growth factor receptor from A431 vulval squamous carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM4626(Anilinoquinazoline deriv. 9 | CHEMBL301018 | N-(3-...)
Affinity DataIC50:  80nMAssay Description:Inhibition of EGF-stimulated proliferation of KB cells in cultureMore data for this Ligand-Target Pair
In DepthDetails Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290632(Acetic acid 7-methoxy-4-(2-phenyl-cyclopropylamino...)
Affinity DataIC50:  84nMAssay Description:Tested for inhibition of Epidermal growth factor receptor from A431 vulval squamous carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290640((6,7-Dimethoxy-quinazolin-4-yl)-(2-phenyl-cyclopro...)
Affinity DataIC50:  140nMAssay Description:Tested for inhibition of Epidermal growth factor receptor from A431 vulval squamous carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290641((6,7-Dimethoxy-quinazolin-4-yl)-(3-methyl-benzyl)-...)
Affinity DataIC50:  170nMAssay Description:Tested for inhibition of Epidermal growth factor receptor from A431 vulval squamous carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290637((6,7-Dimethoxy-quinazolin-4-yl)-isoquinolin-1-yl-a...)
Affinity DataIC50:  200nMAssay Description:Tested for inhibition of Epidermal growth factor receptor from A431 vulval squamous carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290642(CHEMBL420059 | [7-Methoxy-6-(2-morpholin-4-yl-etho...)
Affinity DataIC50:  300nMAssay Description:Tested for inhibition of Epidermal growth factor receptor from A431 vulval squamous carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290638(CHEMBL91484 | [6-(3-Dimethylamino-propoxy)-7-metho...)
Affinity DataIC50:  310nMAssay Description:Inhibition of EGF-stimulated proliferation of KB cells in cultureMore data for this Ligand-Target Pair
In DepthDetails Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290638(CHEMBL91484 | [6-(3-Dimethylamino-propoxy)-7-metho...)
Affinity DataIC50:  310nMAssay Description:Inhibition of EGF-stimulated proliferation of KB cells in cultureMore data for this Ligand-Target Pair
In DepthDetails Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290631((6,7-Dimethoxy-quinazolin-4-yl)-isoquinolin-4-yl-a...)
Affinity DataIC50:  360nMAssay Description:Inhibition of EGF-stimulated proliferation of KB cells in cultureMore data for this Ligand-Target Pair
In DepthDetails Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290643(7-Methoxy-4-(2-phenyl-cyclopropylamino)-quinazolin...)
Affinity DataIC50:  390nMAssay Description:Tested for inhibition of Epidermal growth factor receptor from A431 vulval squamous carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290635(CHEMBL422066 | N-(3-Chloro-4-fluoro-phenyl)-N'-(6,...)
Affinity DataIC50:  430nMAssay Description:Tested for inhibition of Epidermal growth factor receptor from A431 vulval squamous carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290642(CHEMBL420059 | [7-Methoxy-6-(2-morpholin-4-yl-etho...)
Affinity DataIC50:  570nMAssay Description:Inhibition of EGF-stimulated proliferation of KB cells in cultureMore data for this Ligand-Target Pair
In DepthDetails Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290634((6,7-Dimethoxy-quinazolin-4-yl)-isoquinolin-3-yl-a...)
Affinity DataIC50:  660nMAssay Description:Tested for inhibition of Epidermal growth factor receptor from A431 vulval squamous carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290630((3-Chloro-4-fluoro-phenyl)-(6,7-dimethoxy-quinazol...)
Affinity DataIC50:  730nMAssay Description:Tested for inhibition of Epidermal growth factor receptor from A431 vulval squamous carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290635(CHEMBL422066 | N-(3-Chloro-4-fluoro-phenyl)-N'-(6,...)
Affinity DataIC50:  780nMAssay Description:Inhibition of EGF-stimulated proliferation of KB cells in cultureMore data for this Ligand-Target Pair
In DepthDetails Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290644((6,7-Dimethoxy-quinazolin-4-yl)-quinoxalin-2-yl-am...)
Affinity DataIC50:  780nMAssay Description:Tested for inhibition of Epidermal growth factor receptor from A431 vulval squamous carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290634((6,7-Dimethoxy-quinazolin-4-yl)-isoquinolin-3-yl-a...)
Affinity DataIC50:  810nMAssay Description:Inhibition of EGF-stimulated proliferation of KB cells in cultureMore data for this Ligand-Target Pair
In DepthDetails Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290633(4-(2,3-Dihydro-indol-1-yl)-6,7-dimethoxy-quinazoli...)
Affinity DataIC50:  820nMAssay Description:Tested for inhibition of Epidermal growth factor receptor from A431 vulval squamous carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290639(Benzo[1,2,4]triazin-3-yl-(6,7-dimethoxy-quinazolin...)
Affinity DataIC50:  820nMAssay Description:Tested for inhibition of Epidermal growth factor receptor from A431 vulval squamous carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290641((6,7-Dimethoxy-quinazolin-4-yl)-(3-methyl-benzyl)-...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of EGF-stimulated proliferation of KB cells in cultureMore data for this Ligand-Target Pair
In DepthDetails Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290636((6,7-Dimethoxy-quinazolin-4-yl)-indan-1-yl-amine |...)
Affinity DataIC50:  1.73E+3nMAssay Description:Inhibition of EGF-stimulated proliferation of KB cells in cultureMore data for this Ligand-Target Pair
In DepthDetails Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290636((6,7-Dimethoxy-quinazolin-4-yl)-indan-1-yl-amine |...)
Affinity DataIC50:  1.73E+3nMAssay Description:Inhibition of EGF-stimulated proliferation of KB cells in cultureMore data for this Ligand-Target Pair
In DepthDetails Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290637((6,7-Dimethoxy-quinazolin-4-yl)-isoquinolin-1-yl-a...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of EGF-stimulated proliferation of KB cells in cultureMore data for this Ligand-Target Pair
In DepthDetails Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290630((3-Chloro-4-fluoro-phenyl)-(6,7-dimethoxy-quinazol...)
Affinity DataIC50:  3.93E+3nMAssay Description:Tested for inhibition of Epidermal growth factor receptor from A431 vulval squamous carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290633(4-(2,3-Dihydro-indol-1-yl)-6,7-dimethoxy-quinazoli...)
Affinity DataIC50:  4.10E+3nMAssay Description:Inhibition of EGF-stimulated proliferation of KB cells in cultureMore data for this Ligand-Target Pair
In DepthDetails Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290632(Acetic acid 7-methoxy-4-(2-phenyl-cyclopropylamino...)
Affinity DataIC50:  1.14E+4nMAssay Description:Tested for inhibition of Epidermal growth factor receptor from A431 vulval squamous carcinoma cellsMore data for this Ligand-Target Pair
In DepthDetails Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290644((6,7-Dimethoxy-quinazolin-4-yl)-quinoxalin-2-yl-am...)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of EGF-stimulated proliferation of KB cells in cultureMore data for this Ligand-Target Pair
In DepthDetails Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290643(7-Methoxy-4-(2-phenyl-cyclopropylamino)-quinazolin...)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of EGF-stimulated proliferation of KB cells in cultureMore data for this Ligand-Target Pair
In DepthDetails Article

TargetEpidermal growth factor receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290639(Benzo[1,2,4]triazin-3-yl-(6,7-dimethoxy-quinazolin...)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of EGF-stimulated proliferation of KB cells in cultureMore data for this Ligand-Target Pair
In DepthDetails Article