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Found 48 Enz. Inhib. hit(s) with all data for entry = 50030060
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50001859((buspirone) 8-[4-(4-Pyrimidin-2-yl-piperazin-1-yl)...)
Affinity DataIC50:  7.10nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor using receptor binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM21393(7-(dipropylamino)-5,6,7,8-tetrahydronaphthalen-1-o...)
Affinity DataIC50:  8.10nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor using receptor binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50290762(9-{4-[2-(2-Methoxy-phenoxy)-ethylamino]-butyryl}-3...)
Affinity DataIC50:  9.20nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor using receptor binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50290748(9-{3-[2-(2-Methoxy-phenoxy)-ethylamino]-propionyl}...)
Affinity DataIC50:  11nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor using receptor binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50290750(9-{4-[2-(2-Methoxy-phenoxy)-ethylamino]-butyryl}-3...)
Affinity DataIC50:  18nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor using receptor binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50290760(9-{3-[2-(2-Methoxy-phenoxy)-ethylamino]-propionyl}...)
Affinity DataIC50:  20nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor using receptor binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50290757(CHEMBL318260 | N-(5-Ethylsulfanyl-1-methyl-6-oxo-1...)
Affinity DataIC50:  33nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor using receptor binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50290770(9-{2-[2-(2-Methoxy-phenoxy)-ethylamino]-acetyl}-3-...)
Affinity DataIC50:  37nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor using receptor binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50290759(9-{2-[(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-am...)
Affinity DataIC50:  45nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor using receptor binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50290769(9-(3-{4-[2-Hydroxy-3-(3-methoxy-phenoxy)-propyl]-p...)
Affinity DataIC50:  118nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor using receptor binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50290763(9-(3-{[2-(2-Methoxy-phenoxy)-ethyl]-methyl-amino}-...)
Affinity DataIC50:  134nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor using receptor binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50290758(3-Methyl-9-[3-(2-phenoxy-ethylamino)-propionyl]-6,...)
Affinity DataIC50:  150nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor using receptor binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50290766(9-{2-[2-(2-Methoxy-phenoxy)-ethylamino]-acetyl}-3-...)
Affinity DataIC50:  163nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor using receptor binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50290767(9-{3-[2-(3-Chloro-phenoxy)-ethylamino]-propionyl}-...)
Affinity DataIC50:  181nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor using receptor binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50290756(3-Methyl-9-[2-(2-phenoxy-ethylamino)-acetyl]-6,7,8...)
Affinity DataIC50:  230nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor using receptor binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50290748(9-{3-[2-(2-Methoxy-phenoxy)-ethylamino]-propionyl}...)
Affinity DataIC50:  270nMAssay Description:Binding affinity towards Alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50290747(9-{2-[(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-am...)
Affinity DataIC50:  299nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor using receptor binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50290752(9-{3-[2-(3-Chloro-phenoxy)-ethylamino]-propionyl}-...)
Affinity DataIC50:  312nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor using receptor binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50290749(3-Methyl-9-[3-(2-phenoxy-ethylamino)-propionyl]-6,...)
Affinity DataIC50:  524nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor using receptor binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50290749(3-Methyl-9-[3-(2-phenoxy-ethylamino)-propionyl]-6,...)
Affinity DataIC50:  540nMAssay Description:Binding affinity towards Alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50290750(9-{4-[2-(2-Methoxy-phenoxy)-ethylamino]-butyryl}-3...)
Affinity DataIC50:  690nMAssay Description:Binding affinity towards Alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50290762(9-{4-[2-(2-Methoxy-phenoxy)-ethylamino]-butyryl}-3...)
Affinity DataIC50:  860nMAssay Description:Binding affinity towards Alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50290762(9-{4-[2-(2-Methoxy-phenoxy)-ethylamino]-butyryl}-3...)
Affinity DataIC50:  930nMAssay Description:Binding affinity towards Alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50290751(9-{2-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-acetyl}...)
Affinity DataIC50: >1.00E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor using receptor binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50290761(9-(3-{4-[2-Hydroxy-3-(2-methoxy-phenoxy)-propyl]-p...)
Affinity DataIC50: >1.00E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor using receptor binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50290768(9-{2-[2-(2-Methoxy-phenoxy)-ethylamino]-propionyl}...)
Affinity DataIC50: >1.00E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor using receptor binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50290765(9-(3-{Benzyl-[2-(2-methoxy-phenoxy)-ethyl]-amino}-...)
Affinity DataIC50: >1.00E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor using receptor binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50290764(9-(2-{4-[2-Hydroxy-3-(2-methoxy-phenoxy)-propyl]-p...)
Affinity DataIC50: >1.00E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor using receptor binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50290753(9-(3-{[2-(2-Methoxy-phenoxy)-ethyl]-methyl-amino}-...)
Affinity DataIC50: >1.00E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor using receptor binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50290755(9-{2-[2-(2-Methoxy-phenoxy)-ethylamino]-propionyl}...)
Affinity DataIC50: >1.00E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor using receptor binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50290754(9-(3-{Benzyl-[2-(2-methoxy-phenoxy)-ethyl]-amino}-...)
Affinity DataIC50:  1.00E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor using receptor binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50290748(9-{3-[2-(2-Methoxy-phenoxy)-ethylamino]-propionyl}...)
Affinity DataIC50:  1.70E+3nMAssay Description:Binding affinity towards Alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50290760(9-{3-[2-(2-Methoxy-phenoxy)-ethylamino]-propionyl}...)
Affinity DataIC50:  1.70E+3nMAssay Description:Binding affinity towards Alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50290760(9-{3-[2-(2-Methoxy-phenoxy)-ethylamino]-propionyl}...)
Affinity DataIC50:  1.80E+3nMAssay Description:Binding affinity towards Alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50290759(9-{2-[(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-am...)
Affinity DataIC50:  2.33E+3nMAssay Description:Binding affinity towards Alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50290770(9-{2-[2-(2-Methoxy-phenoxy)-ethylamino]-acetyl}-3-...)
Affinity DataIC50:  3.10E+3nMAssay Description:Binding affinity towards Alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50290750(9-{4-[2-(2-Methoxy-phenoxy)-ethylamino]-butyryl}-3...)
Affinity DataIC50:  3.90E+3nMAssay Description:Binding affinity towards Alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50290747(9-{2-[(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-am...)
Affinity DataIC50:  4.60E+3nMAssay Description:Binding affinity towards Alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50290749(3-Methyl-9-[3-(2-phenoxy-ethylamino)-propionyl]-6,...)
Affinity DataIC50:  8.90E+3nMAssay Description:Binding affinity towards Alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50290763(9-(3-{[2-(2-Methoxy-phenoxy)-ethyl]-methyl-amino}-...)
Affinity DataIC50:  9.50E+3nMAssay Description:Binding affinity towards Alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50290747(9-{2-[(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-am...)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity towards Alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50290770(9-{2-[2-(2-Methoxy-phenoxy)-ethylamino]-acetyl}-3-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity towards Alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50290761(9-(3-{4-[2-Hydroxy-3-(2-methoxy-phenoxy)-propyl]-p...)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity towards Alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50290766(9-{2-[2-(2-Methoxy-phenoxy)-ethylamino]-acetyl}-3-...)
Affinity DataIC50:  1.25E+4nMAssay Description:Binding affinity towards Alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50290763(9-(3-{[2-(2-Methoxy-phenoxy)-ethyl]-methyl-amino}-...)
Affinity DataIC50:  1.61E+4nMAssay Description:Binding affinity towards Alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50290759(9-{2-[(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-am...)
Affinity DataIC50:  1.90E+4nMAssay Description:Binding affinity towards Alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50290766(9-{2-[2-(2-Methoxy-phenoxy)-ethylamino]-acetyl}-3-...)
Affinity DataIC50:  2.10E+4nMAssay Description:Binding affinity towards Alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50290761(9-(3-{4-[2-Hydroxy-3-(2-methoxy-phenoxy)-propyl]-p...)
Affinity DataIC50:  4.70E+4nMAssay Description:Binding affinity towards Alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails Article